NO329386B1 - Glukocorticoid-mimetica, farmasoytiske preparater og anvendelser for fremstilling av medikamenterfor behandling av sykdom - Google Patents

Glukocorticoid-mimetica, farmasoytiske preparater og anvendelser for fremstilling av medikamenterfor behandling av sykdom Download PDF

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Publication number
NO329386B1
NO329386B1 NO20044031A NO20044031A NO329386B1 NO 329386 B1 NO329386 B1 NO 329386B1 NO 20044031 A NO20044031 A NO 20044031A NO 20044031 A NO20044031 A NO 20044031A NO 329386 B1 NO329386 B1 NO 329386B1
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Norway
Prior art keywords
trifluoro
methyl
ylmethyl
fluoro
methoxyphenyl
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NO20044031A
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English (en)
Norwegian (no)
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NO20044031L (no
Inventor
Younes Bekkali
Raj Betageri
Thomas A Gilmore
Mario G Cardozo
Thomas M Kirrane
Daniel Kuzmich
John Robert Proudfoot
Hidenori Takahashi
David Thomson
Ji Wang
Renee Zindell
Christian Hanke Justus Joachim Harcken
Doris Riether
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Boehringer Ingelheim Pharma
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Publication of NO20044031L publication Critical patent/NO20044031L/no
Publication of NO329386B1 publication Critical patent/NO329386B1/no

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    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
NO20044031A 2002-03-26 2004-09-24 Glukocorticoid-mimetica, farmasoytiske preparater og anvendelser for fremstilling av medikamenterfor behandling av sykdom NO329386B1 (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US36775802P 2002-03-26 2002-03-26
US43181702P 2002-12-09 2002-12-09
US44240403P 2003-01-24 2003-01-24
PCT/US2003/008901 WO2003082280A1 (en) 2002-03-26 2003-03-21 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof

Publications (2)

Publication Number Publication Date
NO20044031L NO20044031L (no) 2004-10-19
NO329386B1 true NO329386B1 (no) 2010-10-11

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