NO308361B1 - Nye erytromycinderivater, samt legemidler som inneholder slike - Google Patents

Nye erytromycinderivater, samt legemidler som inneholder slike

Info

Publication number
NO308361B1
NO308361B1 NO954942A NO954942A NO308361B1 NO 308361 B1 NO308361 B1 NO 308361B1 NO 954942 A NO954942 A NO 954942A NO 954942 A NO954942 A NO 954942A NO 308361 B1 NO308361 B1 NO 308361B1
Authority
NO
Norway
Prior art keywords
well
drugs containing
erythromycin derivatives
new erythromycin
new
Prior art date
Application number
NO954942A
Other languages
English (en)
Norwegian (no)
Other versions
NO954942D0 (no
NO954942L (no
Inventor
Constantin Agouridas
Yannick Benedetti
Jean-Francois Chantot
Alexis Denis
Odile Le Martret
Original Assignee
Hoechst Marion Roussel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc
Publication of NO954942D0 publication Critical patent/NO954942D0/no
Publication of NO954942L publication Critical patent/NO954942L/no
Publication of NO308361B1 publication Critical patent/NO308361B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
NO954942A 1994-04-08 1995-12-06 Nye erytromycinderivater, samt legemidler som inneholder slike NO308361B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9404154A FR2718450B1 (fr) 1994-04-08 1994-04-08 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
PCT/FR1995/000441 WO1995027720A1 (fr) 1994-04-08 1995-04-06 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (3)

Publication Number Publication Date
NO954942D0 NO954942D0 (no) 1995-12-06
NO954942L NO954942L (no) 1996-02-07
NO308361B1 true NO308361B1 (no) 2000-09-04

Family

ID=9461886

Family Applications (1)

Application Number Title Priority Date Filing Date
NO954942A NO308361B1 (no) 1994-04-08 1995-12-06 Nye erytromycinderivater, samt legemidler som inneholder slike

Country Status (49)

Country Link
US (2) US5656607A (esLanguage)
EP (1) EP0676409B1 (esLanguage)
JP (1) JP3000023B2 (esLanguage)
KR (1) KR100317148B1 (esLanguage)
CN (1) CN1059445C (esLanguage)
AP (1) AP587A (esLanguage)
AT (1) ATE234853T1 (esLanguage)
AU (1) AU684939B2 (esLanguage)
BG (1) BG61916B1 (esLanguage)
BR (1) BR9506147A (esLanguage)
CA (1) CA2164638C (esLanguage)
CO (1) CO4370097A1 (esLanguage)
CZ (1) CZ296005B6 (esLanguage)
DE (1) DE69529934T2 (esLanguage)
DK (1) DK0676409T3 (esLanguage)
DZ (1) DZ1869A1 (esLanguage)
EE (1) EE04498B1 (esLanguage)
ES (1) ES2189820T3 (esLanguage)
FI (1) FI111264B (esLanguage)
FR (1) FR2718450B1 (esLanguage)
GB (1) GB2288174A (esLanguage)
GE (1) GEP19991836B (esLanguage)
HR (1) HRP950217B1 (esLanguage)
HU (1) HU215396B (esLanguage)
IL (1) IL112954A (esLanguage)
IS (1) IS1865B (esLanguage)
JO (1) JO1850B1 (esLanguage)
LV (1) LV11182B (esLanguage)
MA (1) MA23501A1 (esLanguage)
MD (1) MD663G2 (esLanguage)
MY (1) MY114672A (esLanguage)
NO (1) NO308361B1 (esLanguage)
NZ (1) NZ284498A (esLanguage)
OA (1) OA10200A (esLanguage)
PE (1) PE2896A1 (esLanguage)
PL (1) PL180837B1 (esLanguage)
PT (1) PT676409E (esLanguage)
RO (1) RO115634B1 (esLanguage)
RU (1) RU2141965C1 (esLanguage)
SA (1) SA97170757A (esLanguage)
SI (1) SI0676409T1 (esLanguage)
SK (1) SK284079B6 (esLanguage)
SV (1) SV1995000018A (esLanguage)
TN (1) TNSN95026A1 (esLanguage)
TW (1) TW316908B (esLanguage)
UA (1) UA44705C2 (esLanguage)
WO (1) WO1995027720A1 (esLanguage)
YU (1) YU49221B (esLanguage)
ZA (1) ZA952059B (esLanguage)

Families Citing this family (50)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2732023B1 (fr) * 1995-03-22 1997-04-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2745289B1 (fr) * 1996-02-28 1998-05-29 Roussel Uclaf Nouveaux derives de l'acide 1(2h) quinoleine carboxylique, leur procede de preparation et leur application a la synthese de produits doues de proprietes antibiotiques
US5750510A (en) * 1997-04-04 1998-05-12 Abbott Laboratories 3-descladinose-2,3-anhydroerythromycin derivatives
CZ349698A3 (cs) * 1996-05-07 1999-04-14 Abbott Laboratories 3-deskladinoso-2,3-anhydroerythromycinové deriváty
FR2748746B1 (fr) * 1996-05-14 1998-08-14 Hoechst Marion Roussel Inc Nouveau procede d'isomerisation du radical methyle en 10 de derives de l'erythromycine
FR2751656B1 (fr) * 1996-07-24 1998-10-16 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
UA51730C2 (uk) * 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
ATE299508T1 (de) * 1996-09-04 2005-07-15 Abbott Lab 6-o-substituierte ketoliden mit antibakteriellen wirkung
FR2757168B1 (fr) * 1996-12-12 1999-06-11 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2760017B1 (fr) * 1997-02-27 1999-04-30 Hoechst Marion Roussel Inc Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments
AU4472897A (en) * 1997-03-10 1998-09-29 Taisho Pharmaceutical Co., Ltd. Erythromycin a derivatives
WO1998042720A1 (fr) * 1997-03-24 1998-10-01 Taisho Pharmaceutical Co., Ltd. Derives d'erythromycine a
US6162794A (en) * 1997-05-09 2000-12-19 Pfizer Inc. Erythromycin derivatives
US5922683A (en) * 1997-05-29 1999-07-13 Abbott Laboratories Multicyclic erythromycin derivatives
ID24529A (id) * 1997-06-11 2000-07-20 Pfizer Prod Inc Turunan-turunan 9-oksima eritromisin
FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
AP1060A (en) * 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
HRP980189B1 (en) * 1998-04-06 2004-04-30 Pliva Pharm & Chem Works Novel 15-membered lactams ketolides
ES2243066T3 (es) 1998-09-22 2005-11-16 Pfizer Products Inc. Antibioticos de carbamato y carbazato cetolida.
FR2786188B1 (fr) * 1998-11-24 2002-10-31 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments
ES2273964T3 (es) 1998-12-10 2007-05-16 Pfizer Products Inc. Antibioticos de carbamato y carbazato cetolida.
EP1298138B1 (en) * 1998-12-10 2006-11-02 Pfizer Products Inc. Carbamate and Carbazate Ketolide Antibiotics
EP1749832A3 (en) * 1998-12-10 2008-03-26 Pfizer Products Incorporated Carbamate and carbazate ketolide antibiotics
FR2789392B1 (fr) * 1999-02-04 2001-10-05 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
US6054435A (en) * 1999-03-19 2000-04-25 Abbott Laboratories 6-O-substituted macrolides having antibacterial activity
MXPA01010521A (es) 1999-04-16 2003-08-19 Johnson & Johnson Antibacteriales de cetolidos.
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
EP1171446B1 (en) * 1999-04-16 2006-09-20 Kosan Biosciences, Inc. Macrolide antiinfective agents
IL145739A0 (en) * 1999-05-24 2002-07-25 Pfizer Prod Inc 13-methyl-erythromycin derivatives
AU2002316550A1 (en) 2001-07-03 2003-01-21 Chiron Corporation C12 modified erythromycin macrolides and ketolides having antibacterial activity
JP2006508643A (ja) 2002-07-01 2006-03-16 アーキオン ライフ サイエンシーズ エルエルシー ディー／ビー／エー バイオ−テクニカル リソーセズ ディビジョン グルコサミンおよびｎ−アセチルグルコサミン製造のためのプロセスおよび材料
CA2801100A1 (en) * 2003-03-10 2004-09-23 Optimer Pharmaceuticals, Inc. Macrolides and processes for their preparation
US7332476B2 (en) * 2003-04-25 2008-02-19 Novartis Ag Pyridyl substituted ketolide antibiotics
US7163924B2 (en) * 2003-04-25 2007-01-16 Chiron Corporation Ketolide derivatives
AU2008316830B2 (en) * 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
CN102245195B (zh) 2008-10-24 2016-01-13 森普拉制药公司 使用含三唑的大环内酯的生物防御
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
CN102724874B (zh) 2009-09-10 2018-06-01 森普拉制药公司 治疗疟疾、结核病和mac疾病的方法
CN108570083A (zh) 2010-03-22 2018-09-25 森普拉制药公司 大环内脂的结晶形式及其用途
CN102917708B (zh) 2010-05-20 2015-11-25 森普拉制药公司 制备大环内酯和酮内酯及其中间体的方法
US9815863B2 (en) 2010-09-10 2017-11-14 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
KR20140139083A (ko) 2012-03-27 2014-12-04 셈프라 파마슈티컬스, 인크. 마크롤라이드계 항생제를 투여하기 위한 비경구 제제
CA2905975A1 (en) 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
JP6675973B2 (ja) 2013-03-15 2020-04-08 センプラ ファーマシューティカルズ，インコーポレイテッド マクロライド抗菌薬を調製するための集束的な方法
MX377459B (es) 2013-04-04 2025-03-10 Harvard College Macrolidos y metodos para su preparacion y uso.
US10633407B2 (en) * 2014-10-08 2020-04-28 President And Fellows Of Harvard College 14-membered ketolides and methods of their preparation and use
HK1250371A1 (zh) 2015-03-25 2018-12-14 President And Fellows Of Harvard College 具有修饰的脱氧糖胺糖的大环内酯及其用途
MD1222Z (ro) * 2017-05-31 2018-08-31 ИНСТИТУТ ЭЛЕКТРОННОЙ ИНЖЕНЕРИИ И НАНОТЕХНОЛОГИЙ "D. Ghitu" АНМ Procedeu de tratare a materialului săditor al florilor înainte de plantare
JP7199722B2 (ja) 2019-12-25 2023-01-06 旭精工株式会社 硬貨搬送振分機構及びそれを備えた硬貨識別搬送装置

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3868414A (en) * 1973-01-22 1975-02-25 Merck & Co Inc Tetrahydrofluorene carboxylic acids and related compounds
AT342770B (de) * 1975-04-07 1978-04-25 Thomae Gmbh Dr K Verfahren zur herstellung neuer erythromycinderivate
DE2842759A1 (de) * 1978-09-30 1980-04-10 Merck Patent Gmbh Basische aether, diese enthaltende pharmazeutische zubereitungen und verfahren zu ihrer herstellung
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of erythromycin derivatives
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
FR2697524B1 (fr) * 1992-11-05 1994-12-23 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
HRP930014A2 (en) * 1993-01-08 1994-08-31 Pliva Pharm & Chem Works 9-deoxo-9a-aza-11-deoxy-9a-homoeritromycin a 9a, 11-cyclic carbamates
FR2702480B1 (fr) * 1993-03-09 1995-04-28 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Also Published As

Publication number Publication date
ES2189820T3 (es) 2003-07-16
EE04498B1 (et) 2005-06-15
EE9500080A (et) 1996-12-16
YU21695A (sh) 1997-12-05
DE69529934T2 (de) 2003-09-04
MD663F1 (ro) 1997-01-31
WO1995027720A1 (fr) 1995-10-19
US5760233A (en) 1998-06-02
NO954942D0 (no) 1995-12-06
EP0676409A1 (fr) 1995-10-11
CZ322395A3 (en) 1996-08-14
JPH07278177A (ja) 1995-10-24
FI111264B (fi) 2003-06-30
US5656607A (en) 1997-08-12
IL112954A0 (en) 1995-06-29
HRP950217A2 (en) 1997-08-31
MA23501A1 (fr) 1995-12-31
KR100317148B1 (ko) 2002-06-22
CN1059445C (zh) 2000-12-13
IS4309A (is) 1995-11-17
RU2141965C1 (ru) 1999-11-27
BG61916B1 (bg) 1998-09-30
CO4370097A1 (es) 1996-10-07
SV1995000018A (es) 1997-10-24
LV11182A (lv) 1996-04-20
FR2718450A1 (fr) 1995-10-13
AU684939B2 (en) 1998-01-08
PL180837B1 (pl) 2001-04-30
TW316908B (esLanguage) 1997-10-01
ZA952059B (en) 1996-03-13
NO954942L (no) 1996-02-07
MY114672A (en) 2002-12-31
SI0676409T1 (en) 2003-06-30
HRP950217B1 (en) 2004-06-30
PT676409E (pt) 2003-08-29
GB2288174A (en) 1995-10-11
SK154695A3 (en) 1996-10-02
UA44705C2 (uk) 2002-03-15
GEP19991836B (en) 1999-11-05
NZ284498A (en) 1997-07-27
AP9500743A0 (en) 1995-07-31
DE69529934D1 (de) 2003-04-24
RO115634B1 (ro) 2000-04-28
PL311871A1 (en) 1996-03-18
IS1865B (is) 2003-05-02
DZ1869A1 (fr) 2002-02-17
IL112954A (en) 2000-07-16
AU2310795A (en) 1995-10-30
TNSN95026A1 (fr) 1996-02-06
CZ296005B6 (cs) 2005-12-14
DK0676409T3 (da) 2003-06-23
YU49221B (sh) 2004-11-25
FI955913A7 (fi) 1995-12-08
GB9506856D0 (en) 1995-05-24
CA2164638A1 (fr) 1995-10-19
BG100150A (bg) 1996-06-28
FR2718450B1 (fr) 1997-01-10
JP3000023B2 (ja) 2000-01-17
EP0676409B1 (fr) 2003-03-19
JO1850B1 (en) 1995-12-27
FI955913A0 (fi) 1995-12-08
SA97170757A (ar) 2005-12-03
BR9506147A (pt) 1996-04-16
OA10200A (fr) 1996-12-18
CN1126997A (zh) 1996-07-17
LV11182B (en) 1997-04-20
CA2164638C (fr) 2003-12-30
HU9503505D0 (en) 1996-02-28
PE2896A1 (es) 1996-02-12
AP587A (en) 1997-04-29
HU215396B (hu) 1998-12-28
MD663G2 (ro) 1997-07-31
SK284079B6 (sk) 2004-09-08
ATE234853T1 (de) 2003-04-15
HUT73772A (en) 1996-09-30

Similar Documents

Publication Publication Date Title
NO308361B1 (no) Nye erytromycinderivater, samt legemidler som inneholder slike
NO308853B1 (no) Nye erytromycinderivater, farmasøytiske preparater som inneholder dem, samt mellomprodukter for deres fremstilling
NO307459B1 (no) Piperazinderivater, samt farmasøytiske preparater inneholdende slike
NO973923D0 (no) Nye taxoider, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene
FI893581L (fi) Som bilens vindruta anvaendbar, genom pyrolys av pulverformiga foereningar framstaelld, med elledande skikt foersedd glasdel.
FI930989A0 (fi) Foerfarande foer tillverkning av byggelement foer ljusvaogsledningsnaetverk, samt byggelement som tillverkats enligt foerfarandet
FI905958A7 (fi) Foerfarande foer framstaellning av substituerade cyklohexanoler, som verkar pao det centrala nervsystemet.
FI931278L (fi) Polymerer, som innehaoller sulfogrupper
FI922222A7 (fi) Kopplingsanordning, som foermaor laosa spinalosteosyntesfaestanordningar
FI925615L (fi) Stabiliserade farmaceutiska kompositioner, som innehaoller en HMG-CoA-reduktas-inhibitorfoerening
FI923281L (fi) Foerbaettrade desinfektionsloesningar, som innehaoller vaeteperoxid
FI893557A0 (fi) Polyestrar, som innehaoller en eterbrygga.
FI895225A0 (fi) Foerfarande foer borttagning av tungmetaller, saerskilt kadmium, fraon loesningar som innehaoller fosforsyra.
FI903028A0 (fi) Polymerbaserade blandningskompositioner, som innehaoller destrukturerad staerkelse.
FI860842A7 (fi) Labdan-derivat, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.
FI922235L (fi) Foerfarande foer framstaellning av 3-aminopyridazinderivat, som verkar paodet centrala nervsystemet
DK1016669T3 (da) Nye erythromycinderivater, fremgangsmåde til deres fremstilling samt deres anvendelse som lægemidler
FI925993L (fi) Katjoniska polymerer, som filtrations fraemjande tillaegsmedel samt som stabilatorer i hartsinnehaollande papperslim
FI900870A0 (fi) Foerfarande foer belaeggning av papper med kompositioner, som innehaoller mikrokapslar.
FI864164L (fi) Biologiskt aktiva derivat av human- -interferon, deras framstaellning och laekemedel, som innehaoller dylika derivat.
FI932111A7 (fi) Anordning foer att bestryka en materialbana, isynnerhet en pappers- eller kartongbana som foers runt en motvals
NO974563D0 (no) Nye taxoider, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene
FI914453A7 (fi) Foerfarande foer kompressering av en videobild, som kodats digitaliskt
FI885852A7 (fi) Anordning foer sluta en foerpackning runt en vara, som skall foerpackas.
FI905957A7 (fi) Foerfarande foer framstaellning av substituerade cyklohexener, som verkar pao det centrala nervsystemet.

Legal Events

Date Code Title Description
MK1K Patent expired