NO308361B1 - Nye erytromycinderivater, samt legemidler som inneholder slike - Google Patents

Nye erytromycinderivater, samt legemidler som inneholder slike

Info

Publication number
NO308361B1
NO308361B1 NO954942A NO954942A NO308361B1 NO 308361 B1 NO308361 B1 NO 308361B1 NO 954942 A NO954942 A NO 954942A NO 954942 A NO954942 A NO 954942A NO 308361 B1 NO308361 B1 NO 308361B1
Authority
NO
Norway
Prior art keywords
well
drugs containing
erythromycin derivatives
new erythromycin
new
Prior art date
Application number
NO954942A
Other languages
English (en)
Norwegian (no)
Other versions
NO954942D0 (no
NO954942L (no
Inventor
Constantin Agouridas
Yannick Benedetti
Jean-Francois Chantot
Alexis Denis
Odile Le Martret
Original Assignee
Hoechst Marion Roussel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc
Publication of NO954942D0 publication Critical patent/NO954942D0/no
Publication of NO954942L publication Critical patent/NO954942L/no
Publication of NO308361B1 publication Critical patent/NO308361B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NO954942A 1994-04-08 1995-12-06 Nye erytromycinderivater, samt legemidler som inneholder slike NO308361B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9404154A FR2718450B1 (fr) 1994-04-08 1994-04-08 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
PCT/FR1995/000441 WO1995027720A1 (fr) 1994-04-08 1995-04-06 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (3)

Publication Number Publication Date
NO954942D0 NO954942D0 (no) 1995-12-06
NO954942L NO954942L (no) 1996-02-07
NO308361B1 true NO308361B1 (no) 2000-09-04

Family

ID=9461886

Family Applications (1)

Application Number Title Priority Date Filing Date
NO954942A NO308361B1 (no) 1994-04-08 1995-12-06 Nye erytromycinderivater, samt legemidler som inneholder slike

Country Status (49)

Country Link
US (2) US5656607A (da)
EP (1) EP0676409B1 (da)
JP (1) JP3000023B2 (da)
KR (1) KR100317148B1 (da)
CN (1) CN1059445C (da)
AP (1) AP587A (da)
AT (1) ATE234853T1 (da)
AU (1) AU684939B2 (da)
BG (1) BG61916B1 (da)
BR (1) BR9506147A (da)
CA (1) CA2164638C (da)
CO (1) CO4370097A1 (da)
CZ (1) CZ296005B6 (da)
DE (1) DE69529934T2 (da)
DK (1) DK0676409T3 (da)
DZ (1) DZ1869A1 (da)
EE (1) EE04498B1 (da)
ES (1) ES2189820T3 (da)
FI (1) FI111264B (da)
FR (1) FR2718450B1 (da)
GB (1) GB2288174A (da)
GE (1) GEP19991836B (da)
HR (1) HRP950217B1 (da)
HU (1) HU215396B (da)
IL (1) IL112954A (da)
IS (1) IS1865B (da)
JO (1) JO1850B1 (da)
LV (1) LV11182B (da)
MA (1) MA23501A1 (da)
MD (1) MD663G2 (da)
MY (1) MY114672A (da)
NO (1) NO308361B1 (da)
NZ (1) NZ284498A (da)
OA (1) OA10200A (da)
PE (1) PE2896A1 (da)
PL (1) PL180837B1 (da)
PT (1) PT676409E (da)
RO (1) RO115634B1 (da)
RU (1) RU2141965C1 (da)
SA (1) SA97170757A (da)
SI (1) SI0676409T1 (da)
SK (1) SK284079B6 (da)
SV (1) SV1995000018A (da)
TN (1) TNSN95026A1 (da)
TW (1) TW316908B (da)
UA (1) UA44705C2 (da)
WO (1) WO1995027720A1 (da)
YU (1) YU49221B (da)
ZA (1) ZA952059B (da)

Families Citing this family (49)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2732023B1 (fr) * 1995-03-22 1997-04-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2742757B1 (fr) 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2745289B1 (fr) * 1996-02-28 1998-05-29 Roussel Uclaf Nouveaux derives de l'acide 1(2h) quinoleine carboxylique, leur procede de preparation et leur application a la synthese de produits doues de proprietes antibiotiques
US5750510A (en) * 1997-04-04 1998-05-12 Abbott Laboratories 3-descladinose-2,3-anhydroerythromycin derivatives
AU710532B2 (en) * 1996-05-07 1999-09-23 Abbott Laboratories 3-descladinose-2,3-anhydroerythromycin derivatives
FR2748746B1 (fr) * 1996-05-14 1998-08-14 Hoechst Marion Roussel Inc Nouveau procede d'isomerisation du radical methyle en 10 de derives de l'erythromycine
FR2751656B1 (fr) * 1996-07-24 1998-10-16 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
ATE296832T1 (de) * 1996-09-04 2005-06-15 Abbott Lab 6-o-substituierte ketoliden mit antibakteriellen wirkung
UA51730C2 (uk) * 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
FR2757168B1 (fr) * 1996-12-12 1999-06-11 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2760017B1 (fr) * 1997-02-27 1999-04-30 Hoechst Marion Roussel Inc Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments
WO1998040392A1 (fr) * 1997-03-10 1998-09-17 Taisho Pharmaceutical Co., Ltd. Derives d'erythromycine a
WO1998042720A1 (fr) * 1997-03-24 1998-10-01 Taisho Pharmaceutical Co., Ltd. Derives d'erythromycine a
AU6932098A (en) * 1997-05-09 1998-12-08 Pfizer Products Inc. Erythromycin derivatives
US5922683A (en) * 1997-05-29 1999-07-13 Abbott Laboratories Multicyclic erythromycin derivatives
EA199901016A1 (ru) * 1997-06-11 2000-06-26 Пфайзер Продактс Инк. 9-оксим-производные эритромицина
FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
AP1060A (en) * 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
ES2243066T3 (es) * 1998-09-22 2005-11-16 Pfizer Products Inc. Antibioticos de carbamato y carbazato cetolida.
FR2786188B1 (fr) * 1998-11-24 2002-10-31 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments
ATE344269T1 (de) 1998-12-10 2006-11-15 Pfizer Prod Inc Carbamat und carbazat ketolid antibiotika
EP1298138B1 (en) * 1998-12-10 2006-11-02 Pfizer Products Inc. Carbamate and Carbazate Ketolide Antibiotics
EP1749832A3 (en) * 1998-12-10 2008-03-26 Pfizer Products Incorporated Carbamate and carbazate ketolide antibiotics
FR2789392B1 (fr) 1999-02-04 2001-10-05 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
US6054435A (en) * 1999-03-19 2000-04-25 Abbott Laboratories 6-O-substituted macrolides having antibacterial activity
AU4354900A (en) 1999-04-16 2000-11-02 Kosan Biosciences, Inc. Ketolide antibacterials
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
ES2272273T3 (es) * 1999-04-16 2007-05-01 Kosan Biosciences, Inc. Agentes antiinfecciosos macrolidos.
WO2000071557A1 (en) * 1999-05-24 2000-11-30 Pfizer Products Inc. 13-methyl-erythromycin derivatives
WO2003004509A2 (en) * 2001-07-03 2003-01-16 Chiron Corporation C12 modified erythromycin macrolides and ketolides having antibacterial activity
US7332304B2 (en) 2002-07-01 2008-02-19 Arkion Life Sciences Llc Process and materials for production of glucosamine and N-acetylglucosamine
CA2529817C (en) 2003-03-10 2013-02-12 Optimer Pharmaceuticals, Inc. Novel antibacterial agents
EP1618119A2 (en) * 2003-04-25 2006-01-25 Chiron Corporation Pyridyl substituted ketolide antibiotics
US7163924B2 (en) * 2003-04-25 2007-01-16 Chiron Corporation Ketolide derivatives
CN101917850B (zh) 2007-10-25 2016-01-13 森普拉制药公司 大环内酯类抗菌剂的制备方法
WO2010048599A1 (en) 2008-10-24 2010-04-29 Cempra Pharmaceuticals, Inc. Methods for treating gastrointestinal diseases
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
JP5914335B2 (ja) 2009-09-10 2016-05-11 センプラ ファーマシューティカルズ，インコーポレイテッド マラリア、結核、及びｍａｃ病の治療方法
NZ602544A (en) 2010-03-22 2014-11-28 Cempra Pharmaceuticals Inc Crystalline forms of a macrolide, and uses therefor
US9051346B2 (en) 2010-05-20 2015-06-09 Cempra Pharmaceuticals, Inc. Process for preparing triazole-containing ketolide antibiotics
JP6042334B2 (ja) 2010-09-10 2016-12-14 センプラ ファーマシューティカルズ，インコーポレイテッド 疾患治療のための水素結合形成フルオロケトライド
SG11201405895UA (en) 2012-03-27 2014-10-30 Cempra Pharmaceuticals Inc Parenteral formulations for administering macrolide antibiotics
US9861616B2 (en) 2013-03-14 2018-01-09 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
JP6675973B2 (ja) 2013-03-15 2020-04-08 センプラ ファーマシューティカルズ，インコーポレイテッド マクロライド抗菌薬を調製するための集束的な方法
US9982005B2 (en) 2013-04-04 2018-05-29 President And Fellows Of Harvard College Macrolides and methods of their preparation and use
WO2016057798A1 (en) 2014-10-08 2016-04-14 President And Fellows Of Harvard College 14-membered ketolides and methods of their preparation and use
CN107530365A (zh) 2015-03-25 2018-01-02 哈佛大学的校长及成员们 具有修饰的脱氧糖胺糖的大环内酯及其用途
MD1222Z (ro) * 2017-05-31 2018-08-31 ИНСТИТУТ ЭЛЕКТРОННОЙ ИНЖЕНЕРИИ И НАНОТЕХНОЛОГИЙ "D. Ghitu" АНМ Procedeu de tratare a materialului săditor al florilor înainte de plantare
JP7199722B2 (ja) 2019-12-25 2023-01-06 旭精工株式会社 硬貨搬送振分機構及びそれを備えた硬貨識別搬送装置

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3868414A (en) * 1973-01-22 1975-02-25 Merck & Co Inc Tetrahydrofluorene carboxylic acids and related compounds
DE2842759A1 (de) * 1978-09-30 1980-04-10 Merck Patent Gmbh Basische aether, diese enthaltende pharmazeutische zubereitungen und verfahren zu ihrer herstellung
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
FR2697524B1 (fr) * 1992-11-05 1994-12-23 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
HRP930014A2 (en) * 1993-01-08 1994-08-31 Pliva Pharm & Chem Works 9-deoxo-9a-aza-11-deoxy-9a-homoeritromycin a 9a, 11-cyclic carbamates
FR2702480B1 (fr) * 1993-03-09 1995-04-28 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Also Published As

Publication number Publication date
ES2189820T3 (es) 2003-07-16
GB2288174A (en) 1995-10-11
LV11182B (en) 1997-04-20
BG100150A (bg) 1996-06-28
CN1059445C (zh) 2000-12-13
AU684939B2 (en) 1998-01-08
YU21695A (sh) 1997-12-05
LV11182A (lv) 1996-04-20
GB9506856D0 (en) 1995-05-24
HRP950217B1 (en) 2004-06-30
ZA952059B (en) 1996-03-13
FI955913A (fi) 1995-12-08
MD663G2 (ro) 1997-07-31
SI0676409T1 (en) 2003-06-30
US5760233A (en) 1998-06-02
HU215396B (hu) 1998-12-28
MY114672A (en) 2002-12-31
DE69529934T2 (de) 2003-09-04
FI111264B (fi) 2003-06-30
RU2141965C1 (ru) 1999-11-27
PE2896A1 (es) 1996-02-12
PL180837B1 (pl) 2001-04-30
EP0676409A1 (fr) 1995-10-11
MD663F1 (ro) 1997-01-31
FI955913A0 (fi) 1995-12-08
JP3000023B2 (ja) 2000-01-17
PL311871A1 (en) 1996-03-18
NO954942D0 (no) 1995-12-06
SA97170757A (ar) 2005-12-03
AU2310795A (en) 1995-10-30
EE9500080A (et) 1996-12-16
WO1995027720A1 (fr) 1995-10-19
IL112954A0 (en) 1995-06-29
BR9506147A (pt) 1996-04-16
KR100317148B1 (ko) 2002-06-22
HU9503505D0 (en) 1996-02-28
AP9500743A0 (en) 1995-07-31
AP587A (en) 1997-04-29
TW316908B (da) 1997-10-01
UA44705C2 (uk) 2002-03-15
MA23501A1 (fr) 1995-12-31
IS4309A (is) 1995-11-17
EE04498B1 (et) 2005-06-15
DE69529934D1 (de) 2003-04-24
CN1126997A (zh) 1996-07-17
CO4370097A1 (es) 1996-10-07
NO954942L (no) 1996-02-07
IL112954A (en) 2000-07-16
CA2164638A1 (fr) 1995-10-19
SK284079B6 (sk) 2004-09-08
HRP950217A2 (en) 1997-08-31
FR2718450B1 (fr) 1997-01-10
IS1865B (is) 2003-05-02
CZ296005B6 (cs) 2005-12-14
EP0676409B1 (fr) 2003-03-19
TNSN95026A1 (fr) 1996-02-06
SK154695A3 (en) 1996-10-02
OA10200A (fr) 1996-12-18
JPH07278177A (ja) 1995-10-24
RO115634B1 (ro) 2000-04-28
DK0676409T3 (da) 2003-06-23
CZ322395A3 (en) 1996-08-14
DZ1869A1 (fr) 2002-02-17
PT676409E (pt) 2003-08-29
CA2164638C (fr) 2003-12-30
NZ284498A (en) 1997-07-27
JO1850B1 (en) 1995-12-27
YU49221B (sh) 2004-11-25
FR2718450A1 (fr) 1995-10-13
BG61916B1 (bg) 1998-09-30
US5656607A (en) 1997-08-12
SV1995000018A (es) 1997-10-24
ATE234853T1 (de) 2003-04-15
HUT73772A (en) 1996-09-30
GEP19991836B (en) 1999-11-05

Similar Documents

Publication Publication Date Title
NO308361B1 (no) Nye erytromycinderivater, samt legemidler som inneholder slike
NO308853B1 (no) Nye erytromycinderivater, farmasøytiske preparater som inneholder dem, samt mellomprodukter for deres fremstilling
NO973923D0 (no) Nye taxoider, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene
NO307459B1 (no) Piperazinderivater, samt farmasøytiske preparater inneholdende slike
FI930989A0 (fi) Foerfarande foer tillverkning av byggelement foer ljusvaogsledningsnaetverk, samt byggelement som tillverkats enligt foerfarandet
FI931278A0 (fi) Polymerer, som innehaoller sulfogrupper
FI893557A (fi) Polyestrar, som innehaoller en eterbrygga.
FI903028A0 (fi) Polymerbaserade blandningskompositioner, som innehaoller destrukturerad staerkelse.
FI895225A0 (fi) Foerfarande foer borttagning av tungmetaller, saerskilt kadmium, fraon loesningar som innehaoller fosforsyra.
DK1016669T3 (da) Nye erythromycinderivater, fremgangsmåde til deres fremstilling samt deres anvendelse som lægemidler
ATE212635T1 (de) 1,3,8-triazaspiro(4,5)decan-4-on-derivate
FI900870A0 (fi) Foerfarande foer belaeggning av papper med kompositioner, som innehaoller mikrokapslar.
FI915492A0 (fi) 9a-hydroxi-19,11b-oeverbryggade steroider, deras framstaellning och farmaceutiska preparat som innehaoller dem.
NO974563D0 (no) Nye taxoider, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene
FI905020A0 (fi) Orala kompositioner, som innehaoller monoperoxisyror.
DK0931088T3 (da) Nye erythromycinforbindelser, fremgangsmåde til deres fremstilling samt deres anvendelse som lægemidler
FI904191A0 (fi) Nya aminopropanolderivater, foerfarande foer tillverkning av dessa samt farmaceutiska sammansaettningar som innehaoller dessa.
FI890098A (fi) Pyrazol- och indazolpyridinaminer, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.
FI894982A0 (fi) Massaaendlaoden foer maskin som tillverkar fiberband, saerskilt pappersband.
NO993124D0 (no) Nye erytromycinderivater, fremgangsmÕte for fremstilling av disse samt deres anvendelse som medisiner
NO873628L (no) 2,3-dihydro-1h-fenalen-2-amino-forbindelser som antipsykotiske legemidler.
FI903885A0 (fi) Ny oral farmaceutisk doseringsform som foerbaettrar biotillgaengligheten.
NO952426D0 (no) Nytt legemiddel som inneholder 3,7-diazabisyklo[3,3,1Ånonan forbindelser
FI932034A0 (fi) Nya 1-azacykloalkanderivat, farmaceutiska sammansaettningar som innehaoller dessa samt foerfarande foer framstaellning daerav
FI894434A0 (fi) Saett foer bevisning av tillraecklighet av magnetfloede, som framkallas av ett magnetiseringsok vid magnetisk felsoekning.

Legal Events

Date Code Title Description
MK1K Patent expired