NO20004546L - Caspaseinhibitorer - Google Patents

Caspaseinhibitorer

Info

Publication number
NO20004546L
NO20004546L NO20004546A NO20004546A NO20004546L NO 20004546 L NO20004546 L NO 20004546L NO 20004546 A NO20004546 A NO 20004546A NO 20004546 A NO20004546 A NO 20004546A NO 20004546 L NO20004546 L NO 20004546L
Authority
NO
Norway
Prior art keywords
caspaseinhibitorer
Prior art date
Application number
NO20004546A
Other languages
English (en)
Other versions
NO331829B1 (no
NO20004546D0 (no
Inventor
Marion W Wannamaker
Guy W Bemis
Paul S Charifson
David J Lauffer
Michael D Mullican
Mark A Murcko
Keith P Wilson
James W Janetka
Robert J Davies
Anne-Laure Grillot
Zhan Shi
Cornelia J Forster
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of NO20004546D0 publication Critical patent/NO20004546D0/no
Publication of NO20004546L publication Critical patent/NO20004546L/no
Publication of NO331829B1 publication Critical patent/NO331829B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • A—HUMAN NECESSITIES
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
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    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
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  • Diabetes (AREA)
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  • Neurology (AREA)
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  • Biomedical Technology (AREA)
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  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
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  • Proteomics, Peptides & Aminoacids (AREA)
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  • Biochemistry (AREA)
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NO20004546A 1998-03-19 2000-09-12 Cykliske forbindelser med caspaseinhibitor-aktivitet, sammensetninger inneholdende slike samt anvendelse derav ved fremstilling av medikamenter NO331829B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US7877098P 1998-03-19 1998-03-19
PCT/US1999/005919 WO1999047545A2 (en) 1998-03-19 1999-03-19 Inhibitors of caspases

Publications (3)

Publication Number Publication Date
NO20004546D0 NO20004546D0 (no) 2000-09-12
NO20004546L true NO20004546L (no) 2000-11-09
NO331829B1 NO331829B1 (no) 2012-04-16

Family

ID=22146109

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20004546A NO331829B1 (no) 1998-03-19 2000-09-12 Cykliske forbindelser med caspaseinhibitor-aktivitet, sammensetninger inneholdende slike samt anvendelse derav ved fremstilling av medikamenter

Country Status (34)

Country Link
US (3) US6531474B1 (no)
EP (6) EP1064298B1 (no)
JP (3) JP4594520B2 (no)
KR (2) KR100928878B1 (no)
CN (1) CN1321129C (no)
AP (1) AP2000001919A0 (no)
AR (1) AR019011A1 (no)
AT (1) ATE410439T1 (no)
AU (1) AU769033B2 (no)
BG (1) BG104863A (no)
BR (2) BR9909660A (no)
CA (1) CA2324226C (no)
CZ (1) CZ302281B6 (no)
DE (1) DE69939689D1 (no)
DK (1) DK1064298T3 (no)
ES (1) ES2315010T3 (no)
GE (1) GEP20043163B (no)
HK (1) HK1035733A1 (no)
HU (1) HU227920B1 (no)
ID (1) ID27002A (no)
IL (3) IL138469A0 (no)
IS (1) IS5622A (no)
NO (1) NO331829B1 (no)
NZ (2) NZ506963A (no)
PL (1) PL204619B1 (no)
PT (1) PT1064298E (no)
RU (1) RU2274642C2 (no)
SI (1) SI1064298T1 (no)
SK (1) SK286736B6 (no)
TR (1) TR200103406T2 (no)
TW (1) TWI243828B (no)
UA (2) UA74133C2 (no)
WO (1) WO1999047545A2 (no)
ZA (1) ZA200004652B (no)

Families Citing this family (76)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1064298B1 (en) * 1998-03-19 2008-10-08 Vertex Pharmaceuticals Incorporated Inhibitors of caspases
US7157430B2 (en) 1998-10-22 2007-01-02 Idun Pharmaceuticals, Inc. (Substituted)acyl dipeptidyl inhibitors of the ICE/CED-3 family of cysteine proteases
US6242422B1 (en) * 1998-10-22 2001-06-05 Idun Pharmacueticals, Inc. (Substituted)Acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
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JP4594520B2 (ja) 2010-12-08
WO1999047545A3 (en) 1999-11-25
EP2261233A2 (en) 2010-12-15
PT1064298E (pt) 2009-01-02
HU227920B1 (en) 2012-06-28
CZ302281B6 (cs) 2011-01-26
BR9909660A (pt) 2000-11-21
BRPI9909660B8 (pt) 2021-05-25
EP2261234A3 (en) 2011-04-20
HUP0103575A2 (hu) 2002-02-28
AU769033B2 (en) 2004-01-15

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