LV12889B - Kristālisks ceftiofūrs brīvas skābes formā - Google Patents

Kristālisks ceftiofūrs brīvas skābes formā Download PDF

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Publication number
LV12889B
LV12889B LVP-02-107A LV020107A LV12889B LV 12889 B LV12889 B LV 12889B LV 020107 A LV020107 A LV 020107A LV 12889 B LV12889 B LV 12889B
Authority
LV
Latvia
Prior art keywords
crystalline
free acid
ceftiofur
oil
compound
Prior art date
Application number
LVP-02-107A
Other languages
English (en)
Latvian (lv)
Inventor
Michael J. Dunn
Michael S. Bergren
Gregory E. Hardee
Kenneth Paul Shephard
Robert S. Chao
Jeffrey L. Havens
Original Assignee
Pharmacia & Upjohn Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Company filed Critical Pharmacia & Upjohn Company
Publication of LV12889B publication Critical patent/LV12889B/lv

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
LVP-02-107A 1993-03-12 2002-06-13 Kristālisks ceftiofūrs brīvas skābes formā LV12889B (lv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US3329193A 1993-03-12 1993-03-12

Publications (1)

Publication Number Publication Date
LV12889B true LV12889B (lv) 2002-12-20

Family

ID=21869579

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-02-107A LV12889B (lv) 1993-03-12 2002-06-13 Kristālisks ceftiofūrs brīvas skābes formā

Country Status (31)

Country Link
US (1) US5721359A (hr)
EP (1) EP0690864B1 (hr)
JP (1) JP3852946B2 (hr)
KR (1) KR100296810B1 (hr)
CN (1) CN1055090C (hr)
AT (1) ATE202109T1 (hr)
AU (1) AU694419B2 (hr)
BR (1) BR1101034A (hr)
CA (1) CA2155322C (hr)
CZ (1) CZ289332B6 (hr)
DE (2) DE69427469T2 (hr)
DK (1) DK0690864T3 (hr)
ES (1) ES2157254T3 (hr)
FI (1) FI120307B (hr)
FR (1) FR05C0045I2 (hr)
GR (1) GR3036514T3 (hr)
HU (1) HU222244B1 (hr)
IL (1) IL108910A (hr)
LU (1) LU91206I2 (hr)
LV (1) LV12889B (hr)
NL (1) NL300208I2 (hr)
NO (2) NO313199B1 (hr)
NZ (1) NZ263002A (hr)
PL (1) PL184611B1 (hr)
PT (1) PT690864E (hr)
RU (1) RU2136685C1 (hr)
SI (1) SI0690864T1 (hr)
SK (1) SK283674B6 (hr)
TW (1) TW267170B (hr)
WO (1) WO1994020505A1 (hr)
ZA (1) ZA941586B (hr)

Families Citing this family (70)

* Cited by examiner, † Cited by third party
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BR0308523A (pt) 2002-03-21 2005-02-01 Upjohn Co Método de administração de um antibiótico injetável à orelha de um animal
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EP2536701A4 (en) * 2010-02-18 2014-05-07 Astrazeneca Ab SOLID FORMS WITH A CYCLOPROPYLAMID DERIVATIVE
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CN104039369B (zh) 2011-07-20 2017-06-16 布莱阿姆青年大学 疏水性塞拉集宁化合物和包含该化合物的装置
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US9694019B2 (en) 2011-09-13 2017-07-04 Brigham Young University Compositions and methods for treating bone diseases and broken bones
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CN102584855B (zh) * 2012-02-16 2014-06-25 青岛科技大学 一种改进的头孢噻呋的制备方法
US9533063B1 (en) 2012-03-01 2017-01-03 Brigham Young University Aerosols incorporating ceragenin compounds and methods of use thereof
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CN105451742B (zh) 2013-01-07 2021-04-06 布莱阿姆青年大学 减少细胞增殖和治疗某些疾病的方法
US10568893B2 (en) 2013-03-15 2020-02-25 Brigham Young University Methods for treating inflammation, autoimmune disorders and pain
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JP6518230B2 (ja) 2013-03-15 2019-05-22 ブリガム・ヤング・ユニバーシティBrigham Young University 炎症、自己免疫疾患、および疼痛を治療する方法
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US9387215B2 (en) 2013-04-22 2016-07-12 Brigham Young University Animal feed including cationic cholesterol additive and related methods
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US11690855B2 (en) 2013-10-17 2023-07-04 Brigham Young University Methods for treating lung infections and inflammation
US20150203527A1 (en) 2014-01-23 2015-07-23 Brigham Young University Cationic steroidal antimicrobials
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US9867836B2 (en) 2014-03-13 2018-01-16 Brigham Young University Lavage and/or infusion using CSA compounds for increasing fertility in a mammal
US10220045B2 (en) 2014-03-13 2019-03-05 Brigham Young University Compositions and methods for forming stabilized compositions with reduced CSA agglomeration
US9931350B2 (en) 2014-03-14 2018-04-03 Brigham Young University Anti-infective and osteogenic compositions and methods of use
US9686966B2 (en) 2014-04-30 2017-06-27 Brigham Young University Methods and apparatus for cleaning or disinfecting a water delivery system
US10238665B2 (en) 2014-06-26 2019-03-26 Brigham Young University Methods for treating fungal infections
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US10227376B2 (en) 2014-08-22 2019-03-12 Brigham Young University Radiolabeled cationic steroid antimicrobials and diagnostic methods
US10155788B2 (en) 2014-10-07 2018-12-18 Brigham Young University Cationic steroidal antimicrobial prodrug compositions and uses thereof
AU2015335950B2 (en) * 2014-10-21 2018-01-25 Takeda Pharmaceutical Company Limited Crystalline forms of 5-chloro-N4-[-2-(dimethylphosphoryl) phenyl]-N2-{2-methoxy-4-[4-(4-methylpiperazin-1-yl) piperidin-1-yl] phenyl}pyrimidine-2,4-diamine
US9527883B2 (en) 2015-04-22 2016-12-27 Brigham Young University Methods for the synthesis of ceragenins
US10370403B2 (en) 2015-04-22 2019-08-06 Brigham Young University Methods for the synthesis of ceragenins
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Also Published As

Publication number Publication date
HUT73781A (en) 1996-09-30
SK111495A3 (en) 1995-12-06
DE69427469D1 (en) 2001-07-19
NO2005025I1 (no) 2005-12-05
JP3852946B2 (ja) 2006-12-06
DE122005000055I1 (de) 2006-02-23
NL300208I2 (nl) 2006-05-01
WO1994020505A1 (en) 1994-09-15
RU2136685C1 (ru) 1999-09-10
NZ263002A (en) 1996-12-20
NL300208I1 (nl) 2006-02-01
NO313199B1 (no) 2002-08-26
TW267170B (hr) 1996-01-01
FI954250A0 (fi) 1995-09-11
FI120307B (fi) 2009-09-15
FR05C0045I2 (hr) 2007-08-03
BR1101034A (pt) 2002-04-30
CN1055090C (zh) 2000-08-02
IL108910A0 (en) 1994-06-24
EP0690864B1 (en) 2001-06-13
PL184611B1 (pl) 2002-11-29
NO2005025I2 (no) 2010-11-22
US5721359A (en) 1998-02-24
DE69427469T2 (de) 2001-10-31
ATE202109T1 (de) 2001-06-15
PT690864E (pt) 2001-11-30
DE122005000055I2 (de) 2008-06-05
PL310556A1 (en) 1995-12-27
SI0690864T1 (en) 2001-10-31
HU9501960D0 (en) 1995-09-28
DK0690864T3 (da) 2001-09-17
CZ9502290A3 (cs) 2001-08-15
CN1119016A (zh) 1996-03-20
FI954250A (fi) 1995-09-11
GR3036514T3 (en) 2001-12-31
AU6351094A (en) 1994-09-26
SK283674B6 (sk) 2003-11-04
CA2155322C (en) 2000-02-29
NO953564L (no) 1995-11-07
FR05C0045I1 (hr) 2006-01-06
HU222244B1 (hu) 2003-05-28
CA2155322A1 (en) 1994-09-15
ZA941586B (en) 1995-09-07
ES2157254T3 (es) 2001-08-16
JPH08507519A (ja) 1996-08-13
NO953564D0 (no) 1995-09-11
EP0690864A1 (en) 1996-01-10
LU91206I2 (fr) 2006-05-30
KR100296810B1 (ko) 2001-10-24
AU694419B2 (en) 1998-07-23
CZ289332B6 (cs) 2002-01-16
IL108910A (en) 1999-10-28

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