KR20070024601A - 세린 프로테아제 억제제로서 유용한 5원 헤테로사이클 - Google Patents

세린 프로테아제 억제제로서 유용한 5원 헤테로사이클 Download PDF

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KR20070024601A
KR20070024601A KR1020067026365A KR20067026365A KR20070024601A KR 20070024601 A KR20070024601 A KR 20070024601A KR 1020067026365 A KR1020067026365 A KR 1020067026365A KR 20067026365 A KR20067026365 A KR 20067026365A KR 20070024601 A KR20070024601 A KR 20070024601A
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phenyl
substituted
benzyl
imidazol
alkyl
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Korean (ko)
Inventor
존 제이. 한겔란드
미미 엘. 쿠안
조앤 엠. 스몰헤르
그레고리 에스. 비사치
제임스 알. 코르테
토드 제이. 프렌즈
종 순
카렌 에이. 로시
쿨렌 엘. 카발라로
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브리스톨-마이어스 스큅 컴퍼니
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Application filed by 브리스톨-마이어스 스큅 컴퍼니 filed Critical 브리스톨-마이어스 스큅 컴퍼니
Publication of KR20070024601A publication Critical patent/KR20070024601A/ko
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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EP1773786A2 (en) 2007-04-18
US20090036438A1 (en) 2009-02-05
JP2008502700A (ja) 2008-01-31
US7453002B2 (en) 2008-11-18
WO2005123050A3 (en) 2007-01-04
EP1773786B1 (en) 2017-04-26
RU2007101073A (ru) 2008-07-20
BRPI0512084A (pt) 2008-02-06
WO2005123050A2 (en) 2005-12-29
US20170166560A1 (en) 2017-06-15
US9079860B2 (en) 2015-07-14
NO20065864L (no) 2007-03-02
ES2628279T3 (es) 2017-08-02
US20140206706A1 (en) 2014-07-24
US20050282805A1 (en) 2005-12-22
JP4791460B2 (ja) 2011-10-12
US8716492B2 (en) 2014-05-06
US10112936B2 (en) 2018-10-30
CA2570472A1 (en) 2005-12-29
IL179844A0 (en) 2007-07-04
US20120088758A1 (en) 2012-04-12
US9617224B2 (en) 2017-04-11
US20150259297A1 (en) 2015-09-17

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