MXPA06014642A - Heterociclos de cinco miembros utiles como inhibidores de la serina proteasa. - Google Patents

Heterociclos de cinco miembros utiles como inhibidores de la serina proteasa.

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Publication number
MXPA06014642A
MXPA06014642A MXPA06014642A MXPA06014642A MXPA06014642A MX PA06014642 A MXPA06014642 A MX PA06014642A MX PA06014642 A MXPA06014642 A MX PA06014642A MX PA06014642 A MXPA06014642 A MX PA06014642A MX PA06014642 A MXPA06014642 A MX PA06014642A
Authority
MX
Mexico
Prior art keywords
phenyl
substituted
benzyl
imidazol
ethyl
Prior art date
Application number
MXPA06014642A
Other languages
English (en)
Spanish (es)
Inventor
Gregory S Bisacchi
Mimi L Quan
James R Corte
Jon J Hangeland
Joanne M Smallheer
Todd J Friends
Zhong Sun
Karen A Rossi
Cullen L Cavallaro
Original Assignee
Squibb Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35481430&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MXPA06014642(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Squibb Bristol Myers Co filed Critical Squibb Bristol Myers Co
Publication of MXPA06014642A publication Critical patent/MXPA06014642A/es

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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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US9617224B2 (en) 2017-04-11
KR20070024601A (ko) 2007-03-02
US10112936B2 (en) 2018-10-30
US20140206706A1 (en) 2014-07-24
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US20120088758A1 (en) 2012-04-12
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US20090036438A1 (en) 2009-02-05
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US9079860B2 (en) 2015-07-14
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