JPS61249989A - ７−アミノ−３−プロペニルセフアロスポラン酸及びそのエステル - Google Patents

７−アミノ−３−プロペニルセフアロスポラン酸及びそのエステル

Info

Publication number
JPS61249989A
JPS61249989A JP61091419A JP9141986A JPS61249989A JP S61249989 A JPS61249989 A JP S61249989A JP 61091419 A JP61091419 A JP 61091419A JP 9141986 A JP9141986 A JP 9141986A JP S61249989 A JPS61249989 A JP S61249989A
Authority
JP
Japan
Prior art keywords
group
formula
hydrogen
amino
formulas
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP61091419A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0327554B2 (fi
Inventor
星　英秋
奥村　潤
阿部　芳男
隆之 内藤
油木　慎平
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Co
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of JPS61249989A publication Critical patent/JPS61249989A/ja
Publication of JPH0327554B2 publication Critical patent/JPH0327554B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/18—7-Aminocephalosporanic or substituted 7-aminocephalosporanic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/22—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with radicals containing only hydrogen and carbon atoms, attached in position 3
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
JP61091419A 1985-04-22 1986-04-22 ７−アミノ−３−プロペニルセフアロスポラン酸及びそのエステル Granted JPS61249989A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72587185A 1985-04-22 1985-04-22
US725871 1985-04-22

Publications (2)

Publication Number Publication Date
JPS61249989A true JPS61249989A (ja) 1986-11-07
JPH0327554B2 JPH0327554B2 (fi) 1991-04-16

Family

ID=24916301

Family Applications (1)

Application Number Title Priority Date Filing Date
JP61091419A Granted JPS61249989A (ja) 1985-04-22 1986-04-22 ７−アミノ−３−プロペニルセフアロスポラン酸及びそのエステル

Country Status (38)

Country Link
JP (1) JPS61249989A (fi)
KR (1) KR860008189A (fi)
CN (1) CN1015714B (fi)
AR (1) AR242581A1 (fi)
AT (1) AT392072B (fi)
AU (1) AU589170B2 (fi)
BE (1) BE904646A (fi)
CA (1) CA1273629A (fi)
CH (1) CH671399A5 (fi)
CS (1) CS270435B2 (fi)
CY (1) CY1571A (fi)
DD (1) DD244557A5 (fi)
DE (1) DE3613365A1 (fi)
DK (1) DK163584C (fi)
EG (1) EG18001A (fi)
ES (1) ES8800236A1 (fi)
FI (1) FI84268C (fi)
FR (1) FR2580652B1 (fi)
GB (1) GB2173798B (fi)
GR (1) GR861065B (fi)
HK (1) HK106290A (fi)
HU (1) HU195223B (fi)
IE (1) IE59014B1 (fi)
IT (1) IT1228241B (fi)
LU (1) LU86402A1 (fi)
MY (1) MY100694A (fi)
NL (1) NL192205C (fi)
NO (1) NO164659C (fi)
NZ (1) NZ215717A (fi)
OA (1) OA08245A (fi)
PT (1) PT82436B (fi)
SE (1) SE500217C2 (fi)
SG (1) SG90890G (fi)
SU (1) SU1435155A3 (fi)
YU (1) YU43697B (fi)
ZA (1) ZA862985B (fi)
ZM (1) ZM4286A1 (fi)
ZW (1) ZW9086A1 (fi)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005118595A1 (ja) * 2004-06-04 2005-12-15 Otsuka Chemical Co., Ltd. ３−アルケニルセフェム化合物の製造方法

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4708955A (en) * 1985-06-24 1987-11-24 Bristol-Myers Company 3-(substituted)propenyl-7-aminothiazol-ylcephalosporanic acids and esters thereof
US4870168A (en) * 1987-02-26 1989-09-26 Bristol-Myers Company 3-Unsaturated alkyl cephems from 3-triflyl cephems
DE3933934A1 (de) * 1989-10-03 1991-04-11 Bayer Ag Verfahren zur herstellung von 7-amino-3-((z)-1-propen-1-yl)-3-cephem-4-carbonsaeure
DE69231815T2 (de) * 1991-03-08 2001-09-27 Biochemie Gmbh Verfahren zur Herstellung von Cephalosporinen und Zwischenprodukte in diesem Verfahren
JP2825655B2 (ja) * 1992-02-05 1998-11-18 バイオケミ・ゲゼルシヤフト・エム・ベー・ハー ３−セフェム−４−カルボン酸誘導体の精製方法
AT399876B (de) * 1992-02-05 1995-08-25 Biochemie Gmbh Verfahren zur abreicherung von 7-amino-3-((e)-1- propen-1-yl)-3-cephem-4-carbonsäure
JPH07173168A (ja) * 1993-07-14 1995-07-11 Sumitomo Chem Co Ltd セフェム系化合物、その製法、およびそれのセフェム系抗生物質製造への利用
US20060173176A1 (en) * 2002-10-08 2006-08-03 Yatendra Kumar Process for the preparation of (z)-isomer enriched 7-amino-3-propen-1-yl-3-cephem-4-carboxylic acid
WO2005042543A1 (en) * 2003-10-30 2005-05-12 Cj Corporation Processes for the preparation of cephem derivatives
EP1809638B1 (en) 2004-11-01 2010-02-17 Hetero Drugs Limited A novel process for preparation of cefprozil intermediate
CN103183686B (zh) * 2011-12-30 2016-06-29 浙江新和成股份有限公司 7β-氨基-7α-甲氧基-3-头孢烯化合物的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3769277A (en) * 1970-01-23 1973-10-30 Glaxo Lab Ltd Preparation of delta3-4 carboxy cephalosporins having a 3-vinyl or substituted 3-vinyl group
US4110534A (en) * 1970-01-23 1978-08-29 Glaxo Laboratories Limited Process for the preparation of 3-vinyl and substituted vinyl cephalosporins
GB1342241A (en) * 1970-01-23 1974-01-03 Glaxo Lab Ltd Cephalosporin compounds
US4065620A (en) * 1971-06-14 1977-12-27 Eli Lilly And Company 3-(Substituted) vinyl cephalosporins
US4409214A (en) * 1979-11-19 1983-10-11 Fujisawa Pharmaceutical, Co., Ltd. 7-Acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
US4520022A (en) * 1983-01-28 1985-05-28 Bristol-Myers Company Substituted vinyl cephalosporins
AU566944B2 (en) * 1983-10-07 1987-11-05 Gist-Brocades N.V. Preparation of 3-cephem derivatives

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005118595A1 (ja) * 2004-06-04 2005-12-15 Otsuka Chemical Co., Ltd. ３−アルケニルセフェム化合物の製造方法

Also Published As

Publication number Publication date
KR860008189A (ko) 1986-11-12
SE8601825D0 (sv) 1986-04-21
IE59014B1 (en) 1993-12-15
HUT41033A (en) 1987-03-30
IT8620162A0 (it) 1986-04-21
CY1571A (en) 1991-12-20
EG18001A (en) 1991-11-30
DD244557A5 (de) 1987-04-08
DK163584B (da) 1992-03-16
GB2173798B (en) 1988-11-30
BE904646A (fr) 1986-10-21
NO164659C (no) 1990-10-31
FI861634A0 (fi) 1986-04-17
CS270435B2 (en) 1990-06-13
PT82436B (pt) 1988-11-30
LU86402A1 (fr) 1986-11-05
DE3613365A1 (de) 1987-01-02
SE8601825L (sv) 1986-10-23
PT82436A (en) 1986-05-01
DE3613365C2 (fi) 1989-06-15
ZW9086A1 (en) 1986-12-03
NL192205B (nl) 1996-11-01
IE861048L (en) 1986-10-22
NO861430L (no) 1986-10-23
NL192205C (nl) 1997-03-04
ES554215A0 (es) 1987-10-16
AR242581A1 (es) 1993-04-30
GR861065B (en) 1986-09-01
AU589170B2 (en) 1989-10-05
FI84268C (fi) 1991-11-11
NL8601011A (nl) 1986-11-17
SG90890G (en) 1991-01-18
DK182486A (da) 1986-10-23
YU65986A (en) 1987-12-31
HK106290A (en) 1990-12-28
DK163584C (da) 1992-08-10
JPH0327554B2 (fi) 1991-04-16
CN1015714B (zh) 1992-03-04
DK182486D0 (da) 1986-04-21
AT392072B (de) 1991-01-25
ZM4286A1 (en) 1989-03-27
CN86102630A (zh) 1987-02-04
FR2580652A1 (fr) 1986-10-24
MY100694A (en) 1991-01-17
IT1228241B (it) 1991-06-05
NO164659B (no) 1990-07-23
ATA106786A (de) 1990-07-15
NZ215717A (en) 1989-06-28
ES8800236A1 (es) 1987-10-16
FI861634A (fi) 1986-10-23
CH671399A5 (fi) 1989-08-31
YU43697B (en) 1989-10-31
FR2580652B1 (fr) 1989-01-06
CA1273629A (en) 1990-09-04
CS287286A2 (en) 1989-11-14
FI84268B (fi) 1991-07-31
SU1435155A3 (ru) 1988-10-30
GB8609661D0 (en) 1986-05-29
HU195223B (en) 1988-04-28
AU5616886A (en) 1986-11-06
ZA862985B (en) 1986-12-30
SE500217C2 (sv) 1994-05-09
OA08245A (fr) 1987-10-30
GB2173798A (en) 1986-10-22

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