JPS58201792A - 結晶性の、サルタミシリンのベンゼンスルホン酸塩 - Google Patents

結晶性の、サルタミシリンのベンゼンスルホン酸塩

Info

Publication number
JPS58201792A
JPS58201792A JP58071315A JP7131583A JPS58201792A JP S58201792 A JPS58201792 A JP S58201792A JP 58071315 A JP58071315 A JP 58071315A JP 7131583 A JP7131583 A JP 7131583A JP S58201792 A JPS58201792 A JP S58201792A
Authority
JP
Japan
Prior art keywords
crystalline
acid
salt
salts
water
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP58071315A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0119395B2 (enExample
Inventor
ウエイン・ア−ネスト・バ−ス
バイト−タス・ジヨン・ジヤシス
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of JPS58201792A publication Critical patent/JPS58201792A/ja
Publication of JPH0119395B2 publication Critical patent/JPH0119395B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP58071315A 1982-04-23 1983-04-22 結晶性の、サルタミシリンのベンゼンスルホン酸塩 Granted JPS58201792A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/371,156 US4432987A (en) 1982-04-23 1982-04-23 Crystalline benzenesulfonate salts of sultamicillin
US371156 1999-08-09

Publications (2)

Publication Number Publication Date
JPS58201792A true JPS58201792A (ja) 1983-11-24
JPH0119395B2 JPH0119395B2 (enExample) 1989-04-11

Family

ID=23462725

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58071315A Granted JPS58201792A (ja) 1982-04-23 1983-04-22 結晶性の、サルタミシリンのベンゼンスルホン酸塩

Country Status (27)

Country Link
US (1) US4432987A (enExample)
EP (1) EP0092968B1 (enExample)
JP (1) JPS58201792A (enExample)
KR (1) KR860001279B1 (enExample)
AU (1) AU536854B2 (enExample)
CA (1) CA1187484A (enExample)
CS (1) CS235320B2 (enExample)
DD (1) DD209632A5 (enExample)
DE (1) DE3362502D1 (enExample)
DK (1) DK162168C (enExample)
EG (1) EG16412A (enExample)
ES (1) ES8406075A1 (enExample)
FI (1) FI76092C (enExample)
GR (1) GR78582B (enExample)
HK (1) HK20588A (enExample)
HU (1) HU187068B (enExample)
IE (1) IE54628B1 (enExample)
IL (1) IL68453A (enExample)
NO (1) NO156202C (enExample)
NZ (1) NZ203988A (enExample)
PH (1) PH18035A (enExample)
PL (1) PL134978B1 (enExample)
PT (1) PT76587B (enExample)
SG (1) SG104087G (enExample)
SU (1) SU1138030A3 (enExample)
YU (1) YU43170B (enExample)
ZA (1) ZA832845B (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007509973A (ja) * 2003-10-31 2007-04-19 アルザ・コーポレーシヨン 増強された吸収のための組成物および投与形態物
US7304166B2 (en) 2002-08-29 2007-12-04 Taisho Pharmaceutical Co., Ltd. Benzenesulfonate salt of 4-fluoro-2-cyanopyrrolidine derivatives

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AU6621586A (en) * 1985-11-18 1987-06-02 University Of Texas System, The Polychelating agents for image and spectral enhancement (and spectral shift)
US5336762A (en) * 1985-11-18 1994-08-09 Access Pharmaceuticals, Inc. Polychelating agents for image and spectral enhancement (and spectral shift)
KR910009271B1 (ko) * 1989-06-20 1991-11-08 김영설 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
US6111098A (en) * 1994-05-02 2000-08-29 Shionogi & Co., Ltd. Crystal of pyrrolidylthiocarbapenem derivative, lyophilized preparation containing said crystal, and process for producing the same
JP3382159B2 (ja) * 1998-08-05 2003-03-04 株式会社東芝 情報記録媒体とその再生方法及び記録方法
MXPA05010083A (es) * 2003-03-27 2005-11-23 Basilea Pharmaceutica Ag Cefalosporina en forma cristalina.
FR2877696B1 (fr) 2004-11-09 2009-09-18 Renault Sas Dispositif et procede d'estimation en temps reel de l'angle de debut de combustion d'un moteur a combustion interne
BRPI0815591B8 (pt) 2007-08-22 2021-05-25 Astrazeneca Ab composto, composição farmacêutica, e, uso de um composto.
TWI469971B (zh) 2007-10-26 2015-01-21 Univ California 二芳基乙內醯脲類化合物
NZ594064A (en) * 2009-01-30 2012-08-31 Glaxosmithkline Llc Crystalline n-{ (1s)-2-amino-1-[(3-fluorophenyl)methyl]ethyl} -5-chloro-4-(4-chloro-1-methyl-1h-pyrazol-5-yl)-2-thiophenecarboxamide hydrochloride
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
KR20120079054A (ko) * 2009-07-10 2012-07-11 에볼바 아게 디인 조성물
MX2012009537A (es) * 2010-02-18 2012-08-31 Astrazeneca Ab Formas solidas que comprenden un derivado de ciclopropilamida.
AU2011218491C1 (en) * 2010-02-18 2015-05-14 Astrazeneca Ab Processes for making cyclopropyl amide derivatives and intermediates associated therewith
JP6310396B2 (ja) * 2012-12-03 2018-04-11 株式会社カネカ 還元型補酵素ｑ１０誘導体およびその製造方法
TWI637943B (zh) * 2013-09-05 2018-10-11 田邊三菱製藥股份有限公司 新穎結晶性芳烷基胺化合物及其製造方法
PT3209647T (pt) 2014-10-21 2020-09-10 Ariad Pharma Inc Formas cristalinas de 5-cloro-n4-[2-(dimetilfosforil)fenil]-n2-{2-metoxi-4-[4-(4-metilpiperazin-1-il)piperidin-1-il]pirimidino-2,4-diamina
CN104958318A (zh) * 2015-08-04 2015-10-07 青岛蓝盛洋医药生物科技有限责任公司 一种治疗感染性疾病的药物舒巴坦钠组合物
WO2017125557A1 (en) * 2016-01-22 2017-07-27 Sandoz Ag Crystalline eravacycline bis-hydrochloride
EA039753B1 (ru) * 2016-07-07 2022-03-10 Сайклерион Терапьютикс, Инк. ТВЕРДЫЕ ФОРМЫ СТИМУЛЯТОРА sGC
EP3703686A4 (en) * 2017-10-30 2021-11-17 Theracaine LLC HYDROPHOBIC ARENE SULFONATE SALTS
US11186556B1 (en) * 2018-10-16 2021-11-30 Celgene Corporation Salts of a thiazolidinone compound, solid forms, compositions and methods of use thereof
UA119735C2 (uk) 2018-12-20 2019-07-25 Анатолій Семенович Редер Фармацевтична сполука, спосіб її отримання та застосування як лікарського засобу
USD1071069S1 (en) 2019-02-13 2025-04-15 Hs Produkt D.O.O. Stippled textured body for a firearm or the like
USD998740S1 (en) 2019-02-13 2023-09-12 Hs Produkt D.O.O. Firearm
USD1126349S1 (en) 2019-02-13 2026-05-12 Hs Produkt D.O.O. Firearm sight
USD994822S1 (en) 2019-02-13 2023-08-08 Hs Produkt D.O.O. Pistol
USD994821S1 (en) 2019-02-13 2023-08-08 Hs Produkt D.O.O. Pistol
USD1057880S1 (en) 2019-08-09 2025-01-14 Hs Produkt D.O.O. Pistol
CN117120034A (zh) * 2021-02-15 2023-11-24 普洛佩拉治疗公司 阿比特龙前药
CN117242070A (zh) * 2021-03-01 2023-12-15 奥仁公司 4h-吡喃-4-酮结构化cyp11a1抑制剂的固体形式
USD1049292S1 (en) * 2021-04-06 2024-10-29 Springfield, Inc. Pistol
JP7645573B2 (ja) * 2021-05-12 2025-03-14 ジャージアン・ロングチャーム・バイオ－テック・ファーマ・カンパニー・リミテッド ピロロピリミジン類化合物の結晶形およびその調製方法
BR112023021606A2 (pt) * 2021-05-14 2023-12-19 Global Blood Therapeutics Inc Formas sólidas de modulador de hemoglobina
US20240287066A1 (en) * 2021-06-24 2024-08-29 Sandoz Ag Crystalline Form of Sotorasib
USD1069964S1 (en) 2021-11-03 2025-04-08 Hs Produkt D.O.O. Pistol slide
WO2023125700A1 (zh) * 2021-12-28 2023-07-06 南京明德新药研发有限公司 四氢环庚吲唑化合物的盐型、晶型
IL314212A (en) * 2022-01-10 2024-09-01 Azafaros B V Treatment of GM2 gangliosidosis
CA3253725A1 (en) * 2022-05-20 2023-11-23 Caamtech, Inc. TRYPTAMINE DERIVATIVES
USD1057882S1 (en) 2022-08-29 2025-01-14 Springfield, Inc. Combined serrations for a firearm slide
USD1072997S1 (en) 2022-08-29 2025-04-29 Springfield, Inc. Firearm
USD1061781S1 (en) 2022-11-30 2025-02-11 Hs Produkt D.O.O. Pistol
US20240217985A1 (en) * 2022-12-22 2024-07-04 Boehringer Ingelheim International Gmbh CRYSTALLINE FORM OF AN MDM2-p53 INHIBITOR AND PHARMACEUTICAL COMPOSITIONS
ZAA202301171S (en) 2023-04-28 2024-09-25 Hs Produkt D O O Firearm
IL325861A (en) * 2023-07-17 2026-03-01 Kura Oncology Inc Crystalline forms of a menin inhibitor
JP2026525148A (ja) * 2023-07-17 2026-07-29 クラ オンコロジー，インク． メニン阻害剤を含む医薬組成物
USD1127974S1 (en) 2024-01-22 2026-05-26 Rost Martin LLC Firearm
USD1128830S1 (en) 2024-01-22 2026-06-02 Rost Martin LLC Firearm

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55113790A (en) * 1979-02-13 1980-09-02 Leo Pharm Prod Ltd Novel penicillanic ester derivative and its manufacture and use
GB2084572A (en) * 1980-10-06 1982-04-15 Leo Pharm Prod Ltd 1,1-Dioxopenicillanoyloxymethyl 6-(D- alpha -amino- alpha -phenylacetamido)penicillanate napsylate

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate
IL64009A (en) * 1980-10-31 1984-09-30 Rech Applications Therap Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55113790A (en) * 1979-02-13 1980-09-02 Leo Pharm Prod Ltd Novel penicillanic ester derivative and its manufacture and use
GB2084572A (en) * 1980-10-06 1982-04-15 Leo Pharm Prod Ltd 1,1-Dioxopenicillanoyloxymethyl 6-(D- alpha -amino- alpha -phenylacetamido)penicillanate napsylate

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7304166B2 (en) 2002-08-29 2007-12-04 Taisho Pharmaceutical Co., Ltd. Benzenesulfonate salt of 4-fluoro-2-cyanopyrrolidine derivatives
JP2007509973A (ja) * 2003-10-31 2007-04-19 アルザ・コーポレーシヨン 増強された吸収のための組成物および投与形態物

Also Published As

Publication number Publication date
FI76092B (fi) 1988-05-31
FI76092C (fi) 1988-09-09
NO156202C (no) 1987-08-19
PH18035A (en) 1985-03-06
FI831392L (fi) 1983-10-24
EG16412A (en) 1989-03-30
GR78582B (enExample) 1984-09-27
ES521728A0 (es) 1984-07-01
ZA832845B (en) 1984-11-28
DK101783D0 (da) 1983-02-28
KR860001279B1 (ko) 1986-09-05
IL68453A0 (en) 1983-07-31
IL68453A (en) 1986-08-31
PL134978B1 (en) 1985-09-30
SG104087G (en) 1988-07-15
AU536854B2 (en) 1984-05-24
EP0092968B1 (en) 1986-03-12
CA1187484A (en) 1985-05-21
JPH0119395B2 (enExample) 1989-04-11
FI831392A0 (fi) 1983-04-22
CS235320B2 (en) 1985-05-15
IE830926L (en) 1983-10-23
PL241553A1 (en) 1983-11-21
DK101783A (da) 1983-10-24
HK20588A (en) 1988-03-25
KR840004437A (ko) 1984-10-15
YU43170B (en) 1989-04-30
SU1138030A3 (ru) 1985-01-30
US4432987A (en) 1984-02-21
DE3362502D1 (en) 1986-04-17
IE54628B1 (en) 1989-12-20
DK162168C (da) 1992-03-02
PT76587A (en) 1983-05-01
DD209632A5 (de) 1984-05-16
EP0092968A1 (en) 1983-11-02
HU187068B (en) 1985-11-28
NO831430L (no) 1983-10-24
NZ203988A (en) 1986-01-24
PT76587B (en) 1986-02-27
AU1387183A (en) 1983-11-17
YU90483A (en) 1986-04-30
DK162168B (da) 1991-09-23
NO156202B (no) 1987-05-04
ES8406075A1 (es) 1984-07-01

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