JPH0119395B2 - - Google Patents

Info

Publication number
JPH0119395B2
JPH0119395B2 JP58071315A JP7131583A JPH0119395B2 JP H0119395 B2 JPH0119395 B2 JP H0119395B2 JP 58071315 A JP58071315 A JP 58071315A JP 7131583 A JP7131583 A JP 7131583A JP H0119395 B2 JPH0119395 B2 JP H0119395B2
Authority
JP
Japan
Prior art keywords
crystalline
salt
salts
formula
water
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP58071315A
Other languages
English (en)
Japanese (ja)
Other versions
JPS58201792A (ja
Inventor
Aanesuto Baasu Uein
Jon Jashisu Baitootasu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Original Assignee
Pfizer Corp Belgium
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium filed Critical Pfizer Corp Belgium
Publication of JPS58201792A publication Critical patent/JPS58201792A/ja
Publication of JPH0119395B2 publication Critical patent/JPH0119395B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP58071315A 1982-04-23 1983-04-22 結晶性の、サルタミシリンのベンゼンスルホン酸塩 Granted JPS58201792A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/371,156 US4432987A (en) 1982-04-23 1982-04-23 Crystalline benzenesulfonate salts of sultamicillin
US371156 1982-04-23

Publications (2)

Publication Number Publication Date
JPS58201792A JPS58201792A (ja) 1983-11-24
JPH0119395B2 true JPH0119395B2 (enExample) 1989-04-11

Family

ID=23462725

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58071315A Granted JPS58201792A (ja) 1982-04-23 1983-04-22 結晶性の、サルタミシリンのベンゼンスルホン酸塩

Country Status (27)

Country Link
US (1) US4432987A (enExample)
EP (1) EP0092968B1 (enExample)
JP (1) JPS58201792A (enExample)
KR (1) KR860001279B1 (enExample)
AU (1) AU536854B2 (enExample)
CA (1) CA1187484A (enExample)
CS (1) CS235320B2 (enExample)
DD (1) DD209632A5 (enExample)
DE (1) DE3362502D1 (enExample)
DK (1) DK162168C (enExample)
EG (1) EG16412A (enExample)
ES (1) ES521728A0 (enExample)
FI (1) FI76092C (enExample)
GR (1) GR78582B (enExample)
HK (1) HK20588A (enExample)
HU (1) HU187068B (enExample)
IE (1) IE54628B1 (enExample)
IL (1) IL68453A (enExample)
NO (1) NO156202C (enExample)
NZ (1) NZ203988A (enExample)
PH (1) PH18035A (enExample)
PL (1) PL134978B1 (enExample)
PT (1) PT76587B (enExample)
SG (1) SG104087G (enExample)
SU (1) SU1138030A3 (enExample)
YU (1) YU43170B (enExample)
ZA (1) ZA832845B (enExample)

Families Citing this family (44)

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EP0247156B1 (en) * 1985-11-18 1993-06-23 Access Pharmaceuticals Inc. Polychelating agents for image and spectral enhancement (and spectral shift)
US5336762A (en) * 1985-11-18 1994-08-09 Access Pharmaceuticals, Inc. Polychelating agents for image and spectral enhancement (and spectral shift)
KR910009271B1 (ko) * 1989-06-20 1991-11-08 김영설 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
CN1048248C (zh) * 1994-05-02 2000-01-12 盐野义制药株式会社 吡咯烷基硫基碳代青霉烯衍生物的结晶、含该结晶的冷冻干燥制剂及其制造方法
JP3382159B2 (ja) * 1998-08-05 2003-03-04 株式会社東芝 情報記録媒体とその再生方法及び記録方法
PL374664A1 (en) 2002-08-29 2005-10-31 Taisho Pharmaceutical Co, Ltd. Benzenesulfonate of 4-fluoro-2-cyanopyrrolidine derivative
JP5230934B2 (ja) * 2003-03-27 2013-07-10 バジリア ファルマスーチカ アーゲー 結晶形態のセファロスポリン
CA2543945A1 (en) * 2003-10-31 2005-05-12 Alza Corporation Compositions and dosage forms for enhanced absorption of 3-amino-n-butyl-phosphinic acid
FR2877696B1 (fr) 2004-11-09 2009-09-18 Renault Sas Dispositif et procede d'estimation en temps reel de l'angle de debut de combustion d'un moteur a combustion interne
WO2009024823A2 (en) 2007-08-22 2009-02-26 Astrazeneca Ab Oxadiazole derivatives as dgat inhibitors
AR069039A1 (es) 2007-10-26 2009-12-23 Univ California Compuestos de diarilhidantoina, composicion farmaceutica, proceso de obtencion del compuesto, utiles para desordenes hiperproliferativos
CN102405047B (zh) * 2009-01-30 2014-07-09 葛兰素史密斯克莱有限责任公司 结晶型的n-{(1s)-2-氨基-1-[(3-氟苯基)甲基]乙基}-5-氯-4-(4-氯-1-甲基-1h-吡唑-5-基)-2-噻吩甲酰胺盐酸盐
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
WO2011006061A1 (en) * 2009-07-10 2011-01-13 Evolva Sa Diyne compositions
MX2012009473A (es) * 2010-02-18 2012-09-12 Astrazeneca Ab Procesos para preparar derivados de ciclopropilamidas e intermedios asociados con estas.
MX2012009537A (es) * 2010-02-18 2012-08-31 Astrazeneca Ab Formas solidas que comprenden un derivado de ciclopropilamida.
CN104903289B (zh) * 2012-12-03 2017-06-09 株式会社钟化 还元型辅酶q10衍生物及其制造方法
US9643920B2 (en) * 2013-09-05 2017-05-09 Mitsubishi Tanabe Pharma Corporation Crystalline 4-(3S-(1R-(1-napthyl)ethylamino)pyrrolidin-1-yl)phenylacetic acid
PT3209647T (pt) 2014-10-21 2020-09-10 Ariad Pharma Inc Formas cristalinas de 5-cloro-n4-[2-(dimetilfosforil)fenil]-n2-{2-metoxi-4-[4-(4-metilpiperazin-1-il)piperidin-1-il]pirimidino-2,4-diamina
CN104958318A (zh) * 2015-08-04 2015-10-07 青岛蓝盛洋医药生物科技有限责任公司 一种治疗感染性疾病的药物舒巴坦钠组合物
EP3778567A1 (en) * 2016-01-22 2021-02-17 Sandoz Ag Crystalline eravacycline bis-hydrochloride
EA039753B1 (ru) * 2016-07-07 2022-03-10 Сайклерион Терапьютикс, Инк. ТВЕРДЫЕ ФОРМЫ СТИМУЛЯТОРА sGC
WO2019089540A1 (en) * 2017-10-30 2019-05-09 Theracaine Llc Hydrophobic arenesulfonate salts
US11186556B1 (en) * 2018-10-16 2021-11-30 Celgene Corporation Salts of a thiazolidinone compound, solid forms, compositions and methods of use thereof
UA119735C2 (uk) 2018-12-20 2019-07-25 Анатолій Семенович Редер Фармацевтична сполука, спосіб її отримання та застосування як лікарського засобу
USD994821S1 (en) 2019-02-13 2023-08-08 Hs Produkt D.O.O. Pistol
USD1077123S1 (en) 2019-02-13 2025-05-27 Hs Produkt D.O.O. Firearm sight
USD998740S1 (en) 2019-02-13 2023-09-12 Hs Produkt D.O.O. Firearm
USD994822S1 (en) 2019-02-13 2023-08-08 Hs Produkt D.O.O. Pistol
USD1071069S1 (en) 2019-02-13 2025-04-15 Hs Produkt D.O.O. Stippled textured body for a firearm or the like
USD1057880S1 (en) 2019-08-09 2025-01-14 Hs Produkt D.O.O. Pistol
CA3207282A1 (en) * 2021-02-15 2022-08-18 Matthew J. Sharp Abiraterone prodrugs
USD1049292S1 (en) * 2021-04-06 2024-10-29 Springfield, Inc. Pistol
WO2022237808A1 (zh) * 2021-05-12 2022-11-17 浙江龙传生物医药科技有限公司 吡咯并嘧啶类化合物的晶型及其制备方法
BR112023021606A2 (pt) * 2021-05-14 2023-12-19 Global Blood Therapeutics Inc Formas sólidas de modulador de hemoglobina
USD1069964S1 (en) 2021-11-03 2025-04-08 Hs Produkt D.O.O. Pistol slide
US12410155B2 (en) * 2021-12-28 2025-09-09 Zhejiang Yangli Pharmaceutical Technology Co., Ltd. Salt form and crystal form of tetrahydrocyclohepta indazole compound
CA3253725A1 (en) * 2022-05-20 2023-11-23 Caamtech, Inc. TRYPTAMINE DERIVATIVES
USD1072997S1 (en) 2022-08-29 2025-04-29 Springfield, Inc. Firearm
USD1057882S1 (en) 2022-08-29 2025-01-14 Springfield, Inc. Combined serrations for a firearm slide
USD1061781S1 (en) 2022-11-30 2025-02-11 Hs Produkt D.O.O. Pistol
ZAA202301170S (en) 2023-04-28 2024-06-26 Hs Produkt D O O Firearm
WO2025016385A1 (en) * 2023-07-17 2025-01-23 Kura Oncology, Inc. Pharmaceutical compositions comprising a menin inhibitor
AU2024292586A1 (en) * 2023-07-17 2026-01-29 Kura Oncology, Inc. Crystalline forms of a menin inhibitor

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
ZA80796B (en) * 1979-02-13 1981-02-25 Leo Pharm Prod Ltd Chemical compounds
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate
GB2084572B (en) * 1980-10-06 1984-07-11 Leo Pharm Prod Ltd 1,1-dioxopenicillanoyloxymethyl 6-(d-aphenylacetamido)penicillanate napsylate
IL64009A (en) * 1980-10-31 1984-09-30 Rech Applications Therap Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
EG16412A (en) 1989-03-30
SG104087G (en) 1988-07-15
DK162168C (da) 1992-03-02
IL68453A (en) 1986-08-31
EP0092968A1 (en) 1983-11-02
PH18035A (en) 1985-03-06
KR860001279B1 (ko) 1986-09-05
ES8406075A1 (es) 1984-07-01
DE3362502D1 (en) 1986-04-17
CA1187484A (en) 1985-05-21
FI831392A0 (fi) 1983-04-22
DD209632A5 (de) 1984-05-16
FI76092B (fi) 1988-05-31
EP0092968B1 (en) 1986-03-12
YU43170B (en) 1989-04-30
DK101783D0 (da) 1983-02-28
NO156202B (no) 1987-05-04
IE830926L (en) 1983-10-23
GR78582B (enExample) 1984-09-27
HU187068B (en) 1985-11-28
FI76092C (fi) 1988-09-09
SU1138030A3 (ru) 1985-01-30
PT76587B (en) 1986-02-27
HK20588A (en) 1988-03-25
US4432987A (en) 1984-02-21
CS235320B2 (en) 1985-05-15
AU1387183A (en) 1983-11-17
PL241553A1 (en) 1983-11-21
FI831392L (fi) 1983-10-24
JPS58201792A (ja) 1983-11-24
IE54628B1 (en) 1989-12-20
ES521728A0 (es) 1984-07-01
NO156202C (no) 1987-08-19
YU90483A (en) 1986-04-30
NO831430L (no) 1983-10-24
NZ203988A (en) 1986-01-24
PL134978B1 (en) 1985-09-30
PT76587A (en) 1983-05-01
DK101783A (da) 1983-10-24
IL68453A0 (en) 1983-07-31
ZA832845B (en) 1984-11-28
DK162168B (da) 1991-09-23
KR840004437A (ko) 1984-10-15
AU536854B2 (en) 1984-05-24

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