AU536854B2 - 1 1-dioxopenicillanoyl methyl penicillanate esters - Google Patents

1 1-dioxopenicillanoyl methyl penicillanate esters

Info

Publication number
AU536854B2
AU536854B2 AU13871/83A AU1387183A AU536854B2 AU 536854 B2 AU536854 B2 AU 536854B2 AU 13871/83 A AU13871/83 A AU 13871/83A AU 1387183 A AU1387183 A AU 1387183A AU 536854 B2 AU536854 B2 AU 536854B2
Authority
AU
Australia
Prior art keywords
dioxopenicillanoyl
esters
methyl penicillanate
penicillanate
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU13871/83A
Other languages
English (en)
Other versions
AU1387183A (en
Inventor
Wayne Ernest Barth
Vytautas John Jasys
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Publication of AU1387183A publication Critical patent/AU1387183A/en
Application granted granted Critical
Publication of AU536854B2 publication Critical patent/AU536854B2/en
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
AU13871/83A 1982-04-23 1983-04-22 1 1-dioxopenicillanoyl methyl penicillanate esters Expired AU536854B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US371156 1982-04-23
US06/371,156 US4432987A (en) 1982-04-23 1982-04-23 Crystalline benzenesulfonate salts of sultamicillin

Publications (2)

Publication Number Publication Date
AU1387183A AU1387183A (en) 1983-11-17
AU536854B2 true AU536854B2 (en) 1984-05-24

Family

ID=23462725

Family Applications (1)

Application Number Title Priority Date Filing Date
AU13871/83A Expired AU536854B2 (en) 1982-04-23 1983-04-22 1 1-dioxopenicillanoyl methyl penicillanate esters

Country Status (27)

Country Link
US (1) US4432987A (enExample)
EP (1) EP0092968B1 (enExample)
JP (1) JPS58201792A (enExample)
KR (1) KR860001279B1 (enExample)
AU (1) AU536854B2 (enExample)
CA (1) CA1187484A (enExample)
CS (1) CS235320B2 (enExample)
DD (1) DD209632A5 (enExample)
DE (1) DE3362502D1 (enExample)
DK (1) DK162168C (enExample)
EG (1) EG16412A (enExample)
ES (1) ES8406075A1 (enExample)
FI (1) FI76092C (enExample)
GR (1) GR78582B (enExample)
HK (1) HK20588A (enExample)
HU (1) HU187068B (enExample)
IE (1) IE54628B1 (enExample)
IL (1) IL68453A (enExample)
NO (1) NO156202C (enExample)
NZ (1) NZ203988A (enExample)
PH (1) PH18035A (enExample)
PL (1) PL134978B1 (enExample)
PT (1) PT76587B (enExample)
SG (1) SG104087G (enExample)
SU (1) SU1138030A3 (enExample)
YU (1) YU43170B (enExample)
ZA (1) ZA832845B (enExample)

Families Citing this family (42)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH07110815B2 (ja) * 1985-11-18 1995-11-29 ボ−ド・オブ・リ−ジェンツ、ザ・ユニバ−シティ−・オブ・テキサス・システム 画像及びスペクトル向上（およびスペクトルシフト）のためのポリキレ−ト剤
US5336762A (en) * 1985-11-18 1994-08-09 Access Pharmaceuticals, Inc. Polychelating agents for image and spectral enhancement (and spectral shift)
KR910009271B1 (ko) * 1989-06-20 1991-11-08 김영설 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
ATE223916T1 (de) * 1994-05-02 2002-09-15 Shionogi & Co Kristalline pyrrolidylthiocarbapenem derivate, lyophilisierste präparationen dieser kristalle und verfahren zu deren herstellung
JP3382159B2 (ja) * 1998-08-05 2003-03-04 株式会社東芝 情報記録媒体とその再生方法及び記録方法
EP1535907A4 (en) 2002-08-29 2006-11-29 Taisho Pharmaceutical Co Ltd BENZOLSULFONATE OF A 4-FLUORO-2-CYANOPYRROLIDINE DERIVATIVE
CA2519272C (en) * 2003-03-27 2010-06-08 Basilea Pharmaceutica Ag Cephalosporin in crystalline form
JP2007509975A (ja) * 2003-10-31 2007-04-19 アルザ・コーポレーシヨン ギャバペンチン及びプレギャバリンの増加された吸収のための組成物及び投与形態物
FR2877696B1 (fr) 2004-11-09 2009-09-18 Renault Sas Dispositif et procede d'estimation en temps reel de l'angle de debut de combustion d'un moteur a combustion interne
SA08290520B1 (ar) 2007-08-22 2012-02-22 استرازينيكا ايه بي مشتقات سيكلو بروبيل أميد وتركيبات صيدلية تحتوي عليها لعلاج حالة مرضية سببها مستقبلات هيستامين h3
JP5535925B2 (ja) 2007-10-26 2014-07-02 ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア アンドロゲン受容体調節物質としてのジアリールヒダントイン化合物
BRPI1006896B1 (pt) * 2009-01-30 2022-05-24 Novartis Ag Cloridrato de n-{(1s)-2-amino-1-[(3-fluorfenil)metil]etil}-5-cloro-4-(4-cloro-1-metil-1h- pirazol-5-il)-2-tiofenocarboxamida cristalino, composição farmacêutica compreendendo o mesmo e uso do dito composto para tratar ou diminuir a gravidade de câncer e artrite
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
KR20120079054A (ko) * 2009-07-10 2012-07-11 에볼바 아게 디인 조성물
MX2012009537A (es) * 2010-02-18 2012-08-31 Astrazeneca Ab Formas solidas que comprenden un derivado de ciclopropilamida.
SG10201501226VA (en) * 2010-02-18 2015-04-29 Astrazeneca Ab New crystalline form of a cyclopropyl benzamide derivative
CN104903289B (zh) * 2012-12-03 2017-06-09 株式会社钟化 还元型辅酶q10衍生物及其制造方法
EP3360858B1 (en) * 2013-09-05 2020-04-29 Mitsubishi Tanabe Pharma Corporation Process for producing an aminopyrrolidine derivative
CR20170146A (es) * 2014-10-21 2017-08-10 Ariad Pharma Inc Formas cristalinas de 5-cloro-n4-[-2-(dimetilfosforil)fenil]-n2-{2-metoxi-4-[4-(4-metilpiperazin-1-yl)piperidin-1-il]pirimidina-2,4-diamina
CN104958318A (zh) * 2015-08-04 2015-10-07 青岛蓝盛洋医药生物科技有限责任公司 一种治疗感染性疾病的药物舒巴坦钠组合物
WO2017125557A1 (en) * 2016-01-22 2017-07-27 Sandoz Ag Crystalline eravacycline bis-hydrochloride
KR102803160B1 (ko) * 2016-07-07 2025-04-30 사이클리온 테라퓨틱스, 인크. sGC 자극제의 고체 형태
EP3703686A4 (en) * 2017-10-30 2021-11-17 Theracaine LLC HYDROPHOBIC ARENE SULFONATE SALTS
US11186556B1 (en) * 2018-10-16 2021-11-30 Celgene Corporation Salts of a thiazolidinone compound, solid forms, compositions and methods of use thereof
UA119735C2 (uk) 2018-12-20 2019-07-25 Анатолій Семенович Редер Фармацевтична сполука, спосіб її отримання та застосування як лікарського засобу
USD1077123S1 (en) 2019-02-13 2025-05-27 Hs Produkt D.O.O. Firearm sight
USD994822S1 (en) 2019-02-13 2023-08-08 Hs Produkt D.O.O. Pistol
USD994821S1 (en) 2019-02-13 2023-08-08 Hs Produkt D.O.O. Pistol
USD998740S1 (en) 2019-02-13 2023-09-12 Hs Produkt D.O.O. Firearm
USD1071069S1 (en) 2019-02-13 2025-04-15 Hs Produkt D.O.O. Stippled textured body for a firearm or the like
USD1057880S1 (en) 2019-08-09 2025-01-14 Hs Produkt D.O.O. Pistol
EP4291159A1 (en) * 2021-02-15 2023-12-20 Propella Therapeutics, Inc. Abiraterone prodrugs
USD1049292S1 (en) * 2021-04-06 2024-10-29 Springfield, Inc. Pistol
AR126649A1 (es) * 2021-05-14 2023-11-01 Global Blood Therapeutics Inc Formas sólidas de un modulador de hemoglobina
USD1069964S1 (en) 2021-11-03 2025-04-08 Hs Produkt D.O.O. Pistol slide
WO2023125700A1 (zh) * 2021-12-28 2023-07-06 南京明德新药研发有限公司 四氢环庚吲唑化合物的盐型、晶型
USD1057882S1 (en) 2022-08-29 2025-01-14 Springfield, Inc. Combined serrations for a firearm slide
USD1072997S1 (en) 2022-08-29 2025-04-29 Springfield, Inc. Firearm
USD1061781S1 (en) 2022-11-30 2025-02-11 Hs Produkt D.O.O. Pistol
ZAA202301172S (en) 2023-04-28 2024-06-26 Hs Produkt D O O Firearm
TW202517651A (zh) * 2023-07-17 2025-05-01 美商庫拉腫瘤技術股份有限公司 Menin抑制劑之晶型
TW202517650A (zh) * 2023-07-17 2025-05-01 美商庫拉腫瘤技術股份有限公司 包含ｍｅｎｉｎ抑制劑之醫藥組合物

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
BE881675A (fr) * 1979-02-13 1980-08-12 Leo Pharm Prod Ltd B-lactames derives de l'acide penicillanique leur preparation et leurs utilisations therapeutiques
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate
GB2084572B (en) * 1980-10-06 1984-07-11 Leo Pharm Prod Ltd 1,1-dioxopenicillanoyloxymethyl 6-(d-aphenylacetamido)penicillanate napsylate
IL64009A (en) * 1980-10-31 1984-09-30 Rech Applications Therap Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
EP0092968A1 (en) 1983-11-02
PH18035A (en) 1985-03-06
EP0092968B1 (en) 1986-03-12
PL241553A1 (en) 1983-11-21
FI76092B (fi) 1988-05-31
PL134978B1 (en) 1985-09-30
DD209632A5 (de) 1984-05-16
IE54628B1 (en) 1989-12-20
KR840004437A (ko) 1984-10-15
DK101783A (da) 1983-10-24
GR78582B (enExample) 1984-09-27
EG16412A (en) 1989-03-30
YU43170B (en) 1989-04-30
DK101783D0 (da) 1983-02-28
ZA832845B (en) 1984-11-28
IL68453A0 (en) 1983-07-31
FI831392A0 (fi) 1983-04-22
HU187068B (en) 1985-11-28
PT76587B (en) 1986-02-27
DK162168B (da) 1991-09-23
YU90483A (en) 1986-04-30
CA1187484A (en) 1985-05-21
JPH0119395B2 (enExample) 1989-04-11
ES521728A0 (es) 1984-07-01
DE3362502D1 (en) 1986-04-17
PT76587A (en) 1983-05-01
NO156202C (no) 1987-08-19
IL68453A (en) 1986-08-31
SG104087G (en) 1988-07-15
FI76092C (fi) 1988-09-09
SU1138030A3 (ru) 1985-01-30
US4432987A (en) 1984-02-21
ES8406075A1 (es) 1984-07-01
IE830926L (en) 1983-10-23
DK162168C (da) 1992-03-02
KR860001279B1 (ko) 1986-09-05
HK20588A (en) 1988-03-25
FI831392L (fi) 1983-10-24
AU1387183A (en) 1983-11-17
NO156202B (no) 1987-05-04
NO831430L (no) 1983-10-24
NZ203988A (en) 1986-01-24
CS235320B2 (en) 1985-05-15
JPS58201792A (ja) 1983-11-24

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Legal Events

Date Code Title Description
MK14 Patent ceased section 143(a) (annual fees not paid) or expired