JPS55113790A - Novel penicillanic ester derivative and its manufacture and use - Google Patents

Novel penicillanic ester derivative and its manufacture and use

Info

Publication number
JPS55113790A
JPS55113790A JP1719780A JP1719780A JPS55113790A JP S55113790 A JPS55113790 A JP S55113790A JP 1719780 A JP1719780 A JP 1719780A JP 1719780 A JP1719780 A JP 1719780A JP S55113790 A JPS55113790 A JP S55113790A
Authority
JP
Japan
Prior art keywords
manufacture
ester derivative
novel
novel penicillanic
penicillanic ester
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1719780A
Other languages
Japanese (ja)
Other versions
JPS6259709B2 (en
Inventor
Wagn O Godtfredsen
Daehne Welf Von
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Leo Pharma AS
Original Assignee
Leo Pharmaceutical Products Ltd AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharmaceutical Products Ltd AS filed Critical Leo Pharmaceutical Products Ltd AS
Publication of JPS55113790A publication Critical patent/JPS55113790A/en
Publication of JPS6259709B2 publication Critical patent/JPS6259709B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D503/00—Heterocyclic compounds containing 4-oxa-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxapenicillins, clavulanic acid derivatives; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
JP1719780A 1979-02-13 1980-02-13 Novel penicillanic ester derivative and its manufacture and use Granted JPS55113790A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7905020 1979-02-13

Publications (2)

Publication Number Publication Date
JPS55113790A true JPS55113790A (en) 1980-09-02
JPS6259709B2 JPS6259709B2 (en) 1987-12-12

Family

ID=10503160

Family Applications (2)

Application Number Title Priority Date Filing Date
JP1719780A Granted JPS55113790A (en) 1979-02-13 1980-02-13 Novel penicillanic ester derivative and its manufacture and use
JP62114399A Granted JPS62281879A (en) 1979-02-13 1987-05-11 Beta-lactam intermediate and its production

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP62114399A Granted JPS62281879A (en) 1979-02-13 1987-05-11 Beta-lactam intermediate and its production

Country Status (4)

Country Link
JP (2) JPS55113790A (en)
KR (1) KR830001903B1 (en)
BE (1) BE881675A (en)
ZA (1) ZA80796B (en)

Cited By (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55157589A (en) * 1979-05-16 1980-12-08 Pfizer Penicillins of methanediol and bisester of methanediol and penicillanic acid 1*11dioxide
JPS57126493A (en) * 1980-10-31 1982-08-06 Leo Pharm Prod Ltd Cryatal hydrate of penicillanic acid derivative salt, manufacture and use
JPS57169493A (en) * 1981-03-23 1982-10-19 Pfizer 6-(2-amino-2-phenylacetamide)penicillanic acid 1,1-dioxopenicillanoyloxymethyl, manufacture and intermediate
JPS57169486A (en) * 1981-03-23 1982-10-19 Pfizer Manufacture of halomethyl ester ( and related ester) of penicillanic acid 1,1-dioxide
JPS57176989A (en) * 1981-03-23 1982-10-30 Pfizer Improvement on manufacture of penicillanic acid esters
JPS5857384A (en) * 1981-09-09 1983-04-05 フアイザ−・インコ−ポレ−テツド Antibacterial penicillanic acid 6'-(2-amino- 2-(4-acyloxyphenyl)acetamide)penicillanoyloxymethyl- 1,1-dioxide compound
JPS5862179A (en) * 1981-09-18 1983-04-13 フアイザ−・インコ−ポレ−テツド Antibacterial ester of resolcine, ampicillin and penicillanic acid 1,1-dioxide derivative
JPS58116490A (en) * 1981-12-22 1983-07-11 フアイザ−・インコ−ポレ−テツド Antibacterial bridged with bis-hydroxymethyl carbonate
JPS58201792A (en) * 1982-04-23 1983-11-24 フアイザ−・インコ−ポレ−テツド Crystalline benzene sulfonate of saltamiciline
JPS6352260A (en) * 1986-07-28 1988-03-05 ハネイウェル・ブル・インコ−ポレ−テッド Multiplex cpu interlocking system
JPS63211289A (en) * 1982-12-06 1988-09-02 ファイザー・インコーポレーテッド Intermediate for manufacturing sultamicillin and homologue
JP2007534717A (en) * 2004-04-29 2007-11-29 ベーリンガー インゲルハイム フェトメディカ ゲゼルシャフト ミット ベシュレンクテル ハフツング Use of meloxicam formulations in veterinary medicine

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4714761A (en) * 1979-03-05 1987-12-22 Pfizer Inc. 6,6-dihalopenicillanic acid 1,1-dioxides and process
US4420426A (en) 1979-03-05 1983-12-13 Pfizer Inc. 6-Alpha-halopenicillanic acid 1,1-dioxides
US4309347A (en) 1979-05-16 1982-01-05 Pfizer Inc. Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide
US4364957A (en) * 1979-09-26 1982-12-21 Pfizer Inc. Bis-esters of alkanediols as antibacterial agents
US4432970A (en) * 1979-11-23 1984-02-21 Pfizer Inc. 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors
IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate
US4478748A (en) * 1981-02-20 1984-10-23 Pfizer Inc. Bis-esters of alkanediols
US4540687A (en) * 1981-09-09 1985-09-10 Pfizer Inc. Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds
US4582829A (en) * 1981-09-09 1986-04-15 Pfizer Inc. Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds
US4444686A (en) * 1982-01-25 1984-04-24 Pfizer Inc. Crystalline penicillin ester intermediate
KR20020028298A (en) * 2000-10-09 2002-04-17 황해용 Underpaper and manufacturing apparatus thereof

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS52118492A (en) * 1976-03-30 1977-10-04 Leo Pharm Prod As Novel amidinopenicillanoyl oxyalkylamoxylinate salts thereof process for preparing same and pharmaceutical composition containing same

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS52118492A (en) * 1976-03-30 1977-10-04 Leo Pharm Prod As Novel amidinopenicillanoyl oxyalkylamoxylinate salts thereof process for preparing same and pharmaceutical composition containing same

Cited By (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55157589A (en) * 1979-05-16 1980-12-08 Pfizer Penicillins of methanediol and bisester of methanediol and penicillanic acid 1*11dioxide
JPS6318595B2 (en) * 1979-05-16 1988-04-19 Pfizer
JPS57126493A (en) * 1980-10-31 1982-08-06 Leo Pharm Prod Ltd Cryatal hydrate of penicillanic acid derivative salt, manufacture and use
JPH027957B2 (en) * 1980-10-31 1990-02-21 Reo Pharm Purodakutsu Ltd As Reebensu Kemisuke Fuaburitsuku Purodeyukuchionsu As
JPS57169486A (en) * 1981-03-23 1982-10-19 Pfizer Manufacture of halomethyl ester ( and related ester) of penicillanic acid 1,1-dioxide
JPS57176989A (en) * 1981-03-23 1982-10-30 Pfizer Improvement on manufacture of penicillanic acid esters
JPH0446958B2 (en) * 1981-03-23 1992-07-31 Pfizer
JPH0331717B2 (en) * 1981-03-23 1991-05-08 Pfizer
JPS6345287A (en) * 1981-03-23 1988-02-26 ファイザ−・インコ−ポレ−テッド Production of 6-(2-amino-2-phenylacetamide) penicillanic acid 1, 1- dioxopenicillanoyloxymethyl
JPS57169493A (en) * 1981-03-23 1982-10-19 Pfizer 6-(2-amino-2-phenylacetamide)penicillanic acid 1,1-dioxopenicillanoyloxymethyl, manufacture and intermediate
JPS6372693A (en) * 1981-03-23 1988-04-02 ファイザ−・インコ−ポレ−テッド Improvement in production of penicilanoyloxy penicillanates
JPS5857384A (en) * 1981-09-09 1983-04-05 フアイザ−・インコ−ポレ−テツド Antibacterial penicillanic acid 6'-(2-amino- 2-(4-acyloxyphenyl)acetamide)penicillanoyloxymethyl- 1,1-dioxide compound
JPS6318949B2 (en) * 1981-09-09 1988-04-20 Pfizer
JPS5862179A (en) * 1981-09-18 1983-04-13 フアイザ−・インコ−ポレ−テツド Antibacterial ester of resolcine, ampicillin and penicillanic acid 1,1-dioxide derivative
JPS6310156B2 (en) * 1981-09-18 1988-03-04 Pfizer
JPH0119394B2 (en) * 1981-12-22 1989-04-11 Pfizer
JPS58116490A (en) * 1981-12-22 1983-07-11 フアイザ−・インコ−ポレ−テツド Antibacterial bridged with bis-hydroxymethyl carbonate
JPH0119395B2 (en) * 1982-04-23 1989-04-11 Pfizer
JPS58201792A (en) * 1982-04-23 1983-11-24 フアイザ−・インコ−ポレ−テツド Crystalline benzene sulfonate of saltamiciline
JPS63211289A (en) * 1982-12-06 1988-09-02 ファイザー・インコーポレーテッド Intermediate for manufacturing sultamicillin and homologue
JPH026758B2 (en) * 1982-12-06 1990-02-13 Pfizer
JPS6352260A (en) * 1986-07-28 1988-03-05 ハネイウェル・ブル・インコ−ポレ−テッド Multiplex cpu interlocking system
JPH084267B2 (en) * 1986-07-28 1996-01-17 ハネイウェル・ブル・インコ−ポレ−テッド Computer network system
JP2007534717A (en) * 2004-04-29 2007-11-29 ベーリンガー インゲルハイム フェトメディカ ゲゼルシャフト ミット ベシュレンクテル ハフツング Use of meloxicam formulations in veterinary medicine

Also Published As

Publication number Publication date
KR830001947A (en) 1983-05-21
BE881675A (en) 1980-08-12
ZA80796B (en) 1981-02-25
JPS6259709B2 (en) 1987-12-12
KR830001903B1 (en) 1983-09-19
JPS62281879A (en) 1987-12-07
JPH0470315B2 (en) 1992-11-10

Similar Documents

Publication Publication Date Title
GB2051779B (en) Esters of acyl-carnitines
JPS55113790A (en) Novel penicillanic ester derivative and its manufacture and use
JPS5527199A (en) Mercaptoacylproline derivative and its manufacture and use
JPS5764653A (en) Agmatilene derivative and manufacture
JPS5495592A (en) Cephalosporin derivative and manufacture
JPS55154977A (en) Penicillanic acid derivative* its manufacture and use
JPS5679636A (en) Ester manufacture
JPS55154981A (en) Novel 33vinyllcephalosporin derivative and its manufacture
JPS5522690A (en) 11phenylpiperazine derivative and its manufacture
JPS55108871A (en) Novel norrtropane derivative*its manufacture and use
JPS5622799A (en) 255halocholesterr55enee3beta*222diol and its ester
JPS54132565A (en) Substituted steroiddspiroooxazolidinone derivative and its manufacture
JPS54119457A (en) Glyoxall22oxime derivative and its manufacture
JPS55100392A (en) Novel cephalosporin derivative* its manufacture and use
JPS5531063A (en) 22hydroxymethyllpyrazine derivative and its manufacture
JPS5598186A (en) Manufacture of penicillin derivative
JPS56115743A (en) Alpha ester and its manufacture
JPS54125641A (en) Novel 33methyleneecyclopentane derivative and manufacture
JPS54145700A (en) Tetrahydroarstonine derivative and its manufacture
JPS54154784A (en) Cephem derivative and its manufacture
JPS5630949A (en) Manufacture of pentt33eneeaciddc11c44alkyl ester
JPS56115746A (en) Hydroxyaminomethyl derivatives of benzoylldiisubstituteddalphaaphenoxyalkanoyl esters
JPS55157588A (en) Penicillanic acid derivative and its manufacture
JPS54119453A (en) Novel benzothiopyrane derivative*its manufacture and its use
JPS5484594A (en) Clavulanic acid derivative and its manufacture