JPS5686187A - 7-acylamino-3-vinylcephalosporanic acid derivative and its preparation - Google Patents
7-acylamino-3-vinylcephalosporanic acid derivative and its preparationInfo
- Publication number
- JPS5686187A JPS5686187A JP16398980A JP16398980A JPS5686187A JP S5686187 A JPS5686187 A JP S5686187A JP 16398980 A JP16398980 A JP 16398980A JP 16398980 A JP16398980 A JP 16398980A JP S5686187 A JPS5686187 A JP S5686187A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- amino
- salt
- acylamino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000002253 acid Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 150000003839 salts Chemical class 0.000 abstract 3
- 125000003277 amino group Chemical group 0.000 abstract 2
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 2
- OKBVVJOGVLARMR-LNUXAPHWSA-N (6r)-7-[[2-(2-amino-1,3-thiazol-4-yl)-2-(carboxymethoxyimino)acetyl]amino]-3-ethenyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid Chemical compound S1C(N)=NC(C(=NOCC(O)=O)C(=O)NC2C(N3C(=C(C=C)CS[C@@H]32)C(O)=O)=O)=C1 OKBVVJOGVLARMR-LNUXAPHWSA-N 0.000 abstract 1
- 241000894006 Bacteria Species 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- -1 amino, protected amino Chemical group 0.000 abstract 1
- 230000000845 anti-microbial effect Effects 0.000 abstract 1
- 239000004599 antimicrobial Substances 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 244000000010 microbial pathogen Species 0.000 abstract 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1
Landscapes
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pyridine Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Indole Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB7939985 | 1979-11-19 |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP62044400A Division JPS62277391A (ja) | 1979-11-19 | 1987-02-26 | 7−アシルアミノ−3−ビニルセフアロスポラン酸誘導体およびその製法 |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5686187A true JPS5686187A (en) | 1981-07-13 |
JPS6320435B2 JPS6320435B2 (en, 2012) | 1988-04-27 |
Family
ID=10509300
Family Applications (12)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP16398980A Granted JPS5686187A (en) | 1979-11-19 | 1980-11-19 | 7-acylamino-3-vinylcephalosporanic acid derivative and its preparation |
JP16399080A Pending JPS5686188A (en) | 1979-11-19 | 1980-11-19 | 7-acylamino-3-substituted cephalosporanic acid derivative and its preparation |
JP19117582A Granted JPS5896092A (ja) | 1979-11-19 | 1982-10-29 | 7−アシルアミノ−3−置換セフアロスポラン酸誘導体およびその製造法 |
JP22640283A Granted JPS59144788A (ja) | 1979-11-19 | 1983-11-29 | 7−アシルアミノ−3−置換セフアロスポラン酸誘導体およびその製法 |
JP27813884A Pending JPS60185787A (ja) | 1979-11-19 | 1984-12-29 | 7−アシルアミノ−3−置換セフアロスポラン酸誘導体およびその製造方法 |
JP62044400A Granted JPS62277391A (ja) | 1979-11-19 | 1987-02-26 | 7−アシルアミノ−3−ビニルセフアロスポラン酸誘導体およびその製法 |
JP62290251A Granted JPS63152370A (ja) | 1979-11-19 | 1987-11-17 | 新規カルボン酸 |
JP62290253A Granted JPS63146863A (ja) | 1979-11-19 | 1987-11-17 | カルボン酸類 |
JP62290252A Granted JPS63152371A (ja) | 1979-11-19 | 1987-11-17 | アミノチアゾール誘導体 |
JP29025087A Granted JPS63152385A (ja) | 1979-11-19 | 1987-11-17 | 新規な7−置換−3−ビニルセファロスポラン酸 |
JP29024887A Granted JPS63152387A (ja) | 1979-11-19 | 1987-11-17 | 7−アシルアミノ−3−ビニル セファロスポラン酸誘導体 |
JP29024987A Granted JPS63152388A (ja) | 1979-11-19 | 1987-11-17 | 新規なセフェム化合物 |
Family Applications After (11)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP16399080A Pending JPS5686188A (en) | 1979-11-19 | 1980-11-19 | 7-acylamino-3-substituted cephalosporanic acid derivative and its preparation |
JP19117582A Granted JPS5896092A (ja) | 1979-11-19 | 1982-10-29 | 7−アシルアミノ−3−置換セフアロスポラン酸誘導体およびその製造法 |
JP22640283A Granted JPS59144788A (ja) | 1979-11-19 | 1983-11-29 | 7−アシルアミノ−3−置換セフアロスポラン酸誘導体およびその製法 |
JP27813884A Pending JPS60185787A (ja) | 1979-11-19 | 1984-12-29 | 7−アシルアミノ−3−置換セフアロスポラン酸誘導体およびその製造方法 |
JP62044400A Granted JPS62277391A (ja) | 1979-11-19 | 1987-02-26 | 7−アシルアミノ−3−ビニルセフアロスポラン酸誘導体およびその製法 |
JP62290251A Granted JPS63152370A (ja) | 1979-11-19 | 1987-11-17 | 新規カルボン酸 |
JP62290253A Granted JPS63146863A (ja) | 1979-11-19 | 1987-11-17 | カルボン酸類 |
JP62290252A Granted JPS63152371A (ja) | 1979-11-19 | 1987-11-17 | アミノチアゾール誘導体 |
JP29025087A Granted JPS63152385A (ja) | 1979-11-19 | 1987-11-17 | 新規な7−置換−3−ビニルセファロスポラン酸 |
JP29024887A Granted JPS63152387A (ja) | 1979-11-19 | 1987-11-17 | 7−アシルアミノ−3−ビニル セファロスポラン酸誘導体 |
JP29024987A Granted JPS63152388A (ja) | 1979-11-19 | 1987-11-17 | 新規なセフェム化合物 |
Country Status (2)
Country | Link |
---|---|
JP (12) | JPS5686187A (en, 2012) |
ZA (1) | ZA806977B (en, 2012) |
Cited By (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS57126492A (en) * | 1981-01-29 | 1982-08-06 | Yamanouchi Pharmaceut Co Ltd | 7-amino-3-halogenomethyl-delta3-cephem-4-carboxylic acids and their preparations |
JPS58135894A (ja) * | 1982-01-22 | 1983-08-12 | Fujisawa Pharmaceut Co Ltd | 7―置換ブチルアミド―3―ビニルセファロスポラン酸誘導体 |
JPS58164594A (ja) * | 1982-03-08 | 1983-09-29 | Fujisawa Pharmaceut Co Ltd | 7―アシルアミノ―3―セフェム―4―カルボン酸誘導体 |
JPS5921695A (ja) * | 1982-07-29 | 1984-02-03 | Dai Ichi Seiyaku Co Ltd | セフアロスポリン誘導体 |
JPS5989690A (ja) * | 1982-09-30 | 1984-05-23 | Fujisawa Pharmaceut Co Ltd | 7−アシルアミノ−3−ビニルセフアロスポラン酸誘導体、その製法およびそれを含有する抗菌剤 |
JPS59210092A (ja) * | 1983-05-13 | 1984-11-28 | Dai Ichi Seiyaku Co Ltd | セフアロスポリン誘導体 |
JPS6023317A (ja) * | 1983-07-12 | 1985-02-05 | Fujisawa Pharmaceut Co Ltd | 魚の細菌感染症予防治療剤 |
EP0238060A2 (en) | 1986-03-19 | 1987-09-23 | Banyu Pharmaceutical Co., Ltd. | Cephalosporin derivatives, processes for their preparation and antibacterial agents |
JPS62294687A (ja) * | 1982-09-30 | 1987-12-22 | Fujisawa Pharmaceut Co Ltd | 7−アシルアミノ−3−ビニル−3−セフエム化合物 |
US4822786A (en) * | 1986-07-01 | 1989-04-18 | Kaken Pharmaceutical Co., Ltd. | Cephalosporin compounds, and antibacterial agents |
JP2002510694A (ja) * | 1998-04-02 | 2002-04-09 | バイオケミ・ゲゼルシヤフト・エム・ベー・ハー | セファロスポリン誘導体の精製方法 |
JP2006501305A (ja) * | 2002-10-01 | 2006-01-12 | アンティビオーティコス エッセ.ピ.ア. | セフジニル中間体塩 |
JP2015504907A (ja) * | 2012-01-24 | 2015-02-16 | アイクリス ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト | アミジン置換β−ラクタム化合物類、それらの調製及び抗菌剤 |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA806977B (en) * | 1979-11-19 | 1981-10-28 | Fujisawa Pharmaceutical Co | 7-acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof |
FR2476087A1 (fr) * | 1980-02-18 | 1981-08-21 | Roussel Uclaf | Nouvelles oximes derivees de l'acide 3-alkyloxy ou 3-alkyl-thiomethyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments |
EP0046964B1 (en) * | 1980-08-29 | 1986-08-20 | Fujisawa Pharmaceutical Co., Ltd. | New cephem compounds and processes for preparation thereof |
JPS58159496A (ja) * | 1983-03-02 | 1983-09-21 | Kyoto Yakuhin Kogyo Kk | セフエム系化合物 |
GB8329030D0 (en) * | 1983-10-31 | 1983-11-30 | Fujisawa Pharmaceutical Co | Cephem compounds |
JP4157177B2 (ja) * | 1997-06-04 | 2008-09-24 | 大塚化学ホールディングス株式会社 | 3−アルケニルセフェム化合物の製造法 |
US7980324B2 (en) | 2006-02-03 | 2011-07-19 | Black & Decker Inc. | Housing and gearbox for drill or driver |
JP4779741B2 (ja) * | 2006-03-22 | 2011-09-28 | 株式会社日立製作所 | ヒートポンプシステム,ヒートポンプシステムの軸封方法,ヒートポンプシステムの改造方法 |
KR101485316B1 (ko) * | 2014-04-16 | 2015-01-22 | (주)에이치티씨 | 플렛 케이블용 컨넥터 핀 자동 압착장치 |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE789817A (fr) * | 1971-10-07 | 1973-04-06 | Glaxo Lab Ltd | Perfectionnements aux composes de cephalosporine |
GB1325846A (en) * | 1972-02-23 | 1973-08-08 | Lilly Co Eli | Process for the preparation of a 3-thiomethyl cephalosporin |
DE2209019A1 (de) * | 1972-02-25 | 1973-08-30 | Lilly Co Eli | Verfahren zur herstellung von 3-thiomethylcephalosporinverbindungen |
JPS5729474B2 (en, 2012) * | 1974-01-14 | 1982-06-23 | ||
DE2710902A1 (de) * | 1977-03-12 | 1978-09-21 | Hoechst Ag | Cephemderivate und verfahren zu ihrer herstellung |
DE2714880A1 (de) * | 1977-04-02 | 1978-10-26 | Hoechst Ag | Cephemderivate und verfahren zu ihrer herstellung |
US4200745A (en) * | 1977-12-20 | 1980-04-29 | Eli Lilly And Company | 7[2-(2-Aminothiazol-4-yl)-2-alkoxyimino]acetamido 3[4-alkyl-5-oxo-6-hydroxy-3,4 dihydro 1,2,4-triazin 3-yl]thio methyl cephalosporins |
FR2432521A1 (fr) * | 1978-03-31 | 1980-02-29 | Roussel Uclaf | Nouvelles oximes o-substituees derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments |
CY1168A (en) * | 1978-05-26 | 1983-06-10 | Glaxo Group Ltd | Cephalosporin antibiotics |
GB1604723A (en) * | 1978-05-26 | 1981-12-16 | Glaxo Operations Ltd | 7-(2-aminothiazol-4-yl)-2-oxyimino-acetamido)-cephem derivatives |
AU529823B2 (en) * | 1978-10-26 | 1983-06-23 | Glaxo Group Limited | Cephalosporin compounds |
BE879666A (fr) * | 1978-10-27 | 1980-04-28 | Glaxo Group Ltd | Nouvelles cephalosporines, leur preparation et compositions les contenant |
IT1207006B (it) * | 1978-11-15 | 1989-05-17 | Glaxo Group Ltd | Antibiotici cefalosporinici composizioni che li contengono e procedimento per produrli |
NZ192142A (en) * | 1978-11-17 | 1982-12-21 | Glaxo Group Ltd | Cephalosporin derivatives and pharmaceutical compositions |
BE881870A (fr) * | 1979-02-23 | 1980-08-22 | Glaxo Group Ltd | Nouvelles cephalosporines qui exercent une activite contre des organismes gram-negatifs |
JPS55124790A (en) * | 1979-03-19 | 1980-09-26 | Sankyo Co Ltd | Cephem compound, its preparation and antimicrobials consisting the same mainly |
NL160860B (nl) * | 1979-03-22 | American Cyanamid Co | Werkwijze voor het bereiden van een vulcaniseerbaar mengsel. | |
ZA806977B (en) * | 1979-11-19 | 1981-10-28 | Fujisawa Pharmaceutical Co | 7-acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof |
-
1980
- 1980-11-11 ZA ZA00806977A patent/ZA806977B/xx unknown
- 1980-11-19 JP JP16398980A patent/JPS5686187A/ja active Granted
- 1980-11-19 JP JP16399080A patent/JPS5686188A/ja active Pending
-
1982
- 1982-10-29 JP JP19117582A patent/JPS5896092A/ja active Granted
-
1983
- 1983-11-29 JP JP22640283A patent/JPS59144788A/ja active Granted
-
1984
- 1984-12-29 JP JP27813884A patent/JPS60185787A/ja active Pending
-
1987
- 1987-02-26 JP JP62044400A patent/JPS62277391A/ja active Granted
- 1987-11-17 JP JP62290251A patent/JPS63152370A/ja active Granted
- 1987-11-17 JP JP62290253A patent/JPS63146863A/ja active Granted
- 1987-11-17 JP JP62290252A patent/JPS63152371A/ja active Granted
- 1987-11-17 JP JP29025087A patent/JPS63152385A/ja active Granted
- 1987-11-17 JP JP29024887A patent/JPS63152387A/ja active Granted
- 1987-11-17 JP JP29024987A patent/JPS63152388A/ja active Granted
Cited By (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS57126492A (en) * | 1981-01-29 | 1982-08-06 | Yamanouchi Pharmaceut Co Ltd | 7-amino-3-halogenomethyl-delta3-cephem-4-carboxylic acids and their preparations |
JPS58135894A (ja) * | 1982-01-22 | 1983-08-12 | Fujisawa Pharmaceut Co Ltd | 7―置換ブチルアミド―3―ビニルセファロスポラン酸誘導体 |
JPS58164594A (ja) * | 1982-03-08 | 1983-09-29 | Fujisawa Pharmaceut Co Ltd | 7―アシルアミノ―3―セフェム―4―カルボン酸誘導体 |
JPS5921695A (ja) * | 1982-07-29 | 1984-02-03 | Dai Ichi Seiyaku Co Ltd | セフアロスポリン誘導体 |
JPS62294687A (ja) * | 1982-09-30 | 1987-12-22 | Fujisawa Pharmaceut Co Ltd | 7−アシルアミノ−3−ビニル−3−セフエム化合物 |
JPS5989690A (ja) * | 1982-09-30 | 1984-05-23 | Fujisawa Pharmaceut Co Ltd | 7−アシルアミノ−3−ビニルセフアロスポラン酸誘導体、その製法およびそれを含有する抗菌剤 |
JPS59210092A (ja) * | 1983-05-13 | 1984-11-28 | Dai Ichi Seiyaku Co Ltd | セフアロスポリン誘導体 |
JPS6023317A (ja) * | 1983-07-12 | 1985-02-05 | Fujisawa Pharmaceut Co Ltd | 魚の細菌感染症予防治療剤 |
EP0238060A2 (en) | 1986-03-19 | 1987-09-23 | Banyu Pharmaceutical Co., Ltd. | Cephalosporin derivatives, processes for their preparation and antibacterial agents |
US4822786A (en) * | 1986-07-01 | 1989-04-18 | Kaken Pharmaceutical Co., Ltd. | Cephalosporin compounds, and antibacterial agents |
JP2002510694A (ja) * | 1998-04-02 | 2002-04-09 | バイオケミ・ゲゼルシヤフト・エム・ベー・ハー | セファロスポリン誘導体の精製方法 |
JP2006501305A (ja) * | 2002-10-01 | 2006-01-12 | アンティビオーティコス エッセ.ピ.ア. | セフジニル中間体塩 |
JP2015504907A (ja) * | 2012-01-24 | 2015-02-16 | アイクリス ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト | アミジン置換β−ラクタム化合物類、それらの調製及び抗菌剤 |
Also Published As
Publication number | Publication date |
---|---|
JPS63152388A (ja) | 1988-06-24 |
JPS63152385A (ja) | 1988-06-24 |
JPS63152370A (ja) | 1988-06-24 |
JPH0338278B2 (en, 2012) | 1991-06-10 |
JPH0219828B2 (en, 2012) | 1990-05-07 |
JPS63146863A (ja) | 1988-06-18 |
JPS60185787A (ja) | 1985-09-21 |
ZA806977B (en) | 1981-10-28 |
JPH0225905B2 (en, 2012) | 1990-06-06 |
JPS6320435B2 (en, 2012) | 1988-04-27 |
JPS59144788A (ja) | 1984-08-18 |
JPS62277391A (ja) | 1987-12-02 |
JPH0369353B2 (en, 2012) | 1991-10-31 |
JPH0338277B2 (en, 2012) | 1991-06-10 |
JPS6238357B2 (en, 2012) | 1987-08-17 |
JPH0314832B2 (en, 2012) | 1991-02-27 |
JPS63152387A (ja) | 1988-06-24 |
JPS5686188A (en) | 1981-07-13 |
JPH0215556B2 (en, 2012) | 1990-04-12 |
JPS63152371A (ja) | 1988-06-24 |
JPH0333712B2 (en, 2012) | 1991-05-20 |
JPS5896092A (ja) | 1983-06-07 |
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