JP4099224B2 - 舌下又はバッカル医薬組成物 - Google Patents

舌下又はバッカル医薬組成物 Download PDF

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Publication number
JP4099224B2
JP4099224B2 JP52270395A JP52270395A JP4099224B2 JP 4099224 B2 JP4099224 B2 JP 4099224B2 JP 52270395 A JP52270395 A JP 52270395A JP 52270395 A JP52270395 A JP 52270395A JP 4099224 B2 JP4099224 B2 JP 4099224B2
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JP
Japan
Prior art keywords
pharmaceutical composition
sublingual
oxepino
dibenz
tetrahydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP52270395A
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English (en)
Japanese (ja)
Other versions
JPH09509674A (ja
Inventor
デルブレシーネ，レオナルドウス・ペトルス・カルラ
ウイリンガ，ヨハンネス・フベルトウス
Original Assignee
ナームローゼ・フエンノートチヤツプ・オルガノン
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8216678&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JP4099224(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by ナームローゼ・フエンノートチヤツプ・オルガノン filed Critical ナームローゼ・フエンノートチヤツプ・オルガノン
Publication of JPH09509674A publication Critical patent/JPH09509674A/ja
Application granted granted Critical
Publication of JP4099224B2 publication Critical patent/JP4099224B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP52270395A 1994-03-02 1995-03-01 舌下又はバッカル医薬組成物 Expired - Lifetime JP4099224B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
AT94200521.6 1994-03-02
EP94200521 1994-03-02
PCT/EP1995/000765 WO1995023600A1 (en) 1994-03-02 1995-03-01 Sublingual or buccal pharmaceutical composition

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2006217762A Division JP4616810B2 (ja) 1994-03-02 2006-08-10 舌下又はバッカル医薬組成物

Publications (2)

Publication Number Publication Date
JPH09509674A JPH09509674A (ja) 1997-09-30
JP4099224B2 true JP4099224B2 (ja) 2008-06-11

Family

ID=8216678

Family Applications (2)

Application Number Title Priority Date Filing Date
JP52270395A Expired - Lifetime JP4099224B2 (ja) 1994-03-02 1995-03-01 舌下又はバッカル医薬組成物
JP2006217762A Expired - Lifetime JP4616810B2 (ja) 1994-03-02 2006-08-10 舌下又はバッカル医薬組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2006217762A Expired - Lifetime JP4616810B2 (ja) 1994-03-02 2006-08-10 舌下又はバッカル医薬組成物

Country Status (23)

Country Link
US (1) US5763476A (OSRAM)
EP (1) EP0746317B1 (OSRAM)
JP (2) JP4099224B2 (OSRAM)
KR (1) KR100330942B1 (OSRAM)
CN (1) CN1079670C (OSRAM)
AT (1) ATE167057T1 (OSRAM)
AU (1) AU692530B2 (OSRAM)
BR (2) BR9506924A (OSRAM)
CA (1) CA2182981C (OSRAM)
CZ (1) CZ284633B6 (OSRAM)
DE (2) DE69502939T2 (OSRAM)
DK (1) DK0746317T3 (OSRAM)
ES (1) ES2118584T3 (OSRAM)
FI (1) FI117923B (OSRAM)
FR (1) FR10C0056I2 (OSRAM)
HK (1) HK1008417A1 (OSRAM)
HU (1) HU225051B1 (OSRAM)
LU (1) LU91751I2 (OSRAM)
NO (2) NO308772B1 (OSRAM)
NZ (1) NZ282394A (OSRAM)
PL (1) PL180465B1 (OSRAM)
RU (1) RU2139051C1 (OSRAM)
WO (1) WO1995023600A1 (OSRAM)

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MXPA06002766A (es) * 2003-09-22 2006-12-14 Baxter Int Esterilizacion a alta presion para esterilizar terminalmente preparaciones farmaceuticas y productos medicos.
MXPA06013163A (es) * 2004-05-11 2007-02-13 Pfizer Prod Inc Combinacion de antipsicoticos atipicos y antagonistas del receptor 5-ht1b.
GB0416861D0 (en) * 2004-07-29 2004-09-01 Quadrant Drug Delivery Ltd Composition
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ES2293626T3 (es) * 2005-04-07 2008-03-16 N.V. Organon Forma cristalina del maleato de asenapina.
US7872147B2 (en) 2005-04-07 2011-01-18 N. V. Organon Intermediate compounds for the preparation of trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole
AR063188A1 (es) 2005-04-07 2009-01-14 Organon Nv Compuestos intermediarios para la preparacion de trans -5-cloro-2-netil-2,3,3a,12b- tetrahidro-1h-dibenz (2,3:6,7)- oxepina (4,5c) pirrol
US7741358B2 (en) * 2005-04-14 2010-06-22 N.V. Organon Crystal form of asenapine maleate
US7750167B2 (en) 2006-07-05 2010-07-06 N.V. Organon Process for the preparation of asenapine and intermediate products used in said process
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Also Published As

Publication number Publication date
CA2182981C (en) 2006-10-17
EP0746317A1 (en) 1996-12-11
CZ254196A3 (en) 1997-10-15
WO1995023600A1 (en) 1995-09-08
NO963639D0 (no) 1996-08-30
FR10C0056I2 (OSRAM) 2011-11-25
DK0746317T3 (da) 1999-03-22
DE122010000050I2 (de) 2011-07-21
RU2139051C1 (ru) 1999-10-10
CA2182981A1 (en) 1995-09-08
NO963639L (no) 1996-10-30
CZ284633B6 (cs) 1999-01-13
FI963398L (fi) 1996-08-30
FR10C0056I1 (OSRAM) 2011-01-28
KR100330942B1 (ko) 2002-11-16
ES2118584T3 (es) 1998-09-16
AU1947895A (en) 1995-09-18
MX9603713A (es) 1997-12-31
NO2010024I2 (no) 2012-04-10
EP0746317B1 (en) 1998-06-10
FI963398A0 (fi) 1996-08-30
CN1079670C (zh) 2002-02-27
HU225051B1 (en) 2006-05-29
NO308772B1 (no) 2000-10-30
PL316080A1 (en) 1996-12-23
NZ282394A (en) 1997-12-19
CN1143320A (zh) 1997-02-19
BR1100625A (pt) 1999-12-28
ATE167057T1 (de) 1998-06-15
AU692530B2 (en) 1998-06-11
JP4616810B2 (ja) 2011-01-19
LU91751I2 (fr) 2011-01-04
DE69502939D1 (de) 1998-07-16
DE69502939T2 (de) 1998-10-22
NO2010024I1 (no) 2011-01-03
HK1008417A1 (en) 1999-05-07
PL180465B1 (pl) 2001-02-28
JPH09509674A (ja) 1997-09-30
HU9602383D0 (en) 1996-10-28
HUT76319A (en) 1997-08-28
JP2006342178A (ja) 2006-12-21
BR9506924A (pt) 1997-09-30
US5763476A (en) 1998-06-09
DE122010000050I1 (de) 2011-05-05
FI117923B (fi) 2007-04-30

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