LU91751I2 - Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®) - Google Patents

Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®)

Info

Publication number
LU91751I2
LU91751I2 LU91751C LU91751C LU91751I2 LU 91751 I2 LU91751 I2 LU 91751I2 LU 91751 C LU91751 C LU 91751C LU 91751 C LU91751 C LU 91751C LU 91751 I2 LU91751 I2 LU 91751I2
Authority
LU
Luxembourg
Prior art keywords
pharmaceutically acceptable
pct
sublingual
asenapin
sycrest
Prior art date
Application number
LU91751C
Other languages
English (en)
French (fr)
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8216678&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU91751(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Organon Nv filed Critical Organon Nv
Publication of LU91751I2 publication Critical patent/LU91751I2/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
LU91751C 1994-03-02 2010-11-04 Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®) LU91751I2 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP94200521 1994-03-02
PCT/EP1995/000765 WO1995023600A1 (en) 1994-03-02 1995-03-01 Sublingual or buccal pharmaceutical composition
EP95912188A EP0746317B1 (en) 1994-03-02 1995-03-01 Sublingual or buccal pharmaceutical composition

Publications (1)

Publication Number Publication Date
LU91751I2 true LU91751I2 (fr) 2011-01-04

Family

ID=8216678

Family Applications (1)

Application Number Title Priority Date Filing Date
LU91751C LU91751I2 (fr) 1994-03-02 2010-11-04 Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®)

Country Status (22)

Country Link
US (1) US5763476A (OSRAM)
EP (1) EP0746317B1 (OSRAM)
JP (2) JP4099224B2 (OSRAM)
KR (1) KR100330942B1 (OSRAM)
CN (1) CN1079670C (OSRAM)
AT (1) ATE167057T1 (OSRAM)
AU (1) AU692530B2 (OSRAM)
BR (2) BR9506924A (OSRAM)
CA (1) CA2182981C (OSRAM)
CZ (1) CZ284633B6 (OSRAM)
DE (2) DE69502939T2 (OSRAM)
DK (1) DK0746317T3 (OSRAM)
ES (1) ES2118584T3 (OSRAM)
FI (1) FI117923B (OSRAM)
FR (1) FR10C0056I2 (OSRAM)
HU (1) HU225051B1 (OSRAM)
LU (1) LU91751I2 (OSRAM)
NO (2) NO308772B1 (OSRAM)
NZ (1) NZ282394A (OSRAM)
PL (1) PL180465B1 (OSRAM)
RU (1) RU2139051C1 (OSRAM)
WO (1) WO1995023600A1 (OSRAM)

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PT1917267E (pt) * 2005-04-07 2009-02-04 Organon Nv Forma cristalina de maleato de asenapina
PL1710241T3 (pl) 2005-04-07 2010-04-30 Msd Oss Bv Związki pośrednie do wytwarzania trans-5-chloro-2-metylo-2,3,3a,12b-tetrahydro-1H-dibenz-[2,3:6,7]oksepino[4,5-c]pirolu
US7741358B2 (en) * 2005-04-14 2010-06-22 N.V. Organon Crystal form of asenapine maleate
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US7875729B2 (en) 2007-01-05 2011-01-25 Synthon Bv Process for making asenapine
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AR077225A1 (es) 2009-06-24 2011-08-10 Organon Nv Formulaciones inyectables que contienen asenapina y metodo de tratamiento que las utiliza
AR077429A1 (es) 2009-07-29 2011-08-24 Organon Nv Compuestos hidroxiasenapina sus derivados y composiciones farmaceuticas que comprenden los mismos
US8779161B2 (en) 2010-06-18 2014-07-15 Dr. Reddy's Laboratories Limited Asenapine maleate
JP5815702B2 (ja) 2010-07-29 2015-11-17 ラボラトリオス レスヴィ，エス．エル． アセナピンの新規な製造方法
WO2012038975A2 (en) * 2010-09-22 2012-03-29 Msn Laboratories Limited Process for the preparation of (3ars,12brs)-5-chloro-2-methyl-2,3,3a12b-tetrahydro-1hdibenzo[2,3:6,7] oxepino [4,5-c]pyrrole maleate and it's pharmaceutical composition thereof
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US20140206667A1 (en) 2012-11-14 2014-07-24 Michela Gallagher Methods and compositions for treating schizophrenia
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Also Published As

Publication number Publication date
CA2182981C (en) 2006-10-17
HUT76319A (en) 1997-08-28
FI963398L (fi) 1996-08-30
JPH09509674A (ja) 1997-09-30
PL180465B1 (pl) 2001-02-28
BR9506924A (pt) 1997-09-30
NO963639L (no) 1996-10-30
CZ284633B6 (cs) 1999-01-13
HK1008417A1 (en) 1999-05-07
AU692530B2 (en) 1998-06-11
FI963398A0 (fi) 1996-08-30
JP4616810B2 (ja) 2011-01-19
HU9602383D0 (en) 1996-10-28
DE69502939T2 (de) 1998-10-22
ES2118584T3 (es) 1998-09-16
KR100330942B1 (ko) 2002-11-16
BR1100625A (pt) 1999-12-28
FI117923B (fi) 2007-04-30
MX9603713A (es) 1997-12-31
FR10C0056I1 (OSRAM) 2011-01-28
JP4099224B2 (ja) 2008-06-11
NO963639D0 (no) 1996-08-30
EP0746317B1 (en) 1998-06-10
CN1079670C (zh) 2002-02-27
DE122010000050I2 (de) 2011-07-21
CA2182981A1 (en) 1995-09-08
CZ254196A3 (en) 1997-10-15
DE69502939D1 (de) 1998-07-16
DK0746317T3 (da) 1999-03-22
ATE167057T1 (de) 1998-06-15
EP0746317A1 (en) 1996-12-11
NZ282394A (en) 1997-12-19
FR10C0056I2 (OSRAM) 2011-11-25
NO308772B1 (no) 2000-10-30
WO1995023600A1 (en) 1995-09-08
HU225051B1 (en) 2006-05-29
PL316080A1 (en) 1996-12-23
NO2010024I1 (no) 2011-01-03
RU2139051C1 (ru) 1999-10-10
US5763476A (en) 1998-06-09
CN1143320A (zh) 1997-02-19
AU1947895A (en) 1995-09-18
NO2010024I2 (no) 2012-04-10
DE122010000050I1 (de) 2011-05-05
JP2006342178A (ja) 2006-12-21

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