JP2019512469A5 - - Google Patents

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JP2019512469A5
JP2019512469A5 JP2018545336A JP2018545336A JP2019512469A5 JP 2019512469 A5 JP2019512469 A5 JP 2019512469A5 JP 2018545336 A JP2018545336 A JP 2018545336A JP 2018545336 A JP2018545336 A JP 2018545336A JP 2019512469 A5 JP2019512469 A5 JP 2019512469A5
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pharmaceutical composition
treating
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JP2018545336A
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JP2019512469A (ja
JP6814814B2 (ja
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Priority claimed from PCT/EP2017/055885 external-priority patent/WO2017157873A1/en
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JP2018545336A 2016-03-17 2017-03-14 Taarのアゴニストとしての活性を有する5−エチル−4−メチル−ピラゾール−3−カルボキサミド誘導体 Active JP6814814B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP16160790 2016-03-17
EP16160790.8 2016-03-17
PCT/EP2017/055885 WO2017157873A1 (en) 2016-03-17 2017-03-14 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of taar

Publications (3)

Publication Number Publication Date
JP2019512469A JP2019512469A (ja) 2019-05-16
JP2019512469A5 true JP2019512469A5 (enExample) 2020-12-24
JP6814814B2 JP6814814B2 (ja) 2021-01-20

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JP2018545336A Active JP6814814B2 (ja) 2016-03-17 2017-03-14 Taarのアゴニストとしての活性を有する5−エチル−4−メチル−ピラゾール−3−カルボキサミド誘導体

Country Status (33)

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US (2) US10508107B2 (enExample)
EP (2) EP3757102A1 (enExample)
JP (1) JP6814814B2 (enExample)
KR (2) KR102537050B1 (enExample)
CN (1) CN108713019B (enExample)
AR (1) AR107878A1 (enExample)
AU (1) AU2017234042B2 (enExample)
BR (1) BR112018015389B1 (enExample)
CA (1) CA3013696C (enExample)
CL (1) CL2018002583A1 (enExample)
CO (1) CO2018007515A2 (enExample)
CR (1) CR20180443A (enExample)
DK (1) DK3430010T3 (enExample)
ES (1) ES2819830T3 (enExample)
HR (1) HRP20201405T1 (enExample)
HU (1) HUE050986T2 (enExample)
IL (1) IL260473B (enExample)
LT (1) LT3430010T (enExample)
MA (2) MA53755A (enExample)
MX (1) MX377836B (enExample)
MY (1) MY195528A (enExample)
PE (1) PE20181446A1 (enExample)
PH (1) PH12018501588A1 (enExample)
PL (1) PL3430010T3 (enExample)
PT (1) PT3430010T (enExample)
RS (1) RS60825B1 (enExample)
RU (1) RU2731095C2 (enExample)
SG (2) SG11201807516UA (enExample)
SI (1) SI3430010T1 (enExample)
TW (1) TWI634117B (enExample)
UA (1) UA122881C2 (enExample)
WO (1) WO2017157873A1 (enExample)
ZA (1) ZA201804943B (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114144412A (zh) * 2019-07-11 2022-03-04 豪夫迈·罗氏有限公司 用于制备经取代的吡唑衍生物的方法
IL294301A (en) * 2020-03-19 2022-08-01 Hoffmann La Roche Salts and crystalline forms of the taar1 agonist
JP2024538464A (ja) 2021-11-08 2024-10-22 エフ. ホフマン-ラ ロシュ アーゲー 芳香族ニトロ化合物の接触水素化
CN114288304A (zh) * 2021-12-31 2022-04-08 江苏海洋大学 一种抗精神分裂症组合物及其应用
AR129909A1 (es) 2022-07-15 2024-10-09 Hoffmann La Roche Cetorreductasa mutante con mayor actividad de cetorreductasa así como métodos y usos de esta
CN119654138A (zh) 2022-08-12 2025-03-18 豪夫迈·罗氏有限公司 包含5-乙基-4-甲基-n-[4-[(2s)吗啉-2-基]苯基]-1h-吡唑-3-甲酰胺的药物组合物
WO2024033460A1 (en) * 2022-08-12 2024-02-15 F. Hoffmann-La Roche Ag Use of co-processed excipients in continuous manufacturing of solid dosage forms
TW202440563A (zh) * 2022-11-28 2024-10-16 美商住友製藥美國公司 2-苯基嗎啉與2-苯基(硫代)嗎啉化合物及其用途
TW202444712A (zh) * 2023-04-28 2024-11-16 大陸商江蘇豪森藥業集團有限公司 一種嗎啉雜環類化合物的鹽及其製備方法和應用
CN121568694A (zh) * 2023-06-13 2026-02-24 乔治亚大学研究基金会 恶性疟原虫红内期抑制剂

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