JP2019512469A5 - - Google Patents

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JP2019512469A5
JP2019512469A5 JP2018545336A JP2018545336A JP2019512469A5 JP 2019512469 A5 JP2019512469 A5 JP 2019512469A5 JP 2018545336 A JP2018545336 A JP 2018545336A JP 2018545336 A JP2018545336 A JP 2018545336A JP 2019512469 A5 JP2019512469 A5 JP 2019512469A5
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pharmaceutical composition
treating
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composition according
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JP2018545336A
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JP6814814B2 (ja
JP2019512469A (ja
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Priority claimed from PCT/EP2017/055885 external-priority patent/WO2017157873A1/en
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JP2018545336A 2016-03-17 2017-03-14 Taarのアゴニストとしての活性を有する5−エチル−4−メチル−ピラゾール−3−カルボキサミド誘導体 Active JP6814814B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP16160790.8 2016-03-17
EP16160790 2016-03-17
PCT/EP2017/055885 WO2017157873A1 (en) 2016-03-17 2017-03-14 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of taar

Publications (3)

Publication Number Publication Date
JP2019512469A JP2019512469A (ja) 2019-05-16
JP2019512469A5 true JP2019512469A5 (enExample) 2020-12-24
JP6814814B2 JP6814814B2 (ja) 2021-01-20

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JP2018545336A Active JP6814814B2 (ja) 2016-03-17 2017-03-14 Taarのアゴニストとしての活性を有する5−エチル−4−メチル−ピラゾール−3−カルボキサミド誘導体

Country Status (33)

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US (2) US10508107B2 (enExample)
EP (2) EP3430010B1 (enExample)
JP (1) JP6814814B2 (enExample)
KR (2) KR102537050B1 (enExample)
CN (1) CN108713019B (enExample)
AR (1) AR107878A1 (enExample)
AU (1) AU2017234042B2 (enExample)
BR (1) BR112018015389B1 (enExample)
CA (1) CA3013696C (enExample)
CL (1) CL2018002583A1 (enExample)
CO (1) CO2018007515A2 (enExample)
CR (1) CR20180443A (enExample)
DK (1) DK3430010T3 (enExample)
ES (1) ES2819830T3 (enExample)
HR (1) HRP20201405T1 (enExample)
HU (1) HUE050986T2 (enExample)
IL (1) IL260473B (enExample)
LT (1) LT3430010T (enExample)
MA (2) MA53755A (enExample)
MX (1) MX377836B (enExample)
MY (1) MY195528A (enExample)
PE (1) PE20181446A1 (enExample)
PH (1) PH12018501588A1 (enExample)
PL (1) PL3430010T3 (enExample)
PT (1) PT3430010T (enExample)
RS (1) RS60825B1 (enExample)
RU (1) RU2731095C2 (enExample)
SG (2) SG10201913878YA (enExample)
SI (1) SI3430010T1 (enExample)
TW (1) TWI634117B (enExample)
UA (1) UA122881C2 (enExample)
WO (1) WO2017157873A1 (enExample)
ZA (1) ZA201804943B (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20220035106A (ko) * 2019-07-11 2022-03-21 에프. 호프만-라 로슈 아게 치환된 피라졸 유도체의 제조 방법
WO2021185878A1 (en) * 2020-03-19 2021-09-23 F. Hoffmann-La Roche Ag Salts and crystalline forms of a taar1 agonist
CN118251382A (zh) 2021-11-08 2024-06-25 豪夫迈·罗氏有限公司 芳硝基化合物的催化氢化
CN114288304A (zh) * 2021-12-31 2022-04-08 江苏海洋大学 一种抗精神分裂症组合物及其应用
AR129909A1 (es) 2022-07-15 2024-10-09 Hoffmann La Roche Cetorreductasa mutante con mayor actividad de cetorreductasa así como métodos y usos de esta
AU2023323858A1 (en) 2022-08-12 2024-11-21 F. Hoffmann-La Roche Ag Pharmaceutical compositions comprising 5-ethyl-4-methyl- n-[4-[(2 s) morpholin-2-yl]phenyl]-1h-pyrazole-3-carboxamide
WO2024033460A1 (en) * 2022-08-12 2024-02-15 F. Hoffmann-La Roche Ag Use of co-processed excipients in continuous manufacturing of solid dosage forms
WO2024118488A1 (en) * 2022-11-28 2024-06-06 Sumitomo Pharma America, Inc. 2-phenylmorpholine and 2-phenyl(thio)morpholine compounds and uses thereof
CN121311474A (zh) * 2023-04-28 2026-01-09 江苏豪森药业集团有限公司 一种吗啉杂环类化合物的盐及其制备方法和应用
AU2024305453A1 (en) * 2023-06-13 2026-01-08 Northeastern University Plasmodium falciparum blood stage inhibitors

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