JP2011516417A5 - - Google Patents

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Publication number
JP2011516417A5
JP2011516417A5 JP2011501153A JP2011501153A JP2011516417A5 JP 2011516417 A5 JP2011516417 A5 JP 2011516417A5 JP 2011501153 A JP2011501153 A JP 2011501153A JP 2011501153 A JP2011501153 A JP 2011501153A JP 2011516417 A5 JP2011516417 A5 JP 2011516417A5
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JP
Japan
Prior art keywords
pain
disease
pharmaceutical composition
composition according
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011501153A
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English (en)
Japanese (ja)
Other versions
JP2011516417A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2009/002241 external-priority patent/WO2009118187A1/en
Publication of JP2011516417A publication Critical patent/JP2011516417A/ja
Publication of JP2011516417A5 publication Critical patent/JP2011516417A5/ja
Pending legal-status Critical Current

Links

JP2011501153A 2008-03-27 2009-03-26 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法 Pending JP2011516417A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4008708P 2008-03-27 2008-03-27
US61/040,087 2008-03-27
PCT/EP2009/002241 WO2009118187A1 (en) 2008-03-27 2009-03-26 Methods for treating disorders using nmda nr2b-subtype selective antagonist

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014020051A Division JP2014098018A (ja) 2008-03-27 2014-02-05 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法

Publications (2)

Publication Number Publication Date
JP2011516417A JP2011516417A (ja) 2011-05-26
JP2011516417A5 true JP2011516417A5 (enExample) 2012-01-05

Family

ID=40910288

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011501153A Pending JP2011516417A (ja) 2008-03-27 2009-03-26 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法
JP2014020051A Pending JP2014098018A (ja) 2008-03-27 2014-02-05 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法
JP2015236571A Pending JP2016094430A (ja) 2008-03-27 2015-12-03 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2014020051A Pending JP2014098018A (ja) 2008-03-27 2014-02-05 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法
JP2015236571A Pending JP2016094430A (ja) 2008-03-27 2015-12-03 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法

Country Status (14)

Country Link
US (1) US20110053951A1 (enExample)
EP (1) EP2254580A1 (enExample)
JP (3) JP2011516417A (enExample)
KR (1) KR20100135847A (enExample)
CN (1) CN101977606A (enExample)
AU (1) AU2009228660B2 (enExample)
BR (1) BRPI0909378A2 (enExample)
CA (1) CA2719749A1 (enExample)
IL (1) IL207835A0 (enExample)
MX (1) MX2010009649A (enExample)
NZ (1) NZ588698A (enExample)
RU (1) RU2499598C2 (enExample)
WO (1) WO2009118187A1 (enExample)
ZA (1) ZA201006587B (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2013251079B2 (en) 2012-04-20 2017-03-23 Ucb Pharma S.A. Methods for treating Parkinson's disease
US11232319B2 (en) 2014-05-16 2022-01-25 The Trustees Of The University Of Pennsylvania Applications of automatic anatomy recognition in medical tomographic imagery based on fuzzy anatomy models
HUE049278T2 (hu) * 2014-08-15 2020-09-28 Janssen Pharmaceuticals Inc Pirazolok
PT3180329T (pt) 2014-08-15 2020-06-08 Janssen Pharmaceuticals Inc Triazóis como inibidores do recetor nr2b
MX380424B (es) 2015-06-01 2025-03-12 Rugen Holdings Cayman Ltd Compuestos heterociclicos de 3,3-difluorpiperidina carbamato como antagonistas del receptor de n-metil-d-aspartato (nmda) nr2b.
LT3319963T (lt) 2015-07-09 2020-03-25 Janssen Pharmaceutica Nv Pakeistieji 4-azaindolai ir jų, kaip glun2b receptoriaus moduliatorių, panaudojimas
CA3014314A1 (en) 2016-02-10 2017-08-17 Janssen Pharmaceutica Nv Substituted 1,2,3-triazoles as nr2b-selective nmda modulators
US10487055B2 (en) 2016-06-01 2019-11-26 Rhode Island Board Of Education Diindole compounds useful in treatment of nervous system disorders
TW201819376A (zh) 2016-10-06 2018-06-01 比利時商健生藥品公司 經取代之1H-咪唑並[4,5-b]吡啶-2(3H)-酮及其作為GLUN2B受體調節劑之用途
WO2018098128A1 (en) 2016-11-22 2018-05-31 Rugen Holdings (Cayman) Limited Treatment of autism spectrum disorders, obsessive-compulsive disorder and anxiety disorders
US11447503B2 (en) 2019-06-14 2022-09-20 Janssen Pharmaceutica Nv Pyridine carbamates and their use as GLUN2B receptor modulators
US10732235B2 (en) * 2018-03-29 2020-08-04 Siemens Healthcare Gmbh Magnetic resonance method and apparatus using atlas-based masking for quantitative susceptibility mapping
WO2019193516A2 (en) 2018-04-04 2019-10-10 Janssen Pharmaceutica Nv Substituted pyridine and pyrimidines and their use as glun2b receptor modulators
CN113993583A (zh) 2019-06-14 2022-01-28 詹森药业有限公司 取代的吡唑并[4,3-b]吡啶及其作为GLUN2B受体调节剂的用途
PH12021552839A1 (en) 2019-06-14 2022-10-03 Janssen Pharmaceutica Nv Substituted pyrazolo-pyridine amides and their use as glun2b receptor modulators
US11459336B2 (en) 2019-06-14 2022-10-04 Janssen Pharmaceutica Nv Pyrazine carbamates and their use as GluN2B receptor modulators
KR20220024403A (ko) 2019-06-14 2022-03-03 얀센 파마슈티카 엔.브이. 치환된 피라졸로-피라진 및 이들의 glun2b 수용체 조절제로서의 용도
BR112021025141A2 (pt) 2019-06-14 2022-01-25 Janssen Pharmaceutica Nv Pirazolo-piridinas heteroaromáticas substituídas e seu uso como moduladores do receptor glun2b
EP3983075A1 (en) 2019-06-14 2022-04-20 Janssen Pharmaceutica NV Substituted pyrazolo-pyridine amides and their use as glun2b receptor modulators

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2174220T3 (es) * 1996-03-08 2002-11-01 Hoffmann La Roche Uso de derivados de 4-fenil-3,6-dihidro-2h-piridilo como agentes bloqueantes de subtipos de receptores nmda.
US5985936A (en) * 1997-12-18 1999-11-16 Forbes Medi-Tech, Inc. Method of preventing and delaying onset of Alzheimer's disease and composition therefor
US6015824A (en) * 1998-02-10 2000-01-18 Hoffmann-La Roche Ag Pyrrolidine and piperidine derivatives and treatment of neurodegenerative disorders
TWI254043B (en) * 1999-06-08 2006-05-01 Hoffmann La Roche Ethanesulfonyl-piperidine derivatives having good affinity to N-methyl-D-aspartate (NMDA) receptor
ATE257827T1 (de) * 1999-07-21 2004-01-15 Hoffmann La Roche Triazolderivate
CN1178911C (zh) * 2000-04-20 2004-12-08 弗·哈夫曼-拉罗切有限公司 吡咯烷与哌啶衍生物和它们用于治疗神经变性疾病的用途
US6432985B2 (en) * 2000-04-25 2002-08-13 Hoffmann-La Roche Inc. Neuroprotective substituted piperidine compounds with activity as NMDA NR2B subtype selective antagonists
US7022882B2 (en) * 2000-10-06 2006-04-04 The Regents Of The University Of California NMDA receptor channel blocker with neuroprotective activity
US7005432B2 (en) * 2002-05-16 2006-02-28 Hoffman-La Roche Inc. Substituted imidazol-pyridazine derivatives
JP2009503520A (ja) * 2005-07-29 2009-01-29 リージェンツ オブ ザ ユニバーシティ オブ ミネソタ ベータアミロイド受容体及びその使用

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