RU2731095C2 - Производное 5-этил-4-метил-пиразол-3-карбоксамида, обладающее активностью агониста taar - Google Patents
Производное 5-этил-4-метил-пиразол-3-карбоксамида, обладающее активностью агониста taar Download PDFInfo
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- RU2731095C2 RU2731095C2 RU2018134262A RU2018134262A RU2731095C2 RU 2731095 C2 RU2731095 C2 RU 2731095C2 RU 2018134262 A RU2018134262 A RU 2018134262A RU 2018134262 A RU2018134262 A RU 2018134262A RU 2731095 C2 RU2731095 C2 RU 2731095C2
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- taar
- htaar1
- pyrazole
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Landscapes
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Applications Claiming Priority (3)
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| EP16160790 | 2016-03-17 | ||
| EP16160790.8 | 2016-03-17 | ||
| PCT/EP2017/055885 WO2017157873A1 (en) | 2016-03-17 | 2017-03-14 | 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of taar |
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| RU2018134262A RU2018134262A (ru) | 2020-04-17 |
| RU2018134262A3 RU2018134262A3 (enExample) | 2020-04-17 |
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| CN114144412A (zh) * | 2019-07-11 | 2022-03-04 | 豪夫迈·罗氏有限公司 | 用于制备经取代的吡唑衍生物的方法 |
| AU2021238632A1 (en) * | 2020-03-19 | 2022-07-14 | F. Hoffmann-La Roche Ag | Salts and crystalline forms of a TAAR1 agonist |
| EP4430032A1 (en) | 2021-11-08 | 2024-09-18 | F. Hoffmann-La Roche AG | Catalytic hydrogenation of aromatic nitro compounds |
| CN114288304A (zh) * | 2021-12-31 | 2022-04-08 | 江苏海洋大学 | 一种抗精神分裂症组合物及其应用 |
| AR129909A1 (es) | 2022-07-15 | 2024-10-09 | Hoffmann La Roche | Cetorreductasa mutante con mayor actividad de cetorreductasa así como métodos y usos de esta |
| KR20250044870A (ko) | 2022-08-12 | 2025-04-01 | 에프. 호프만-라 로슈 아게 | 5-에틸-4-메틸-n-[4-[(2s) 모르폴린-2-일]페닐]-1h-피라졸-3-카르복스아미드를 포함하는 약제학적 조성물 |
| EP4568654A1 (en) * | 2022-08-12 | 2025-06-18 | F. Hoffmann-La Roche AG | Use of co-processed excipients in continuous manufacturing of solid dosage forms |
| WO2024118488A1 (en) * | 2022-11-28 | 2024-06-06 | Sumitomo Pharma America, Inc. | 2-phenylmorpholine and 2-phenyl(thio)morpholine compounds and uses thereof |
| TW202444712A (zh) * | 2023-04-28 | 2024-11-16 | 大陸商江蘇豪森藥業集團有限公司 | 一種嗎啉雜環類化合物的鹽及其製備方法和應用 |
| WO2024258900A2 (en) * | 2023-06-13 | 2024-12-19 | University Of Georgia Research Foundation, Inc. | Plasmodium falciparum blood stage inhibitors |
Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2012129737A (ru) * | 2009-12-22 | 2014-01-27 | Ф. Хоффманн-Ля Рош Аг | Замещенные бензамидные производные |
| WO2014041106A1 (en) * | 2012-09-17 | 2014-03-20 | F. Hoffmann-La Roche Ag | Triazole carboxamide derivatives |
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