JP2017535550A5 - - Google Patents

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JP2017535550A5
JP2017535550A5 JP2017526116A JP2017526116A JP2017535550A5 JP 2017535550 A5 JP2017535550 A5 JP 2017535550A5 JP 2017526116 A JP2017526116 A JP 2017526116A JP 2017526116 A JP2017526116 A JP 2017526116A JP 2017535550 A5 JP2017535550 A5 JP 2017535550A5
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trka
crystalline form
composition
cancer
trkb
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JP2017526116A
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JP2017535550A (ja
JP6914834B2 (ja
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JP2017526116A 2014-11-16 2015-11-16 （Ｓ）−Ｎ−（５−（（Ｒ）−２−（２，５−ジフルオロフェニル）−ピロリジン−１−イル）−ピラゾロ［１，５−ａ］ピリミジン−３−イル）−３−ヒドロキシピロリジン−１−カルボキサミド硫酸水素塩の結晶形 Active JP6914834B2 (ja)

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JP2021116073A JP2021169496A (ja) 2014-11-16 2021-07-14 （Ｓ）−Ｎ−（５−（（Ｒ）−２−（２，５−ジフルオロフェニル）−ピロリジン−１−イル）−ピラゾロ［１，５−ａ］ピリミジン−３−イル）−３−ヒドロキシピロリジン−１−カルボキサミド硫酸水素塩の結晶形

Applications Claiming Priority (5)

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US201462080374P 2014-11-16 2014-11-16
US62/080,374 2014-11-16
US201562169545P 2015-06-01 2015-06-01
US62/169,545 2015-06-01
PCT/US2015/060953 WO2016077841A1 (en) 2014-11-16 2015-11-16 Crystalline form of (s)-n-(5-((r)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide hydrogen sulfate

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JP2021116073A Division JP2021169496A (ja) 2014-11-16 2021-07-14 （Ｓ）−Ｎ−（５−（（Ｒ）−２−（２，５−ジフルオロフェニル）−ピロリジン−１−イル）−ピラゾロ［１，５−ａ］ピリミジン−３−イル）−３−ヒドロキシピロリジン−１−カルボキサミド硫酸水素塩の結晶形

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JP2017535550A JP2017535550A (ja) 2017-11-30
JP2017535550A5 true JP2017535550A5 (OSRAM) 2018-12-27
JP6914834B2 JP6914834B2 (ja) 2021-08-04

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JP2017526116A Active JP6914834B2 (ja) 2014-11-16 2015-11-16 （Ｓ）−Ｎ−（５−（（Ｒ）−２−（２，５−ジフルオロフェニル）−ピロリジン−１−イル）−ピラゾロ［１，５−ａ］ピリミジン−３−イル）−３−ヒドロキシピロリジン−１−カルボキサミド硫酸水素塩の結晶形
JP2021116073A Pending JP2021169496A (ja) 2014-11-16 2021-07-14 （Ｓ）−Ｎ−（５−（（Ｒ）−２−（２，５−ジフルオロフェニル）−ピロリジン−１−イル）−ピラゾロ［１，５−ａ］ピリミジン−３−イル）−３−ヒドロキシピロリジン−１−カルボキサミド硫酸水素塩の結晶形

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Country Status (30)

Country Link
US (5) US10799505B2 (OSRAM)
EP (2) EP3218380B1 (OSRAM)
JP (2) JP6914834B2 (OSRAM)
KR (1) KR102649887B1 (OSRAM)
CN (2) CN107428760B (OSRAM)
AU (1) AU2015346046B2 (OSRAM)
BR (1) BR112017010141A2 (OSRAM)
CA (1) CA2967951C (OSRAM)
CL (1) CL2017001249A1 (OSRAM)
CO (1) CO2017005483A2 (OSRAM)
CR (1) CR20170263A (OSRAM)
DK (1) DK3699181T3 (OSRAM)
ES (1) ES2941630T3 (OSRAM)
FI (1) FI3699181T3 (OSRAM)
HK (1) HK1244483A1 (OSRAM)
HR (1) HRP20230271T1 (OSRAM)
HU (1) HUE061448T2 (OSRAM)
IL (2) IL290905B2 (OSRAM)
LT (1) LT3699181T (OSRAM)
MX (2) MX376478B (OSRAM)
PH (2) PH12017500900A1 (OSRAM)
PL (1) PL3699181T3 (OSRAM)
PT (1) PT3699181T (OSRAM)
RS (1) RS64122B1 (OSRAM)
SG (1) SG11201703962XA (OSRAM)
SI (1) SI3699181T1 (OSRAM)
TW (2) TWI746426B (OSRAM)
UA (1) UA123044C2 (OSRAM)
WO (1) WO2016077841A1 (OSRAM)
ZA (1) ZA201703501B (OSRAM)

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