JP2017524704A5 - - Google Patents
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- Publication number
- JP2017524704A5 JP2017524704A5 JP2017504421A JP2017504421A JP2017524704A5 JP 2017524704 A5 JP2017524704 A5 JP 2017524704A5 JP 2017504421 A JP2017504421 A JP 2017504421A JP 2017504421 A JP2017504421 A JP 2017504421A JP 2017524704 A5 JP2017524704 A5 JP 2017524704A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutically acceptable
- substituted
- acceptable salt
- compound according
- hydroxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- RHASGUGQMCVYMQ-UHFFFAOYSA-N N#Cc(cc1)ccc1-c1cnccc1SCC1(CC(O)=O)CC1 Chemical compound N#Cc(cc1)ccc1-c1cnccc1SCC1(CC(O)=O)CC1 RHASGUGQMCVYMQ-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201410398333.4 | 2014-08-13 | ||
| CN201410398333.4A CN105439946B (zh) | 2014-08-13 | 2014-08-13 | 羧酸化合物及其制备方法和用途 |
| PCT/CN2015/086605 WO2016023460A1 (zh) | 2014-08-13 | 2015-08-11 | 羧酸化合物及其制备方法和用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017524704A JP2017524704A (ja) | 2017-08-31 |
| JP2017524704A5 true JP2017524704A5 (enExample) | 2018-09-13 |
| JP6568929B2 JP6568929B2 (ja) | 2019-08-28 |
Family
ID=55303876
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017504421A Active JP6568929B2 (ja) | 2014-08-13 | 2015-08-11 | カルボン酸化合物、その製造方法および使用 |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US9809580B2 (enExample) |
| EP (1) | EP3181557B1 (enExample) |
| JP (1) | JP6568929B2 (enExample) |
| KR (1) | KR102474640B1 (enExample) |
| CN (2) | CN105439946B (enExample) |
| AU (1) | AU2015303597B2 (enExample) |
| CA (1) | CA2956045C (enExample) |
| ES (1) | ES2942259T3 (enExample) |
| IL (1) | IL250524B (enExample) |
| NZ (1) | NZ729037A (enExample) |
| WO (1) | WO2016023460A1 (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105439946B (zh) * | 2014-08-13 | 2018-02-02 | 益方生物科技(上海)有限公司 | 羧酸化合物及其制备方法和用途 |
| WO2017114352A1 (en) * | 2015-12-28 | 2017-07-06 | Chongqing Fochon Pharmaceutical Co., Ltd. | Indolizine derivatives, composition and methods of use |
| CN105884807A (zh) * | 2016-04-26 | 2016-08-24 | 昆药集团股份有限公司 | 硼酸频那醇酯衍生物的制备方法、硫代乙酸盐化合物的制备方法 |
| CN106748987B (zh) * | 2016-11-18 | 2019-05-31 | 昆药集团股份有限公司 | 2-((3-(4-氰基萘-1-基)吡啶-4-基)硫基)-2-甲基丙酸钠盐的晶型 |
| TW201922706A (zh) * | 2017-10-04 | 2019-06-16 | 日商日本煙草產業股份有限公司 | 含氮雜芳基化合物及該化合物之醫藥用途 |
| CN108069940B (zh) * | 2017-12-20 | 2021-04-30 | 广东赛烽医药科技有限公司 | 硫代乙酸化合物、组合物及其应用 |
| CN108084153A (zh) * | 2017-12-20 | 2018-05-29 | 广东赛烽医药科技有限公司 | 吡啶基硫代乙酸化合物、组合物及其应用 |
| CN108440397B (zh) * | 2018-03-06 | 2020-06-05 | 南方医科大学 | 3-(萘-1-甲基取代)吡啶衍生物及其合成方法和应用 |
| WO2019183835A1 (en) * | 2018-03-28 | 2019-10-03 | Inventisbio Shanghai Ltd. | Novel salt forms of urat-1 inhibitors |
| CN108484494B (zh) * | 2018-06-15 | 2021-07-30 | 沈阳药科大学 | 2-氧代-1,2-二氢吡啶-4-甲酸类化合物 |
| CN111943957B (zh) * | 2019-05-17 | 2023-01-06 | 中国医学科学院药物研究所 | 喹啉甲酰胺类化合物及其制备方法和用途 |
| CN113493407B (zh) * | 2020-04-03 | 2025-01-28 | 中国医学科学院药物研究所 | 一种吡啶类化合物及其制法和药物用途 |
| AR124985A1 (es) * | 2021-03-01 | 2023-05-24 | Orion Corp | Nuevas formas de sal de un inhibidor de cyp11a1 estructurado en 4h-piran-4-ona |
| WO2022184977A1 (en) * | 2021-03-01 | 2022-09-09 | Orion Corporation | Solid forms of a 4h-pyran-4-one structured cyp11a1 inhibitor |
| CN113979931B (zh) * | 2021-10-08 | 2023-06-13 | 南方医科大学 | 一种吡啶3-胺衍生物及其制备方法和应用 |
| JP7792730B2 (ja) * | 2022-04-27 | 2025-12-26 | 杭州新元素▲薬▼▲業▼有限公司 | 尿酸を降下させるために使用できる化合物 |
| WO2025060752A1 (zh) * | 2023-09-19 | 2025-03-27 | 湘北威尔曼制药股份有限公司 | 一种硫醚衍生物及其制备方法和应用 |
| WO2025060786A1 (zh) * | 2023-09-19 | 2025-03-27 | 湘北威尔曼制药股份有限公司 | 一种六元并五元稠环衍生物及其制备方法和应用 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19541146A1 (de) * | 1995-10-25 | 1997-04-30 | Schering Ag | Imidazolderivate und deren Verwendung als Stickstoffmonoxid-Synthase-Inhibitoren |
| SE0301010D0 (sv) * | 2003-04-07 | 2003-04-07 | Astrazeneca Ab | Novel compounds |
| FR2903984B1 (fr) * | 2006-07-24 | 2008-10-03 | Genfit Sa | Derives d'imidazolones substitues, preparation et utilisations |
| EP2471792B1 (en) * | 2009-08-28 | 2014-04-09 | Daiichi Sankyo Company, Limited | 3-(biaryloxy) propionic acid derivative |
| CA2802692C (en) * | 2010-06-16 | 2016-01-05 | Ardea Biosciences, Inc. | Phenylthioacetate compounds useful as uricosuric agents |
| AR081930A1 (es) * | 2010-06-16 | 2012-10-31 | Ardea Biosciences Inc | Compuestos de tioacetato |
| BR112014010495A2 (pt) * | 2011-11-03 | 2017-04-25 | Ardea Biosciences Inc | composto de piridina 3,4-di-substituído, métodos de uso e composições compreendendo o mesmo |
| CA2860553C (en) * | 2012-01-04 | 2016-08-23 | Pfizer Limited | N-aminosulfonyl benzamides |
| WO2013158422A1 (en) * | 2012-04-17 | 2013-10-24 | E. I. Du Pont De Nemours And Company | Heterocyclic compounds for controlling invertebrate pests |
| CN105439946B (zh) * | 2014-08-13 | 2018-02-02 | 益方生物科技(上海)有限公司 | 羧酸化合物及其制备方法和用途 |
-
2014
- 2014-08-13 CN CN201410398333.4A patent/CN105439946B/zh active Active
-
2015
- 2015-08-11 US US15/501,387 patent/US9809580B2/en active Active
- 2015-08-11 CN CN201580043042.6A patent/CN106573908B/zh active Active
- 2015-08-11 EP EP15831615.8A patent/EP3181557B1/en active Active
- 2015-08-11 NZ NZ729037A patent/NZ729037A/en unknown
- 2015-08-11 CA CA2956045A patent/CA2956045C/en active Active
- 2015-08-11 ES ES15831615T patent/ES2942259T3/es active Active
- 2015-08-11 AU AU2015303597A patent/AU2015303597B2/en active Active
- 2015-08-11 JP JP2017504421A patent/JP6568929B2/ja active Active
- 2015-08-11 KR KR1020177006929A patent/KR102474640B1/ko active Active
- 2015-08-11 WO PCT/CN2015/086605 patent/WO2016023460A1/zh not_active Ceased
-
2017
- 2017-02-09 IL IL250524A patent/IL250524B/en active IP Right Grant
- 2017-10-03 US US15/723,785 patent/US9856239B1/en active Active
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