JP2012525393A5 - - Google Patents

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JP2012525393A5
JP2012525393A5 JP2012508590A JP2012508590A JP2012525393A5 JP 2012525393 A5 JP2012525393 A5 JP 2012525393A5 JP 2012508590 A JP2012508590 A JP 2012508590A JP 2012508590 A JP2012508590 A JP 2012508590A JP 2012525393 A5 JP2012525393 A5 JP 2012525393A5
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Japan
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alkanyl
alkenyl
alkynyl
aryl
compound
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JP2012508590A
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JP5726171B2 (ja
JP2012525393A (ja
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Priority claimed from PCT/US2010/032568 external-priority patent/WO2010126888A1/en
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JP2012508590A 2009-05-01 2010-04-27 E−セレクチンおよびcxcr4ケモカイン受容体のヘテロ二官能性阻害剤 Active JP5726171B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17458009P 2009-05-01 2009-05-01
US61/174,580 2009-05-01
PCT/US2010/032568 WO2010126888A1 (en) 2009-05-01 2010-04-27 Heterobifunctional inhibitors of e-selectins and cxcr4 chemokine receptors

Publications (3)

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JP2012525393A JP2012525393A (ja) 2012-10-22
JP2012525393A5 true JP2012525393A5 (enExample) 2014-10-09
JP5726171B2 JP5726171B2 (ja) 2015-05-27

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JP2012508590A Active JP5726171B2 (ja) 2009-05-01 2010-04-27 E−セレクチンおよびcxcr4ケモカイン受容体のヘテロ二官能性阻害剤

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US (2) US8410066B2 (enExample)
EP (1) EP2424544A1 (enExample)
JP (1) JP5726171B2 (enExample)
CN (1) CN102421441B (enExample)
AU (1) AU2010241807B2 (enExample)
CA (1) CA2760292A1 (enExample)
WO (1) WO2010126888A1 (enExample)

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JP2023529485A (ja) 2020-06-14 2023-07-10 グリコミメティクス, インコーポレイテッド E-セレクチン標的化を介して微小環境媒介耐性を克服するための組成物および方法
US20230364277A1 (en) * 2020-09-17 2023-11-16 Glycomimetics, Inc. E-selectin targeting agents
WO2023014690A1 (en) 2021-08-03 2023-02-09 Glycomimetics, Inc. Compositions and methods for overcoming microenvironment-mediated resistance via e-selectin targeting

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