CN105439946B - 羧酸化合物及其制备方法和用途 - Google Patents

羧酸化合物及其制备方法和用途 Download PDF

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CN105439946B
CN105439946B CN201410398333.4A CN201410398333A CN105439946B CN 105439946 B CN105439946 B CN 105439946B CN 201410398333 A CN201410398333 A CN 201410398333A CN 105439946 B CN105439946 B CN 105439946B
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added
compound
synthesis
methyl
ethyl acetate
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CN105439946A (zh
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江岳恒
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Yifang Biotechnology Shanghai Co ltd
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Yi Fang Biotechnology (shanghai) Co Ltd
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Priority to CN201410398333.4A priority Critical patent/CN105439946B/zh
Application filed by Yi Fang Biotechnology (shanghai) Co Ltd filed Critical Yi Fang Biotechnology (shanghai) Co Ltd
Priority to EP15831615.8A priority patent/EP3181557B1/en
Priority to ES15831615T priority patent/ES2942259T3/es
Priority to KR1020177006929A priority patent/KR102474640B1/ko
Priority to CA2956045A priority patent/CA2956045C/en
Priority to NZ729037A priority patent/NZ729037A/en
Priority to AU2015303597A priority patent/AU2015303597B2/en
Priority to CN201580043042.6A priority patent/CN106573908B/zh
Priority to PCT/CN2015/086605 priority patent/WO2016023460A1/zh
Priority to JP2017504421A priority patent/JP6568929B2/ja
Priority to US15/501,387 priority patent/US9809580B2/en
Publication of CN105439946A publication Critical patent/CN105439946A/zh
Priority to IL250524A priority patent/IL250524B/en
Priority to US15/723,785 priority patent/US9856239B1/en
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    • C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418—Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
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    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
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    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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CN201410398333.4A 2014-08-13 2014-08-13 羧酸化合物及其制备方法和用途 Active CN105439946B (zh)

Priority Applications (13)

Application Number Priority Date Filing Date Title
CN201410398333.4A CN105439946B (zh) 2014-08-13 2014-08-13 羧酸化合物及其制备方法和用途
US15/501,387 US9809580B2 (en) 2014-08-13 2015-08-11 Carboxylic acid compound, method for preparation thereof, and use thereof
KR1020177006929A KR102474640B1 (ko) 2014-08-13 2015-08-11 카르복실산 화합물, 이의 제조방법, 및 이의 용도
CA2956045A CA2956045C (en) 2014-08-13 2015-08-11 Carboxylic acid compound, method for preparation thereof, and use thereof
NZ729037A NZ729037A (en) 2014-08-13 2015-08-11 Carboxylic acid compound, method for preparation thereof, and use thereof
AU2015303597A AU2015303597B2 (en) 2014-08-13 2015-08-11 Carboxylic acid compound, method for preparation thereof, and use thereof
EP15831615.8A EP3181557B1 (en) 2014-08-13 2015-08-11 Carboxylic acid compound, method for preparation thereof, and use thereof
PCT/CN2015/086605 WO2016023460A1 (zh) 2014-08-13 2015-08-11 羧酸化合物及其制备方法和用途
JP2017504421A JP6568929B2 (ja) 2014-08-13 2015-08-11 カルボン酸化合物、その製造方法および使用
ES15831615T ES2942259T3 (es) 2014-08-13 2015-08-11 Compuesto de ácido carboxílico, método para la preparación del mismo y uso del mismo
CN201580043042.6A CN106573908B (zh) 2014-08-13 2015-08-11 羧酸化合物及其制备方法和用途
IL250524A IL250524B (en) 2014-08-13 2017-02-09 Carboxylic acid compound, method for its preparation and use
US15/723,785 US9856239B1 (en) 2014-08-13 2017-10-03 Carboxylic acid compound, method for preparation thereof, and use thereof

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