JP2014501740A5 - - Google Patents
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- JP2014501740A5 JP2014501740A5 JP2013544980A JP2013544980A JP2014501740A5 JP 2014501740 A5 JP2014501740 A5 JP 2014501740A5 JP 2013544980 A JP2013544980 A JP 2013544980A JP 2013544980 A JP2013544980 A JP 2013544980A JP 2014501740 A5 JP2014501740 A5 JP 2014501740A5
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- JP
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- Prior art keywords
- pharmaceutically acceptable
- acceptable salt
- effective amount
- medicament
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201061426773P | 2010-12-23 | 2010-12-23 | |
| US61/426,773 | 2010-12-23 | ||
| PCT/CN2011/074569 WO2012159262A1 (en) | 2011-05-24 | 2011-05-24 | Selective glycosidase inhibitors and uses thereof |
| CNPCT/CN2011/074569 | 2011-05-24 | ||
| US201161507684P | 2011-07-14 | 2011-07-14 | |
| US61/507,684 | 2011-07-14 | ||
| PCT/CA2011/001397 WO2012083435A1 (en) | 2010-12-23 | 2011-12-21 | Selective glycosidase inhibitors and uses thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015230912A Division JP6322177B2 (ja) | 2010-12-23 | 2015-11-26 | 選択的グルコシダーゼインヒビターおよびその使用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2014501740A JP2014501740A (ja) | 2014-01-23 |
| JP2014501740A5 true JP2014501740A5 (enExample) | 2015-10-15 |
| JP5861194B2 JP5861194B2 (ja) | 2016-02-16 |
Family
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Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013544980A Expired - Fee Related JP5861194B2 (ja) | 2010-12-23 | 2011-12-21 | 選択的グルコシダーゼインヒビターおよびその使用 |
| JP2015230912A Active JP6322177B2 (ja) | 2010-12-23 | 2015-11-26 | 選択的グルコシダーゼインヒビターおよびその使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015230912A Active JP6322177B2 (ja) | 2010-12-23 | 2015-11-26 | 選択的グルコシダーゼインヒビターおよびその使用 |
Country Status (26)
| Country | Link |
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| CA2599843C (en) * | 2005-03-01 | 2013-08-27 | Simon Fraser University | Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof |
| JP5380293B2 (ja) | 2006-08-31 | 2014-01-08 | サイモン・フレーザー・ユニバーシティ | 選択的グリコシダーゼ阻害剤およびその使用 |
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| US9120781B2 (en) | 2010-05-11 | 2015-09-01 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
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| RU2609210C2 (ru) * | 2010-12-23 | 2017-01-31 | Алектос Терапьютикс Инк. | Селективные ингибиторы гликозидазы и их применение |
| WO2012126091A1 (en) | 2011-03-24 | 2012-09-27 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| WO2012129651A1 (en) | 2011-03-31 | 2012-10-04 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2726468B1 (en) | 2011-06-27 | 2017-04-12 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| RU2625308C2 (ru) * | 2011-06-27 | 2017-07-13 | Алектос Терапьютикс Инк. | Селективные ингибиторы гликозидазы и их применение |
| US9701693B2 (en) | 2011-06-27 | 2017-07-11 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
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| EP2890676B1 (en) | 2012-08-31 | 2018-12-05 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| EP2890675A4 (en) | 2012-08-31 | 2016-01-13 | Alectos Therapeutics Inc | GLYCOSIDASE INHIBITORS AND USES THEREOF |
| KR20150079711A (ko) * | 2012-10-31 | 2015-07-08 | 알렉토스 테라퓨틱스 인크. | 글리코시다아제 저해제 및 이의 용도 |
| WO2014100934A1 (en) | 2012-12-24 | 2014-07-03 | Merck Sharp & Dohme Corp. | Glycosidase inhibitors and uses thereof |
| SG11201701315VA (en) | 2014-08-28 | 2017-03-30 | Asceneuron Sa | Glycosidase inhibitors |
| KR101777164B1 (ko) | 2015-07-20 | 2017-09-11 | 순천향대학교 산학협력단 | O-GlcNAc 트랜스퍼레즈 억제제용 UDP-GlcNAc의 C1-포스포네이트 유도체 |
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| JP2019506430A (ja) | 2016-02-25 | 2019-03-07 | エースニューロン・ソシエテ・アノニム | グリコシダーゼ阻害剤 |
| CA3014572C (en) | 2016-02-25 | 2023-10-03 | Asceneuron S.A. | Acid addition salts of piperazine derivatives |
| US11261183B2 (en) | 2016-02-25 | 2022-03-01 | Asceneuron Sa | Sulfoximine glycosidase inhibitors |
| MX2018010192A (es) | 2016-02-25 | 2019-01-31 | Asceneuron S A | Inhibidores de glucosidasa. |
| EP3672959A1 (en) | 2017-08-24 | 2020-07-01 | Asceneuron SA | Linear glycosidase inhibitors |
| CN107814773B (zh) * | 2017-11-13 | 2020-05-22 | 西安交通大学 | 含有喹唑啉酮的二芳基脲类化合物及其制备方法和应用 |
| JP2021527662A (ja) * | 2018-06-20 | 2021-10-14 | ヤンセン ファーマシューティカ エヌ．ベー． | Ｏｇａ阻害化合物 |
| AU2019324522B2 (en) | 2018-08-22 | 2024-11-14 | Asceneuron S. A. | Succinate and fumarate acid addition salts of piperazine derivatives useful as glycosidase inhibitors |
| US12016852B2 (en) | 2018-08-22 | 2024-06-25 | Asceneuron Sa | Pyrrolidine glycosidase inhibitors |
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| US11795165B2 (en) | 2018-08-22 | 2023-10-24 | Asceneuron Sa | Tetrahydro-benzoazepine glycosidase inhibitors |
| CN114174263B (zh) * | 2019-05-10 | 2025-01-10 | 阿勒克图治疗公司 | 非溶酶体葡糖神经酰胺酶抑制剂及其用途 |
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