JP2011529858A5 - - Google Patents

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Publication number
JP2011529858A5
JP2011529858A5 JP2011520297A JP2011520297A JP2011529858A5 JP 2011529858 A5 JP2011529858 A5 JP 2011529858A5 JP 2011520297 A JP2011520297 A JP 2011520297A JP 2011520297 A JP2011520297 A JP 2011520297A JP 2011529858 A5 JP2011529858 A5 JP 2011529858A5
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JP
Japan
Prior art keywords
disease
compound
pharmaceutically acceptable
acceptable salt
composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2011520297A
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English (en)
Japanese (ja)
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JP2011529858A (ja
JP5687194B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/CA2009/001088 external-priority patent/WO2010012107A1/en
Publication of JP2011529858A publication Critical patent/JP2011529858A/ja
Publication of JP2011529858A5 publication Critical patent/JP2011529858A5/ja
Application granted granted Critical
Publication of JP5687194B2 publication Critical patent/JP5687194B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2011520297A 2008-08-01 2009-07-31 選択的グリコシダーゼインヒビターおよびその使用 Expired - Fee Related JP5687194B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8553808P 2008-08-01 2008-08-01
US61/085,538 2008-08-01
PCT/CA2009/001088 WO2010012107A1 (en) 2008-08-01 2009-07-31 Selective glycosidase inhibitors and uses thereof

Publications (3)

Publication Number Publication Date
JP2011529858A JP2011529858A (ja) 2011-12-15
JP2011529858A5 true JP2011529858A5 (enExample) 2012-09-06
JP5687194B2 JP5687194B2 (ja) 2015-03-18

Family

ID=41609897

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011520297A Expired - Fee Related JP5687194B2 (ja) 2008-08-01 2009-07-31 選択的グリコシダーゼインヒビターおよびその使用

Country Status (6)

Country Link
US (1) US9079868B2 (enExample)
EP (1) EP2321289A4 (enExample)
JP (1) JP5687194B2 (enExample)
AU (1) AU2009276223B2 (enExample)
CA (1) CA2732336A1 (enExample)
WO (1) WO2010012107A1 (enExample)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2819464A1 (en) * 2005-03-01 2006-09-08 Matthew Macauley Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof
EP2057171A4 (en) 2006-08-31 2010-04-21 Univ Fraser Simon SELECTIVE GLYCOSIDASE INHIBITORS AND APPLICATIONS THEREOF
US9120781B2 (en) 2010-05-11 2015-09-01 Simon Fraser University Selective glycosidase inhibitors and uses thereof
US8901087B2 (en) 2010-11-08 2014-12-02 Merck Sharp & Dohme Corp. Selective glycosidase inhibitors and uses thereof
EP2638052B1 (en) 2010-11-08 2017-03-22 Alectos Therapeutics, Inc. Selective glycosidase inhibitors and uses thereof
TW201249848A (en) 2010-11-08 2012-12-16 Merck Sharp & Dohme Selective glycosidase inhibitors and uses thereof
CA2822493C (en) 2010-12-23 2018-11-20 Merck Sharp & Dohme Corp. Selective glycosidase inhibitors and uses thereof
WO2012159262A1 (en) * 2011-05-24 2012-11-29 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
US8927507B2 (en) 2011-03-24 2015-01-06 Ernest J. McEachern Selective glycosidase inhibitors and uses thereof
US9718854B2 (en) 2011-03-31 2017-08-01 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
US9199949B2 (en) 2011-06-27 2015-12-01 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
JP6147737B2 (ja) 2011-06-27 2017-06-14 アレクトス・セラピューティクス・インコーポレイテッド 選択的グリコシダーゼ阻害剤およびその使用
EP2726492B1 (en) 2011-06-27 2017-11-01 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
US9126957B2 (en) * 2011-08-18 2015-09-08 Merck Sharp & Dohme Corp. Selective glycosidase inhibitors and uses thereof
US20150010527A1 (en) 2012-02-01 2015-01-08 Protalix Ltd. Dnase i polypeptides, polynucleotides encoding same, methods of producing dnase i and uses thereof in therapy
AU2013259892B2 (en) 2012-05-08 2017-09-14 Alectos Therapeutics Inc. Permeable glycosidase inhibitors and uses thereof
EP2890676B1 (en) 2012-08-31 2018-12-05 Alectos Therapeutics Inc. Glycosidase inhibitors and uses thereof
EP2890675A4 (en) 2012-08-31 2016-01-13 Alectos Therapeutics Inc GLYCOSIDASE INHIBITORS AND USES THEREOF
US9695197B2 (en) 2012-10-31 2017-07-04 Alectos Therapeutics Inc. Glycosidase inhibitors and uses thereof
WO2014136113A1 (en) 2013-03-06 2014-09-12 Protalix Ltd. Chimeric polypeptides, polynucleotides encoding same, cells expressing same and methods of producing same
WO2019173506A1 (en) * 2018-03-07 2019-09-12 The Broad Institute, Inc. Cyclopentaimidazolones for the treatment of cancer
WO2024083820A1 (en) 2022-10-18 2024-04-25 Institut National de la Santé et de la Recherche Médicale Method and composition for determining the level of o-glcnacylation in horses

Family Cites Families (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1131672A (zh) * 1994-11-22 1996-09-25 生化学工业株式会社 氨基环戊烷衍生物
JPH11349541A (ja) * 1998-06-08 1999-12-21 Sankyo Co Ltd アロサミゾリン誘導体の新規な中間体
US7214373B2 (en) 2001-07-24 2007-05-08 Yale University Methods, compositions and kits relating to chitinases and chitinase-like molecules and inflammatory disease
CA2819464A1 (en) * 2005-03-01 2006-09-08 Matthew Macauley Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof
EP2057171A4 (en) * 2006-08-31 2010-04-21 Univ Fraser Simon SELECTIVE GLYCOSIDASE INHIBITORS AND APPLICATIONS THEREOF
EP2113589A1 (en) * 2008-04-29 2009-11-04 Total Petrochemicals Research Feluy Fibers and nonwovens with improved bonding properties
AU2009276222B2 (en) * 2008-08-01 2015-03-05 Simon Fraser University Selective glycosidase inhibitors and uses thereof
WO2010037207A1 (en) * 2008-09-16 2010-04-08 Simon Fraser University Selective glycosidase inhibitors and uses thereof
US9120781B2 (en) * 2010-05-11 2015-09-01 Simon Fraser University Selective glycosidase inhibitors and uses thereof
TW201249848A (en) 2010-11-08 2012-12-16 Merck Sharp & Dohme Selective glycosidase inhibitors and uses thereof
EP2638052B1 (en) * 2010-11-08 2017-03-22 Alectos Therapeutics, Inc. Selective glycosidase inhibitors and uses thereof
CA2822493C (en) * 2010-12-23 2018-11-20 Merck Sharp & Dohme Corp. Selective glycosidase inhibitors and uses thereof
US8927507B2 (en) * 2011-03-24 2015-01-06 Ernest J. McEachern Selective glycosidase inhibitors and uses thereof
US9718854B2 (en) * 2011-03-31 2017-08-01 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
US9199949B2 (en) 2011-06-27 2015-12-01 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
EP2726492B1 (en) 2011-06-27 2017-11-01 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
JP6147737B2 (ja) 2011-06-27 2017-06-14 アレクトス・セラピューティクス・インコーポレイテッド 選択的グリコシダーゼ阻害剤およびその使用
US9126957B2 (en) 2011-08-18 2015-09-08 Merck Sharp & Dohme Corp. Selective glycosidase inhibitors and uses thereof
AU2013259892B2 (en) 2012-05-08 2017-09-14 Alectos Therapeutics Inc. Permeable glycosidase inhibitors and uses thereof
US20150299122A1 (en) 2012-08-31 2015-10-22 Alectos Therapeutics Inc. Glycosidase inhibitors and uses thereof
US9522883B2 (en) 2012-08-31 2016-12-20 Alectos Therapeutics Inc. Glycosidase inhibitors and uses thereof
EP2890675A4 (en) 2012-08-31 2016-01-13 Alectos Therapeutics Inc GLYCOSIDASE INHIBITORS AND USES THEREOF
EP2890676B1 (en) 2012-08-31 2018-12-05 Alectos Therapeutics Inc. Glycosidase inhibitors and uses thereof
US9695197B2 (en) 2012-10-31 2017-07-04 Alectos Therapeutics Inc. Glycosidase inhibitors and uses thereof
WO2014100934A1 (en) 2012-12-24 2014-07-03 Merck Sharp & Dohme Corp. Glycosidase inhibitors and uses thereof

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