JP5687194B2 - 選択的グリコシダーゼインヒビターおよびその使用 - Google Patents
選択的グリコシダーゼインヒビターおよびその使用 Download PDFInfo
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- JP5687194B2 JP5687194B2 JP2011520297A JP2011520297A JP5687194B2 JP 5687194 B2 JP5687194 B2 JP 5687194B2 JP 2011520297 A JP2011520297 A JP 2011520297A JP 2011520297 A JP2011520297 A JP 2011520297A JP 5687194 B2 JP5687194 B2 JP 5687194B2
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Classifications
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Landscapes
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| US8553808P | 2008-08-01 | 2008-08-01 | |
| US61/085,538 | 2008-08-01 | ||
| PCT/CA2009/001088 WO2010012107A1 (en) | 2008-08-01 | 2009-07-31 | Selective glycosidase inhibitors and uses thereof |
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| JP2011529858A JP2011529858A (ja) | 2011-12-15 |
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| CA (1) | CA2732336A1 (enExample) |
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| EP1869060B1 (en) * | 2005-03-01 | 2012-08-15 | Simon Fraser University | Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof |
| CA2661582C (en) | 2006-08-31 | 2015-09-29 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| WO2011140640A1 (en) | 2010-05-11 | 2011-11-17 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| US8933040B2 (en) | 2010-11-08 | 2015-01-13 | Craig A. Coburn | Selective glycosidase inhibitors and uses thereof |
| TW201249848A (en) | 2010-11-08 | 2012-12-16 | Merck Sharp & Dohme | Selective glycosidase inhibitors and uses thereof |
| US8901087B2 (en) | 2010-11-08 | 2014-12-02 | Merck Sharp & Dohme Corp. | Selective glycosidase inhibitors and uses thereof |
| WO2012159262A1 (en) * | 2011-05-24 | 2012-11-29 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| LT2655388T (lt) | 2010-12-23 | 2016-11-10 | Alectos Therapeutics Inc. | Selektyvieji glikozidazės inhibitoriai ir jų panaudojimas |
| EP2688899B1 (en) | 2011-03-24 | 2017-02-22 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9718854B2 (en) | 2011-03-31 | 2017-08-01 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9701693B2 (en) | 2011-06-27 | 2017-07-11 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| WO2013000085A1 (en) | 2011-06-27 | 2013-01-03 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9409924B2 (en) | 2011-06-27 | 2016-08-09 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2744338B1 (en) * | 2011-08-18 | 2016-04-27 | Merck Sharp & Dohme Corp. | Selective glycosidase inhibitors and uses thereof |
| US9603906B2 (en) | 2012-02-01 | 2017-03-28 | Protalix Ltd. | Inhalable liquid formulations of DNase I |
| RU2707292C2 (ru) | 2012-05-08 | 2019-11-26 | Мерк Шарп И Доум Корп. | Проницаемые ингибиторы гликозидазы и их применения |
| WO2014032188A1 (en) | 2012-08-31 | 2014-03-06 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| US9670195B2 (en) | 2012-08-31 | 2017-06-06 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| AU2013337570B2 (en) | 2012-10-31 | 2018-01-18 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| AU2014224171B2 (en) | 2013-03-06 | 2018-02-01 | Protalix Ltd. | Tnf alpha inhibitor polypeptides, polynucleotides encoding same, cells expressing same and methods of producing same |
| WO2019173506A1 (en) * | 2018-03-07 | 2019-09-12 | The Broad Institute, Inc. | Cyclopentaimidazolones for the treatment of cancer |
| WO2024083820A1 (en) | 2022-10-18 | 2024-04-25 | Institut National de la Santé et de la Recherche Médicale | Method and composition for determining the level of o-glcnacylation in horses |
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| CN1131672A (zh) * | 1994-11-22 | 1996-09-25 | 生化学工业株式会社 | 氨基环戊烷衍生物 |
| JPH11349541A (ja) * | 1998-06-08 | 1999-12-21 | Sankyo Co Ltd | アロサミゾリン誘導体の新規な中間体 |
| US7214373B2 (en) | 2001-07-24 | 2007-05-08 | Yale University | Methods, compositions and kits relating to chitinases and chitinase-like molecules and inflammatory disease |
| EP1869060B1 (en) | 2005-03-01 | 2012-08-15 | Simon Fraser University | Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof |
| CA2661582C (en) | 2006-08-31 | 2015-09-29 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| EP2113589A1 (en) | 2008-04-29 | 2009-11-04 | Total Petrochemicals Research Feluy | Fibers and nonwovens with improved bonding properties |
| JP2011529857A (ja) | 2008-08-01 | 2011-12-15 | サイモン フレイザー ユニバーシティ | 選択的グリコシダーゼインヒビターおよびその使用 |
| AU2009299073B2 (en) | 2008-09-16 | 2015-04-02 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| WO2011140640A1 (en) | 2010-05-11 | 2011-11-17 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| TW201249848A (en) | 2010-11-08 | 2012-12-16 | Merck Sharp & Dohme | Selective glycosidase inhibitors and uses thereof |
| US8933040B2 (en) | 2010-11-08 | 2015-01-13 | Craig A. Coburn | Selective glycosidase inhibitors and uses thereof |
| LT2655388T (lt) | 2010-12-23 | 2016-11-10 | Alectos Therapeutics Inc. | Selektyvieji glikozidazės inhibitoriai ir jų panaudojimas |
| EP2688899B1 (en) | 2011-03-24 | 2017-02-22 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9718854B2 (en) | 2011-03-31 | 2017-08-01 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| WO2013000085A1 (en) | 2011-06-27 | 2013-01-03 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9409924B2 (en) | 2011-06-27 | 2016-08-09 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9701693B2 (en) | 2011-06-27 | 2017-07-11 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2744338B1 (en) | 2011-08-18 | 2016-04-27 | Merck Sharp & Dohme Corp. | Selective glycosidase inhibitors and uses thereof |
| RU2707292C2 (ru) | 2012-05-08 | 2019-11-26 | Мерк Шарп И Доум Корп. | Проницаемые ингибиторы гликозидазы и их применения |
| US9670195B2 (en) | 2012-08-31 | 2017-06-06 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| EP2890679A4 (en) | 2012-08-31 | 2016-05-04 | Alectos Therapeutics Inc | GLYCOSIDASE INHIBITORS AND USES THEREOF |
| WO2014032187A1 (en) | 2012-08-31 | 2014-03-06 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| WO2014032188A1 (en) | 2012-08-31 | 2014-03-06 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| AU2013337570B2 (en) | 2012-10-31 | 2018-01-18 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| WO2014100934A1 (en) | 2012-12-24 | 2014-07-03 | Merck Sharp & Dohme Corp. | Glycosidase inhibitors and uses thereof |
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- 2009-07-31 JP JP2011520297A patent/JP5687194B2/ja not_active Expired - Fee Related
- 2009-07-31 EP EP09802333A patent/EP2321289A4/en not_active Withdrawn
- 2009-07-31 WO PCT/CA2009/001088 patent/WO2010012107A1/en not_active Ceased
- 2009-07-31 AU AU2009276223A patent/AU2009276223B2/en not_active Ceased
- 2009-07-31 CA CA2732336A patent/CA2732336A1/en not_active Abandoned
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| EP2321289A4 (en) | 2011-11-16 |
| EP2321289A1 (en) | 2011-05-18 |
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| AU2009276223B2 (en) | 2015-04-02 |
| AU2009276223A1 (en) | 2010-02-04 |
| WO2010012107A1 (en) | 2010-02-04 |
| US20110237631A1 (en) | 2011-09-29 |
| US9079868B2 (en) | 2015-07-14 |
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