JP2013540102A - アミド結合を介して修飾されたグルカゴンスーパーファミリーのペプチドプロドラッグ - Google Patents
アミド結合を介して修飾されたグルカゴンスーパーファミリーのペプチドプロドラッグ Download PDFInfo
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- JP2013540102A JP2013540102A JP2013516609A JP2013516609A JP2013540102A JP 2013540102 A JP2013540102 A JP 2013540102A JP 2013516609 A JP2013516609 A JP 2013516609A JP 2013516609 A JP2013516609 A JP 2013516609A JP 2013540102 A JP2013540102 A JP 2013540102A
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- glucagon
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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| US61/358,188 | 2010-06-24 | ||
| PCT/US2011/040330 WO2011163012A2 (en) | 2010-06-24 | 2011-06-14 | Amide based glucagon superfamily peptide prodrugs |
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- 2011-06-14 EP EP11798640.6A patent/EP2588126A4/en not_active Withdrawn
- 2011-06-14 CN CN201180031415XA patent/CN103179979A/zh active Pending
- 2011-06-14 CA CA2796894A patent/CA2796894A1/en not_active Abandoned
- 2011-06-14 KR KR1020127033177A patent/KR20130102470A/ko not_active Withdrawn
- 2011-06-14 US US13/697,021 patent/US8778872B2/en active Active
- 2011-06-14 RU RU2013103093/04A patent/RU2580317C2/ru not_active IP Right Cessation
- 2011-06-14 WO PCT/US2011/040330 patent/WO2011163012A2/en not_active Ceased
- 2011-06-14 MX MX2012014576A patent/MX2012014576A/es not_active Application Discontinuation
- 2011-06-14 JP JP2013516609A patent/JP2013540102A/ja active Pending
- 2011-06-23 TW TW100121933A patent/TW201209062A/zh unknown
- 2011-06-23 AR ARP110102184A patent/AR081471A1/es unknown
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| WO2009099763A1 (en) * | 2008-01-30 | 2009-08-13 | Indiana University Research And Technology Corporation | Ester-based peptide prodrugs |
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Also Published As
| Publication number | Publication date |
|---|---|
| KR20130102470A (ko) | 2013-09-17 |
| RU2013103093A (ru) | 2014-07-27 |
| CN103179979A (zh) | 2013-06-26 |
| EP2588126A2 (en) | 2013-05-08 |
| RU2580317C2 (ru) | 2016-04-10 |
| MX2012014576A (es) | 2013-02-21 |
| TW201209062A (en) | 2012-03-01 |
| EP2588126A4 (en) | 2015-07-08 |
| US20130123462A1 (en) | 2013-05-16 |
| WO2011163012A3 (en) | 2013-07-11 |
| AR081471A1 (es) | 2012-09-05 |
| US8778872B2 (en) | 2014-07-15 |
| WO2011163012A2 (en) | 2011-12-29 |
| CA2796894A1 (en) | 2011-12-29 |
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