KR20130102470A - 아미드계 글루카곤 슈퍼패밀리 펩티드 프로드러그 - Google Patents
아미드계 글루카곤 슈퍼패밀리 펩티드 프로드러그 Download PDFInfo
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- KR20130102470A KR20130102470A KR1020127033177A KR20127033177A KR20130102470A KR 20130102470 A KR20130102470 A KR 20130102470A KR 1020127033177 A KR1020127033177 A KR 1020127033177A KR 20127033177 A KR20127033177 A KR 20127033177A KR 20130102470 A KR20130102470 A KR 20130102470A
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- Prior art keywords
- alkyl
- group
- glucagon
- amino acid
- peptide
- Prior art date
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| JP6017754B2 (ja) | 2007-02-15 | 2016-11-02 | インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーションＩｎｄｉａｎａ Ｕｎｉｖｅｒｓｉｔｙ Ｒｅｓｅａｒｃｈ Ａｎｄ Ｔｅｃｈｎｏｌｏｇｙ Ｃｏｒｐｏｒａｔｉｏｎ | グルカゴン／ｇｌｐ−１受容体コアゴニスト |
| KR101623985B1 (ko) | 2007-03-28 | 2016-05-25 | 프레지던트 앤드 펠로우즈 오브 하바드 칼리지 | 스티칭된 폴리펩티드 |
| US8981047B2 (en) | 2007-10-30 | 2015-03-17 | Indiana University Research And Technology Corporation | Glucagon antagonists |
| CA2702289A1 (en) | 2007-10-30 | 2009-05-07 | Indiana University Research And Technology Corporation | Compounds exhibiting glucagon antagonist and glp-1 agonist activity |
| JP2011511778A (ja) | 2008-01-30 | 2011-04-14 | インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーション | エステルに基づいたペプチドプロドラッグ |
| CA2728284C (en) | 2008-06-17 | 2019-09-10 | Richard D. Dimarchi | Glucagon/glp-1 receptor co-agonists |
| BRPI0915282A2 (pt) | 2008-06-17 | 2017-02-07 | Univ Indiana Res & Tech Corp | agonistas mistos baseados no gip para o tratamento de distúrbios metabólicos e obesidade |
| CN102245624B (zh) | 2008-12-19 | 2016-08-10 | 印第安纳大学研究及科技有限公司 | 基于酰胺的胰岛素前药 |
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-
2011
- 2011-06-14 CA CA2796894A patent/CA2796894A1/en not_active Abandoned
- 2011-06-14 KR KR1020127033177A patent/KR20130102470A/ko not_active Withdrawn
- 2011-06-14 JP JP2013516609A patent/JP2013540102A/ja active Pending
- 2011-06-14 US US13/697,021 patent/US8778872B2/en active Active
- 2011-06-14 EP EP11798640.6A patent/EP2588126A4/en not_active Withdrawn
- 2011-06-14 MX MX2012014576A patent/MX2012014576A/es not_active Application Discontinuation
- 2011-06-14 WO PCT/US2011/040330 patent/WO2011163012A2/en not_active Ceased
- 2011-06-14 RU RU2013103093/04A patent/RU2580317C2/ru not_active IP Right Cessation
- 2011-06-14 CN CN201180031415XA patent/CN103179979A/zh active Pending
- 2011-06-23 AR ARP110102184A patent/AR081471A1/es unknown
- 2011-06-23 TW TW100121933A patent/TW201209062A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2580317C2 (ru) | 2016-04-10 |
| MX2012014576A (es) | 2013-02-21 |
| CA2796894A1 (en) | 2011-12-29 |
| EP2588126A4 (en) | 2015-07-08 |
| TW201209062A (en) | 2012-03-01 |
| WO2011163012A2 (en) | 2011-12-29 |
| US8778872B2 (en) | 2014-07-15 |
| EP2588126A2 (en) | 2013-05-08 |
| WO2011163012A3 (en) | 2013-07-11 |
| AR081471A1 (es) | 2012-09-05 |
| RU2013103093A (ru) | 2014-07-27 |
| US20130123462A1 (en) | 2013-05-16 |
| CN103179979A (zh) | 2013-06-26 |
| JP2013540102A (ja) | 2013-10-31 |
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