JP2011105738A5 - - Google Patents

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Publication number
JP2011105738A5
JP2011105738A5 JP2011010997A JP2011010997A JP2011105738A5 JP 2011105738 A5 JP2011105738 A5 JP 2011105738A5 JP 2011010997 A JP2011010997 A JP 2011010997A JP 2011010997 A JP2011010997 A JP 2011010997A JP 2011105738 A5 JP2011105738 A5 JP 2011105738A5
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JP
Japan
Prior art keywords
pharmaceutical composition
compound
pharmaceutically acceptable
acceptable salt
composition according
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JP2011010997A
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English (en)
Japanese (ja)
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JP2011105738A (ja
JP5400812B2 (ja
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Priority claimed from GBGB0412769.2A external-priority patent/GB0412769D0/en
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Publication of JP2011105738A publication Critical patent/JP2011105738A/ja
Publication of JP2011105738A5 publication Critical patent/JP2011105738A5/ja
Application granted granted Critical
Publication of JP5400812B2 publication Critical patent/JP5400812B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2011010997A 2004-06-08 2011-01-21 バニロイドアンタゴニストとして有用なキナゾリノン誘導体 Expired - Lifetime JP5400812B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0412769.2A GB0412769D0 (en) 2004-06-08 2004-06-08 Organic compounds
GB0412769.2 2004-06-08

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2007526311A Division JP4703650B2 (ja) 2004-06-08 2005-06-08 バニロイドアンタゴニストとして有用なキナゾリノン誘導体

Publications (3)

Publication Number Publication Date
JP2011105738A JP2011105738A (ja) 2011-06-02
JP2011105738A5 true JP2011105738A5 (enExample) 2012-03-08
JP5400812B2 JP5400812B2 (ja) 2014-01-29

Family

ID=32696854

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2007526311A Expired - Lifetime JP4703650B2 (ja) 2004-06-08 2005-06-08 バニロイドアンタゴニストとして有用なキナゾリノン誘導体
JP2011010997A Expired - Lifetime JP5400812B2 (ja) 2004-06-08 2011-01-21 バニロイドアンタゴニストとして有用なキナゾリノン誘導体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2007526311A Expired - Lifetime JP4703650B2 (ja) 2004-06-08 2005-06-08 バニロイドアンタゴニストとして有用なキナゾリノン誘導体

Country Status (29)

Country Link
US (4) US7960399B2 (enExample)
EP (1) EP1755606B2 (enExample)
JP (2) JP4703650B2 (enExample)
KR (2) KR101018607B1 (enExample)
CN (1) CN1956721B (enExample)
AT (1) ATE376833T1 (enExample)
AU (2) AU2005251476C1 (enExample)
BR (1) BRPI0511933B8 (enExample)
CA (1) CA2567821C (enExample)
CY (1) CY1107846T1 (enExample)
DE (1) DE602005003128T3 (enExample)
DK (1) DK1755606T4 (enExample)
EC (2) ECSP067067A (enExample)
ES (1) ES2293584T5 (enExample)
GB (1) GB0412769D0 (enExample)
HR (1) HRP20070577T4 (enExample)
IL (1) IL179532A (enExample)
MA (1) MA28685B1 (enExample)
MX (1) MXPA06014249A (enExample)
NO (1) NO338181B1 (enExample)
NZ (1) NZ551630A (enExample)
PL (1) PL1755606T5 (enExample)
PT (1) PT1755606E (enExample)
RU (2) RU2449995C2 (enExample)
SG (1) SG153811A1 (enExample)
SI (1) SI1755606T2 (enExample)
TN (1) TNSN06405A1 (enExample)
WO (1) WO2005120510A1 (enExample)
ZA (1) ZA200609634B (enExample)

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US8349852B2 (en) * 2009-01-13 2013-01-08 Novartis Ag Quinazolinone derivatives useful as vanilloid antagonists
AR080056A1 (es) 2010-02-01 2012-03-07 Novartis Ag Derivados de ciclohexil-amida como antagonistas de los receptores de crf
CN102762572A (zh) 2010-02-01 2012-10-31 诺瓦提斯公司 作为CRF-1受体拮抗剂的吡唑并[5,1b]*唑衍生物
JP5748777B2 (ja) 2010-02-02 2015-07-15 ノバルティス アーゲー Crf受容体アンタゴニストとしてのシクロヘキシルアミド誘導体
US8546416B2 (en) 2011-05-27 2013-10-01 Novartis Ag 3-spirocyclic piperidine derivatives as ghrelin receptor agonists
CA2867043A1 (en) 2012-05-03 2013-11-07 Novartis Ag L-malate salt of 2,7-diaza-spiro[4.5]dec-7-yle derivatives and crystalline forms thereof as ghrelin receptor agonists
JP2016510749A (ja) 2013-03-05 2016-04-11 ユニヴァーシティー オブ ノートル ダム デュ ラック キナゾリノン抗生物質
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FI3873903T3 (fi) 2018-10-31 2024-03-26 Gilead Sciences Inc Substituoituja 6-azabentsiimidatsoliyhdisteitä HPK1-inhibiittoreina
KR102658602B1 (ko) 2018-10-31 2024-04-19 길리애드 사이언시즈, 인코포레이티드 Hpk1 억제 활성을 갖는 치환된 6-아자벤즈이미다졸 화합물
AU2020222348B2 (en) * 2019-02-15 2023-03-16 Bausch + Lomb Ireland Limited Methods for treating ocular surface pain
JP6994061B2 (ja) 2019-02-15 2022-01-14 ノバルティス アーゲー 4-(7-ヒドロキシ-2-イソプロピル-4-オキソ-4h-キナゾリン-3-イル)-ベンゾニトリルの製剤
EP3924345A1 (en) 2019-02-15 2021-12-22 Novartis AG Crystalline forms of 4-(7-hydroxy-2-isopropyl-4-oxo-4h-quinazolin-3-yl)-benzonitrile and formulations thereof
TWI826690B (zh) 2019-05-23 2023-12-21 美商基利科學股份有限公司 經取代之烯吲哚酮化物及其用途
RU2755206C1 (ru) 2020-05-20 2021-09-14 Федеральное государственное бюджетное учреждение науки Тихоокеанский институт биоорганической химии им. Г.Б. Елякова Дальневосточного отделения Российской академии наук (ТИБОХ ДВО РАН) Средство пролонгированного анальгетического действия и лекарственный препарат на его основе
US12459902B2 (en) * 2020-08-06 2025-11-04 Bausch + Lomb Ireland Limited Crystalline forms of 4-(7-hydroxy-2-isopropyl-4-oxo-4H-quinazolin-3-yl)-benzonitrile and formulations thereof
US20230416207A1 (en) * 2020-11-17 2023-12-28 Crystal Pharmatech Co., Ltd. Crystalline forms of quinazolinone compound and process for preparing the same
UY39681A (es) 2021-03-26 2022-10-31 Novartis Ag Derivados de ciclobutilo 1,3–sustituidos y sus usos
AU2023346366A1 (en) 2022-09-21 2025-03-20 Bausch + Lomb Ireland Limited Crystalline polymorph forms of a trpv1 antagonist and formulations thereof
KR20250030194A (ko) 2023-08-24 2025-03-05 코웨이 주식회사 출수 장치

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