NO338181B1 - Kinazolinderivat og farmasøytisk sammensetning omfattende dette - Google Patents
Kinazolinderivat og farmasøytisk sammensetning omfattende dette Download PDFInfo
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- NO338181B1 NO338181B1 NO20070122A NO20070122A NO338181B1 NO 338181 B1 NO338181 B1 NO 338181B1 NO 20070122 A NO20070122 A NO 20070122A NO 20070122 A NO20070122 A NO 20070122A NO 338181 B1 NO338181 B1 NO 338181B1
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- compound
- pain
- formula
- inflammatory
- treatment
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Landscapes
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- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Cereal-Derived Products (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0412769.2A GB0412769D0 (en) | 2004-06-08 | 2004-06-08 | Organic compounds |
| PCT/EP2005/006253 WO2005120510A1 (en) | 2004-06-08 | 2005-06-08 | Quinazolinone derivatives useful as vanilloid antagonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20070122L NO20070122L (no) | 2007-03-01 |
| NO338181B1 true NO338181B1 (no) | 2016-08-01 |
Family
ID=32696854
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20070122A NO338181B1 (no) | 2004-06-08 | 2007-01-08 | Kinazolinderivat og farmasøytisk sammensetning omfattende dette |
Country Status (29)
| Country | Link |
|---|---|
| US (4) | US7960399B2 (enExample) |
| EP (1) | EP1755606B2 (enExample) |
| JP (2) | JP4703650B2 (enExample) |
| KR (2) | KR20100101017A (enExample) |
| CN (1) | CN1956721B (enExample) |
| AT (1) | ATE376833T1 (enExample) |
| AU (2) | AU2005251476C1 (enExample) |
| BR (1) | BRPI0511933B8 (enExample) |
| CA (1) | CA2567821C (enExample) |
| CY (1) | CY1107846T1 (enExample) |
| DE (1) | DE602005003128T3 (enExample) |
| DK (1) | DK1755606T4 (enExample) |
| EC (2) | ECSP067067A (enExample) |
| ES (1) | ES2293584T5 (enExample) |
| GB (1) | GB0412769D0 (enExample) |
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| RU (2) | RU2449995C2 (enExample) |
| SG (1) | SG153811A1 (enExample) |
| SI (1) | SI1755606T2 (enExample) |
| TN (1) | TNSN06405A1 (enExample) |
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| GB0412769D0 (en) | 2004-06-08 | 2004-07-07 | Novartis Ag | Organic compounds |
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| CA2668579A1 (en) * | 2006-11-06 | 2008-06-05 | Neurogen Corporation | Cis-cyclohexyl substituted pyrimidinone derivatives |
| WO2009010529A1 (en) | 2007-07-18 | 2009-01-22 | Novartis Ag | Synergistic combinations of vr-1 antagonists and cox-2 inhibitors |
| US8915362B2 (en) | 2008-10-08 | 2014-12-23 | Ultimed, Inc. | Sharps container |
| US8349852B2 (en) * | 2009-01-13 | 2013-01-08 | Novartis Ag | Quinazolinone derivatives useful as vanilloid antagonists |
| AR080055A1 (es) | 2010-02-01 | 2012-03-07 | Novartis Ag | Derivados de pirazolo-[5,1-b]-oxazol como antagonistas de los receptores de crf -1 |
| AR080056A1 (es) | 2010-02-01 | 2012-03-07 | Novartis Ag | Derivados de ciclohexil-amida como antagonistas de los receptores de crf |
| WO2011095450A1 (en) | 2010-02-02 | 2011-08-11 | Novartis Ag | Cyclohexyl amide derivatives as crf receptor antagonists |
| UY34094A (es) | 2011-05-27 | 2013-01-03 | Novartis Ag | Derivados de la piperidina 3-espirocíclica como agonistas de receptores de la ghrelina |
| EP2852591A1 (en) | 2012-05-03 | 2015-04-01 | Novartis AG | L-malate salt of 2, 7 - diaza - spiro [4.5]dec- 7 - yle derivatives and crystalline forms thereof as ghrelin receptor agonists |
| WO2014138302A1 (en) * | 2013-03-05 | 2014-09-12 | University Of Notre Dame | Quinazolinone antibiotics |
| US10016425B2 (en) | 2016-11-03 | 2018-07-10 | King Saud University | Anti-ulcerative colitis compound |
| JP7273172B2 (ja) | 2018-10-31 | 2023-05-12 | ギリアード サイエンシーズ， インコーポレイテッド | Ｈｐｋ１阻害活性を有する置換６－アザベンゾイミダゾール化合物 |
| BR112021008255A2 (pt) | 2018-10-31 | 2021-08-03 | Gilead Sciences, Inc. | compostos de 6-azabenzimidazol substituídos como inibidores de hpk1 |
| TWI878266B (zh) | 2019-02-15 | 2025-04-01 | 愛爾蘭商博士倫愛爾蘭有限公司 | 治療眼表痛之方法 |
| US20220162170A1 (en) * | 2019-02-15 | 2022-05-26 | Novartis Ag | Crystalline forms of 4-(7-hydroxy-2-isopropyl-4-oxo-4h-quinazolin-3-yl)-benzonitrile and formulations thereof |
| JP6994061B2 (ja) | 2019-02-15 | 2022-01-14 | ノバルティス アーゲー | ４－（７－ヒドロキシ－２－イソプロピル－４－オキソ－４ｈ－キナゾリン－３－イル）－ベンゾニトリルの製剤 |
| EP3972695A1 (en) | 2019-05-23 | 2022-03-30 | Gilead Sciences, Inc. | Substituted exo-methylene-oxindoles which are hpk1/map4k1 inhibitors |
| RU2755206C1 (ru) | 2020-05-20 | 2021-09-14 | Федеральное государственное бюджетное учреждение науки Тихоокеанский институт биоорганической химии им. Г.Б. Елякова Дальневосточного отделения Российской академии наук (ТИБОХ ДВО РАН) | Средство пролонгированного анальгетического действия и лекарственный препарат на его основе |
| WO2022029656A1 (en) | 2020-08-06 | 2022-02-10 | Novartis Ag | Crystalline forms of 4-(7-hydroxy-2-isopropyl-4-oxo-4h-quinazolin-3-yl)-benzonitrile and formulations thereof |
| CN116456986A (zh) * | 2020-11-17 | 2023-07-18 | 苏州晶云药物科技股份有限公司 | 一种喹唑啉酮衍生物的新晶型及其制备方法 |
| AR125196A1 (es) | 2021-03-26 | 2023-06-21 | Novartis Ag | Derivados de ciclobutilo 1,3-sustituidos y sus usos |
| CN120112515A (zh) | 2022-09-21 | 2025-06-06 | 博士伦爱尔兰有限公司 | Trpv1拮抗剂的结晶多晶型形式及其制剂 |
| KR20250030194A (ko) | 2023-08-24 | 2025-03-05 | 코웨이 주식회사 | 출수 장치 |
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2004
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2005
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- 2005-06-08 RU RU2010112450/04A patent/RU2449995C2/ru active
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- 2005-06-08 BR BRPI0511933A patent/BRPI0511933B8/pt active IP Right Grant
- 2005-06-08 DE DE602005003128T patent/DE602005003128T3/de not_active Expired - Lifetime
- 2005-06-08 SI SI200530141T patent/SI1755606T2/sl unknown
- 2005-06-08 RU RU2006146632/04A patent/RU2396261C2/ru active
- 2005-06-08 US US11/569,802 patent/US7960399B2/en not_active Expired - Lifetime
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- 2005-06-08 JP JP2007526311A patent/JP4703650B2/ja not_active Expired - Lifetime
- 2005-06-08 DK DK05750584.4T patent/DK1755606T4/da active
- 2005-06-08 WO PCT/EP2005/006253 patent/WO2005120510A1/en not_active Ceased
- 2005-06-08 PT PT05750584T patent/PT1755606E/pt unknown
- 2005-06-08 SG SG200903909-0A patent/SG153811A1/en unknown
- 2005-06-08 KR KR1020107019024A patent/KR20100101017A/ko not_active Ceased
- 2005-06-08 KR KR1020067025788A patent/KR101018607B1/ko not_active Expired - Lifetime
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- 2006-11-20 ZA ZA200609634A patent/ZA200609634B/xx unknown
- 2006-11-23 IL IL179532A patent/IL179532A/en active IP Right Grant
- 2006-12-07 EC EC2006007067A patent/ECSP067067A/es unknown
- 2006-12-07 TN TNP2006000405A patent/TNSN06405A1/en unknown
- 2006-12-28 MA MA29565A patent/MA28685B1/fr unknown
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