JP2011105738A5 - - Google Patents

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Publication number
JP2011105738A5
JP2011105738A5 JP2011010997A JP2011010997A JP2011105738A5 JP 2011105738 A5 JP2011105738 A5 JP 2011105738A5 JP 2011010997 A JP2011010997 A JP 2011010997A JP 2011010997 A JP2011010997 A JP 2011010997A JP 2011105738 A5 JP2011105738 A5 JP 2011105738A5
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Japan
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pharmaceutical composition
compound
pharmaceutically acceptable
acceptable salt
composition according
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JP2011010997A
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JP5400812B2 (ja
JP2011105738A (ja
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Priority claimed from GBGB0412769.2A external-priority patent/GB0412769D0/en
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Claims (6)

  1. 遊離型または薬学的に許容される塩形態の、
    Figure 2011105738
    Figure 2011105738
    Figure 2011105738
    から選択される化合物を薬学的担体または希釈剤と合わせて含む、医薬組成物。
  2. 遊離型または薬学的に許容される塩形態の、次式
    Figure 2011105738
    を有する化合物を含む、請求項1に記載の医薬組成物。
  3. 遊離型または薬学的に許容される塩形態の、次式
    Figure 2011105738
    を有する化合物を含む、請求項1に記載の医薬組成物。
  4. 遊離型または薬学的に許容される塩形態の、次式
    Figure 2011105738
    を有する化合物を含む、請求項1に記載の医薬組成物。
  5. 化合物が遊離型である、請求項1〜4のいずれかに記載の医薬組成物。
  6. 化合物が薬学的に許容される塩形態である、請求項1〜4のいずれかに記載の医薬組成物。
JP2011010997A 2004-06-08 2011-01-21 バニロイドアンタゴニストとして有用なキナゾリノン誘導体 Active JP5400812B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0412769.2A GB0412769D0 (en) 2004-06-08 2004-06-08 Organic compounds
GB0412769.2 2004-06-08

Related Parent Applications (1)

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JP2007526311A Division JP4703650B2 (ja) 2004-06-08 2005-06-08 バニロイドアンタゴニストとして有用なキナゾリノン誘導体

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JP2011105738A JP2011105738A (ja) 2011-06-02
JP2011105738A5 true JP2011105738A5 (ja) 2012-03-08
JP5400812B2 JP5400812B2 (ja) 2014-01-29

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JP2007526311A Active JP4703650B2 (ja) 2004-06-08 2005-06-08 バニロイドアンタゴニストとして有用なキナゾリノン誘導体
JP2011010997A Active JP5400812B2 (ja) 2004-06-08 2011-01-21 バニロイドアンタゴニストとして有用なキナゾリノン誘導体

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Country Status (30)

Country Link
US (4) US7960399B2 (ja)
EP (1) EP1755606B2 (ja)
JP (2) JP4703650B2 (ja)
KR (2) KR20100101017A (ja)
CN (1) CN1956721B (ja)
AT (1) ATE376833T1 (ja)
AU (2) AU2005251476C1 (ja)
BR (1) BRPI0511933B8 (ja)
CA (1) CA2567821C (ja)
CY (1) CY1107846T1 (ja)
DE (1) DE602005003128T3 (ja)
DK (1) DK1755606T4 (ja)
EC (2) ECSP067067A (ja)
ES (1) ES2293584T5 (ja)
GB (1) GB0412769D0 (ja)
HK (1) HK1105577A1 (ja)
HR (1) HRP20070577T4 (ja)
IL (1) IL179532A (ja)
MA (1) MA28685B1 (ja)
MX (1) MXPA06014249A (ja)
NO (1) NO338181B1 (ja)
NZ (1) NZ551630A (ja)
PL (1) PL1755606T5 (ja)
PT (1) PT1755606E (ja)
RU (2) RU2396261C2 (ja)
SG (1) SG153811A1 (ja)
SI (1) SI1755606T2 (ja)
TN (1) TNSN06405A1 (ja)
WO (1) WO2005120510A1 (ja)
ZA (1) ZA200609634B (ja)

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TWI721624B (zh) 2018-10-31 2021-03-11 美商基利科學股份有限公司 經取代之6-氮雜苯并咪唑化合物
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JP2022520410A (ja) 2019-02-15 2022-03-30 ノバルティス アーゲー 4-(7-ヒドロキシ-2-イソプロピル-4-オキソ-4h-キナゾリン-3-イル)-ベンゾニトリルの結晶形態及びその製剤
CN113453686A (zh) 2019-02-15 2021-09-28 诺华股份有限公司 治疗眼表痛的方法
TWI826690B (zh) 2019-05-23 2023-12-21 美商基利科學股份有限公司 經取代之烯吲哚酮化物及其用途
RU2755206C1 (ru) 2020-05-20 2021-09-14 Федеральное государственное бюджетное учреждение науки Тихоокеанский институт биоорганической химии им. Г.Б. Елякова Дальневосточного отделения Российской академии наук (ТИБОХ ДВО РАН) Средство пролонгированного анальгетического действия и лекарственный препарат на его основе
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