JP2013032389A5 - - Google Patents

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JP2013032389A5
JP2013032389A5 JP2012243691A JP2012243691A JP2013032389A5 JP 2013032389 A5 JP2013032389 A5 JP 2013032389A5 JP 2012243691 A JP2012243691 A JP 2012243691A JP 2012243691 A JP2012243691 A JP 2012243691A JP 2013032389 A5 JP2013032389 A5 JP 2013032389A5
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mixture
following structural
formula
structural formula
pharmaceutically acceptable
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JP2012243691A
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JP2013032389A (ja
JP5775505B2 (ja
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Claims (4)

  1. 下記構造式：
    Figure 2013032389
     で示される化合物および医薬上許容される担体を含む医薬組成物。
  2. 下記構造式：
    Figure 2013032389
     で示される立体異性体の混合物（ただし、該立体異性体の混合物はラセミ体ではない）。
  3. 下記構造式：
    Figure 2013032389
     で示される２つのジアステレオマーの混合物である、請求項２記載の立体異性体の混合物。
  4. 請求項２または３記載の混合物および医薬上許容される担体を含む医薬組成物。
JP2012243691A 2000-07-21 2012-11-05 Ｃ型肝炎ウイルスのｎｓ３−セリンプロテアーゼ阻害剤としての新規ペプチド Expired - Fee Related JP5775505B2 (ja)

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US22010800P 2000-07-21 2000-07-21
US60/220,108 2000-07-21

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JP2008275159A Division JP2009051860A (ja) 2000-07-21 2008-10-27 Ｃ型肝炎ウイルスのｎｓ３−セリンプロテアーゼ阻害剤としての新規ペプチド

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JP2013032389A JP2013032389A (ja) 2013-02-14
JP2013032389A5 true JP2013032389A5 (ja) 2013-03-28
JP5775505B2 JP5775505B2 (ja) 2015-09-09

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JP2002514149A Expired - Fee Related JP4298289B2 (ja) 2000-07-21 2001-07-19 Ｃ型肝炎ウイルスのｎｓ３−セリンプロテアーゼ阻害剤としての新規ペプチド
JP2008275159A Pending JP2009051860A (ja) 2000-07-21 2008-10-27 Ｃ型肝炎ウイルスのｎｓ３−セリンプロテアーゼ阻害剤としての新規ペプチド
JP2012243691A Expired - Fee Related JP5775505B2 (ja) 2000-07-21 2012-11-05 Ｃ型肝炎ウイルスのｎｓ３−セリンプロテアーゼ阻害剤としての新規ペプチド

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JP2002514149A Expired - Fee Related JP4298289B2 (ja) 2000-07-21 2001-07-19 Ｃ型肝炎ウイルスのｎｓ３−セリンプロテアーゼ阻害剤としての新規ペプチド
JP2008275159A Pending JP2009051860A (ja) 2000-07-21 2008-10-27 Ｃ型肝炎ウイルスのｎｓ３−セリンプロテアーゼ阻害剤としての新規ペプチド

Country Status (32)

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US (4) US7012066B2 (ja)
EP (1) EP1385870B1 (ja)
JP (3) JP4298289B2 (ja)
KR (2) KR100904788B1 (ja)
CN (3) CN1498224A (ja)
AR (2) AR033985A1 (ja)
AT (1) ATE461207T1 (ja)
AU (2) AU7698801A (ja)
BR (1) BR0112540A (ja)
CA (1) CA2410662C (ja)
CY (2) CY1112267T1 (ja)
CZ (1) CZ303213B6 (ja)
DE (2) DE60141608D1 (ja)
DK (1) DK1385870T3 (ja)
EC (1) ECSP034438A (ja)
ES (1) ES2341534T3 (ja)
HK (1) HK1058047A1 (ja)
HU (1) HU229997B1 (ja)
IL (2) IL153670A0 (ja)
LU (1) LU91910I2 (ja)
MX (1) MXPA03000627A (ja)
MY (2) MY139078A (ja)
NO (2) NO332329B1 (ja)
NZ (1) NZ523782A (ja)
PL (1) PL206255B1 (ja)
PT (1) PT1385870E (ja)
RU (2) RU2355700C9 (ja)
SI (1) SI1385870T1 (ja)
SK (1) SK288064B6 (ja)
TW (1) TWI324611B (ja)
WO (1) WO2002008244A2 (ja)
ZA (1) ZA200210312B (ja)

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