JP2013014622A5 - - Google Patents

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Publication number
JP2013014622A5
JP2013014622A5 JP2012230565A JP2012230565A JP2013014622A5 JP 2013014622 A5 JP2013014622 A5 JP 2013014622A5 JP 2012230565 A JP2012230565 A JP 2012230565A JP 2012230565 A JP2012230565 A JP 2012230565A JP 2013014622 A5 JP2013014622 A5 JP 2013014622A5
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JP
Japan
Prior art keywords
solvate
pharmaceutically acceptable
acceptable salt
compound
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012230565A
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English (en)
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JP2013014622A (ja
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Application filed filed Critical
Publication of JP2013014622A publication Critical patent/JP2013014622A/ja
Publication of JP2013014622A5 publication Critical patent/JP2013014622A5/ja
Pending legal-status Critical Current

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Claims (4)

  1. 化合物


    またはその薬学的に許容される塩もしくは溶媒和物。
  2. 化合物



    またはその薬学的に許容される塩もしくは溶媒和物。
  3. 請求項１または２に記載の化合物またはその薬学的に許容される塩もしくは溶媒和物を含む、薬学的組成物。
  4. 医薬の製造における、請求項１または２に記載の化合物またはその薬学的に許容される塩もしくは溶媒和物の使用。
JP2012230565A 2007-03-15 2012-10-18 グルカン合成酵素阻害剤として有用であるピリダジノン誘導体 Pending JP2013014622A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US91817107P 2007-03-15 2007-03-15
US60/918,171 2007-03-15

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2009553612A Division JP5147866B2 (ja) 2007-03-15 2008-03-12 グルカン合成酵素阻害剤として有用であるピリダジノン誘導体

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013259117A Division JP2014051529A (ja) 2007-03-15 2013-12-16 グルカン合成酵素阻害剤として有用であるピリダジノン誘導体

Publications (2)

Publication Number Publication Date
JP2013014622A JP2013014622A (ja) 2013-01-24
JP2013014622A5 true JP2013014622A5 (ja) 2014-02-06

Family

ID=39525788

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2009553612A Expired - Fee Related JP5147866B2 (ja) 2007-03-15 2008-03-12 グルカン合成酵素阻害剤として有用であるピリダジノン誘導体
JP2012230565A Pending JP2013014622A (ja) 2007-03-15 2012-10-18 グルカン合成酵素阻害剤として有用であるピリダジノン誘導体
JP2013259117A Pending JP2014051529A (ja) 2007-03-15 2013-12-16 グルカン合成酵素阻害剤として有用であるピリダジノン誘導体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2009553612A Expired - Fee Related JP5147866B2 (ja) 2007-03-15 2008-03-12 グルカン合成酵素阻害剤として有用であるピリダジノン誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2013259117A Pending JP2014051529A (ja) 2007-03-15 2013-12-16 グルカン合成酵素阻害剤として有用であるピリダジノン誘導体

Country Status (18)

Country Link
US (1) US8232274B2 (ja)
EP (2) EP2137179B1 (ja)
JP (3) JP5147866B2 (ja)
KR (1) KR20100049500A (ja)
CN (1) CN101730692A (ja)
AR (1) AR065721A1 (ja)
AU (1) AU2008227100B2 (ja)
BR (1) BRPI0809238A2 (ja)
CA (1) CA2680583A1 (ja)
CL (1) CL2008000725A1 (ja)
CO (1) CO6220966A2 (ja)
EC (1) ECSP099634A (ja)
IL (1) IL200906A0 (ja)
MX (1) MX2009009948A (ja)
PE (1) PE20081882A1 (ja)
RU (1) RU2009137946A (ja)
TW (1) TW200902516A (ja)
WO (1) WO2008115381A1 (ja)

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CA2697551C (en) * 2007-09-20 2013-03-12 Irm Llc Piperidine derivatives as modulators of gpr119 activity
JP5627574B2 (ja) 2008-06-03 2014-11-19 インターミューン， インコーポレイテッド 炎症性および線維性疾患を治療するための化合物および方法
US20100041663A1 (en) 2008-07-18 2010-02-18 Novartis Ag Organic Compounds as Smo Inhibitors
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FI20115234A0 (fi) 2011-03-08 2011-03-08 Biotie Therapies Corp Uusia pyridatsinoni- ja pyridoniyhdisteitä
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JO3115B1 (ar) 2011-08-22 2017-09-20 Takeda Pharmaceuticals Co مركبات بيريدازينون واستخدامها كمثبطات daao
US9212147B2 (en) 2011-11-15 2015-12-15 Takeda Pharmaceutical Company Limited Dihydroxy aromatic heterocyclic compound
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AU2013203000B9 (en) * 2012-08-10 2017-02-02 Lantheus Medical Imaging, Inc. Compositions, methods, and systems for the synthesis and use of imaging agents
CN103664795B (zh) * 2012-09-06 2017-10-03 华东理工大学 哒嗪酮类化合物及其用途
AR092742A1 (es) 2012-10-02 2015-04-29 Intermune Inc Piridinonas antifibroticas
US11224395B2 (en) 2012-10-05 2022-01-18 Koninklijke Philips N.V. Medical imaging system and method for providing an enhanced X-ray image
GB201222711D0 (en) 2012-12-17 2013-01-30 Takeda Pharmaceutical Novel compounds
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
WO2015031036A1 (en) * 2013-08-26 2015-03-05 Purdue Pharma L.P. Azaspiro[4.5] decane derivatives and use thereof
KR102373700B1 (ko) 2014-04-02 2022-03-11 인터뮨, 인크. 항섬유성 피리디논
TW201735792A (zh) 2016-03-07 2017-10-16 農業保鮮股份有限公司 使用苯并氧雜硼雜環戊烯化合物和防腐氣體作為作物的抗微生物劑之協同方法
NZ756854A (en) 2017-03-15 2022-02-25 Lunella Biotech Inc Mitoriboscins: mitochondrial-based therapeutics targeting cancer cells, bacteria, and pathogenic yeast
EP3606913B1 (en) 2017-04-03 2022-04-27 Syngenta Participations AG Microbiocidal oxadiazole derivatives
CN109912476A (zh) * 2019-03-27 2019-06-21 南通宝凯化工有限公司 一种异丙氨基磺酰氯的生产工艺
WO2020253862A1 (zh) * 2019-06-21 2020-12-24 上海翰森生物医药科技有限公司 含氮芳基磷氧化物类衍生物、其制备方法和应用
WO2021113625A1 (en) * 2019-12-06 2021-06-10 Plexxikon Inc. Compounds and methods for cd73 modulation and indications therefor
WO2021222353A1 (en) 2020-04-30 2021-11-04 Gilead Sciences, Inc. Macrocyclic inhibitors of peptidylarginine deiminases
WO2023204124A1 (ja) * 2022-04-20 2023-10-26 日本曹達株式会社 ピリダジノン化合物並びに農園芸用殺菌剤、殺線虫剤、および医療用・動物用抗真菌剤

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