JP2007501185A - Ｃ型肝炎を含むフラビウイルス関連疾患を治療するためのプリンヌクレオシド類似体 - Google Patents

Ｃ型肝炎を含むフラビウイルス関連疾患を治療するためのプリンヌクレオシド類似体 Download PDF

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JP2007501185A
JP2007501185A JP2006520940A JP2006520940A JP2007501185A JP 2007501185 A JP2007501185 A JP 2007501185A JP 2006520940 A JP2006520940 A JP 2006520940A JP 2006520940 A JP2006520940 A JP 2006520940A JP 2007501185 A JP2007501185 A JP 2007501185A
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alkyl
alkenyl
alkynyl
acyl
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ストラー，リチヤード
ゴスラン，ジル
ドユカーン，ダビツド
ルロワ，フレデリク
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イデニクス（ケイマン）リミテツド
サントル・ナシオナル・ドウ・ラ・ルシエルシユ・シアンテイフイク
リユニベルシテ・モンペリエ・ドウー
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    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
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    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
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    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
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    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
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    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
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    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/056—Triazole or tetrazole radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/23—Heterocyclic radicals containing two or more heterocyclic rings condensed among themselves or condensed with a common carbocyclic ring system, not provided for in groups C07H19/14 - C07H19/22

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JP2006520940A 2003-07-25 2004-07-26 Ｃ型肝炎を含むフラビウイルス関連疾患を治療するためのプリンヌクレオシド類似体 Pending JP2007501185A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US49021603P 2003-07-25 2003-07-25
PCT/IB2004/002703 WO2005009418A2 (en) 2003-07-25 2004-07-26 Purine nucleoside analogues for treating diseases caused by flaviviridae including hepatitis c

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JP2007501185A true JP2007501185A (ja) 2007-01-25
JP2007501185A5 JP2007501185A5 (https=) 2007-09-20

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US (3) US20050075309A1 (https=)
EP (1) EP1658302B1 (https=)
JP (1) JP2007501185A (https=)
KR (1) KR20060084845A (https=)
CN (1) CN1852915A (https=)
AT (1) ATE478886T1 (https=)
AU (1) AU2004258750A1 (https=)
BR (1) BRPI0412849A (https=)
CA (1) CA2533367C (https=)
DE (1) DE602004028841D1 (https=)
DK (1) DK1658302T3 (https=)
ES (1) ES2351603T3 (https=)
NO (1) NO20060914L (https=)
PL (1) PL1658302T3 (https=)
PT (1) PT1658302E (https=)
RU (1) RU2006105640A (https=)
WO (1) WO2005009418A2 (https=)

Cited By (1)

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JP2016138078A (ja) * 2015-01-29 2016-08-04 学校法人日本大学 ８−アザ−３，７−ジデアザアデニンヌクレオシド誘導体、８−アザ−３，７−ジデアザアデニンヌクレオチド誘導体及びポリヌクレオチド誘導体ならびにプローブ

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