JP2002500675A5 - - Google Patents

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Publication number
JP2002500675A5
JP2002500675A5 JP1999500965A JP50096599A JP2002500675A5 JP 2002500675 A5 JP2002500675 A5 JP 2002500675A5 JP 1999500965 A JP1999500965 A JP 1999500965A JP 50096599 A JP50096599 A JP 50096599A JP 2002500675 A5 JP2002500675 A5 JP 2002500675A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP1999500965A
Other languages
English (en)
Japanese (ja)
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JP2002500675A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1998/011000 external-priority patent/WO1998054157A1/en
Publication of JP2002500675A publication Critical patent/JP2002500675A/ja
Publication of JP2002500675A5 publication Critical patent/JP2002500675A5/ja
Ceased legal-status Critical Current

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JP50096599A 1997-05-28 1998-05-28 血小板由来成長因子及び/又はp56▲上lck▼チロシンキナーゼを阻害するキノリン及びキノキサリン化合物 Ceased JP2002500675A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US86445597A 1997-05-28 1997-05-28
US08/864,455 1997-05-28
US97261497A 1997-11-18 1997-11-18
US08/972,614 1997-11-18
PCT/US1998/011000 WO1998054157A1 (en) 1997-05-28 1998-05-28 QUINOLINE AND QUINOXALINE COMPOUNDS WHICH INHIBIT PLATELET-DERIVED GROWTH FACTOR AND/OR p561ck TYROSINE KINASES

Publications (2)

Publication Number Publication Date
JP2002500675A JP2002500675A (ja) 2002-01-08
JP2002500675A5 true JP2002500675A5 (https=) 2005-12-22

Family

ID=27127839

Family Applications (3)

Application Number Title Priority Date Filing Date
JP50098799A Ceased JP2002500676A (ja) 1997-05-28 1998-05-28 血小板由来成長因子及び/又はp56▲上lck▼チロシンキナーゼを阻害するキノリン及びキノキサリン化合物
JP50096599A Ceased JP2002500675A (ja) 1997-05-28 1998-05-28 血小板由来成長因子及び/又はp56▲上lck▼チロシンキナーゼを阻害するキノリン及びキノキサリン化合物
JP50096499A Ceased JP2002513417A (ja) 1997-05-28 1998-05-28 血小板由来成長因子及び/又はP56▲上lck▼チロシンキナーゼを阻害するキノリン及びキノキサリン化合物

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP50098799A Ceased JP2002500676A (ja) 1997-05-28 1998-05-28 血小板由来成長因子及び/又はp56▲上lck▼チロシンキナーゼを阻害するキノリン及びキノキサリン化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP50096499A Ceased JP2002513417A (ja) 1997-05-28 1998-05-28 血小板由来成長因子及び/又はP56▲上lck▼チロシンキナーゼを阻害するキノリン及びキノキサリン化合物

Country Status (25)

Country Link
EP (3) EP1001945B1 (https=)
JP (3) JP2002500676A (https=)
KR (2) KR100440756B1 (https=)
CN (3) CN1261353A (https=)
AP (3) AP1362A (https=)
AT (3) ATE493389T1 (https=)
AU (3) AU742739B2 (https=)
BG (3) BG64419B1 (https=)
BR (3) BR9809172A (https=)
CA (3) CA2291774A1 (https=)
CZ (3) CZ298521B6 (https=)
DE (3) DE69828607T2 (https=)
DK (1) DK0991628T3 (https=)
EA (4) EA008136B1 (https=)
ES (1) ES2235331T3 (https=)
HU (2) HUP0002084A3 (https=)
IL (3) IL133008A0 (https=)
NO (3) NO323720B1 (https=)
OA (3) OA11222A (https=)
PL (3) PL195552B1 (https=)
PT (1) PT991628E (https=)
SI (1) SI0991628T1 (https=)
SK (4) SK158199A3 (https=)
UA (1) UA57790C2 (https=)
WO (3) WO1998054157A1 (https=)

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US9126946B2 (en) 2008-10-28 2015-09-08 Arena Pharmaceuticals, Inc. Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)urea and crystalline forms related thereto
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RS58514B1 (sr) 2012-06-13 2019-04-30 Incyte Holdings Corp Supstituisana triciklična jedinjenja kao inhibitori fgfr
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JP6408569B2 (ja) 2013-10-17 2018-10-17 バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated Dna−pk阻害剤としての(s)−n−メチル−8−(1−((2’−メチル−[4,5’−ビピリミジン]−6−イル)アミノ)プロパン−2−イル)キノリン−4−カルボキサミドおよびその重水素化誘導体の共結晶
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TWI719960B (zh) 2015-02-10 2021-03-01 英商阿斯迪克治療公司 新穎組成物
TWI712601B (zh) 2015-02-20 2020-12-11 美商英塞特公司 作為fgfr抑制劑之雙環雜環
US9580423B2 (en) 2015-02-20 2017-02-28 Incyte Corporation Bicyclic heterocycles as FGFR4 inhibitors
MA41551A (fr) 2015-02-20 2017-12-26 Incyte Corp Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4
US10478494B2 (en) 2015-04-03 2019-11-19 Astex Therapeutics Ltd FGFR/PD-1 combination therapy for the treatment of cancer
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