IL57400A - (6r,7r)-7-((z)-2-(2-aminothiazol-4-yl-2(2-carboxyprop-2-oxyimino)acetamido)-3-(1-pyridiniummethyl)ceph-3-em-4-carboxylic acid and its derivatives,process for their preparation and pharmaceutical compositions comprising them - Google Patents

(6r,7r)-7-((z)-2-(2-aminothiazol-4-yl-2(2-carboxyprop-2-oxyimino)acetamido)-3-(1-pyridiniummethyl)ceph-3-em-4-carboxylic acid and its derivatives,process for their preparation and pharmaceutical compositions comprising them

Info

Publication number
IL57400A
IL57400A IL57400A IL5740079A IL57400A IL 57400 A IL57400 A IL 57400A IL 57400 A IL57400 A IL 57400A IL 5740079 A IL5740079 A IL 5740079A IL 57400 A IL57400 A IL 57400A
Authority
IL
Israel
Prior art keywords
pyridiniummethyl
carboxyprop
ceph
aminothiazol
oxyimino
Prior art date
Application number
IL57400A
Other languages
English (en)
Other versions
IL57400A0 (en
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Priority to IL59793A priority Critical patent/IL59793A/xx
Publication of IL57400A0 publication Critical patent/IL57400A0/xx
Publication of IL57400A publication Critical patent/IL57400A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
IL57400A 1978-05-26 1979-05-25 (6r,7r)-7-((z)-2-(2-aminothiazol-4-yl-2(2-carboxyprop-2-oxyimino)acetamido)-3-(1-pyridiniummethyl)ceph-3-em-4-carboxylic acid and its derivatives,process for their preparation and pharmaceutical compositions comprising them IL57400A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IL59793A IL59793A (en) 1978-05-26 1979-05-25 Derivatives of(6r,7r)-7-((z)-2-(2-aminothiazol-4-yl)-2-(carboxy-(lower alkyl or cycloalkyl)oxyimino)acetamido)-3-(1-pyridinium-methyl)ceph-3-em-4-carboxylate,process for their preparation and pharmaceutical compositions comprising them

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB2291378 1978-05-26
GB2291178 1978-05-26

Publications (2)

Publication Number Publication Date
IL57400A0 IL57400A0 (en) 1979-09-30
IL57400A true IL57400A (en) 1982-08-31

Family

ID=26256190

Family Applications (3)

Application Number Title Priority Date Filing Date
IL57400A IL57400A (en) 1978-05-26 1979-05-25 (6r,7r)-7-((z)-2-(2-aminothiazol-4-yl-2(2-carboxyprop-2-oxyimino)acetamido)-3-(1-pyridiniummethyl)ceph-3-em-4-carboxylic acid and its derivatives,process for their preparation and pharmaceutical compositions comprising them
IL59793A IL59793A (en) 1978-05-26 1979-05-25 Derivatives of(6r,7r)-7-((z)-2-(2-aminothiazol-4-yl)-2-(carboxy-(lower alkyl or cycloalkyl)oxyimino)acetamido)-3-(1-pyridinium-methyl)ceph-3-em-4-carboxylate,process for their preparation and pharmaceutical compositions comprising them
IL59793A IL59793A0 (en) 1978-05-26 1980-04-09 Cephalosporin antibiotics

Family Applications After (2)

Application Number Title Priority Date Filing Date
IL59793A IL59793A (en) 1978-05-26 1979-05-25 Derivatives of(6r,7r)-7-((z)-2-(2-aminothiazol-4-yl)-2-(carboxy-(lower alkyl or cycloalkyl)oxyimino)acetamido)-3-(1-pyridinium-methyl)ceph-3-em-4-carboxylate,process for their preparation and pharmaceutical compositions comprising them
IL59793A IL59793A0 (en) 1978-05-26 1980-04-09 Cephalosporin antibiotics

Country Status (27)

Country Link
US (2) US4258041A (de)
AR (2) AR228726A1 (de)
AT (1) AT370420B (de)
AU (1) AU524671B2 (de)
CA (1) CA1127633A (de)
CH (2) CH649556A5 (de)
DE (1) DE2921316C2 (de)
DK (1) DK157685C (de)
ES (2) ES480914A1 (de)
FI (2) FI67555C (de)
FR (2) FR2426695A1 (de)
HK (1) HK40183A (de)
IE (2) IE49172B1 (de)
IL (3) IL57400A (de)
IT (1) IT1116198B (de)
KE (1) KE3252A (de)
LU (1) LU81319A1 (de)
MY (1) MY8400017A (de)
NL (2) NL176855C (de)
NO (2) NO155347C (de)
NZ (2) NZ190558A (de)
PH (1) PH16961A (de)
PT (2) PT69670A (de)
SE (2) SE438507B (de)
SG (1) SG58382G (de)
SI (2) SI7911231A8 (de)
YU (2) YU41635B (de)

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ATA239281A (de) 1982-08-15
IE49172B1 (en) 1985-08-21
DE2921316A1 (de) 1979-12-06
US4258041A (en) 1981-03-24
YU223482A (en) 1983-04-30
AU4742279A (en) 1979-11-29
AT370420B (de) 1983-03-25
NL8001348A (nl) 1980-06-30
FI67705B (fi) 1985-01-31
SE438507B (sv) 1985-04-22
MY8400017A (en) 1984-12-31
NO155347B (no) 1966-12-08
SE8402887L (sv) 1984-05-28
SI7911231A8 (en) 1997-06-30
FI67555C (fi) 1985-04-10
NL7904122A (nl) 1979-11-28
FR2445835B1 (de) 1983-06-03
NO155347C (no) 1987-03-18
US4600772A (en) 1986-07-15
SE7904576L (sv) 1980-02-11
YU123179A (en) 1983-01-21
IL59793A (en) 1982-08-31
FR2426695A1 (fr) 1979-12-21
FI801609A (fi) 1980-05-19
NO850153L (no) 1979-11-27
SG58382G (en) 1983-09-02
IE802453L (en) 1979-11-26
DE2921316C2 (de) 1982-09-16
YU41635B (en) 1987-12-31
LU81319A1 (fr) 1979-09-11
NZ193326A (en) 1982-05-31
AR228726A1 (es) 1983-04-15
NZ190558A (en) 1982-05-31
CA1127633A (en) 1982-07-13
FI791678A (fi) 1979-11-27
HK40183A (en) 1983-10-21
CH646178A5 (de) 1984-11-15
PT69669A (en) 1979-06-01
FR2426695B1 (de) 1982-06-11
AU524671B2 (en) 1982-09-30
SI8212234A8 (en) 1997-06-30
NL176855C (nl) 1985-06-17
YU43097B (en) 1989-02-28
FI67705C (fi) 1985-05-10
DK157685B (da) 1990-02-05
AR229883A1 (es) 1983-12-30
IL59793A0 (en) 1980-06-30
CH649556A5 (de) 1985-05-31
IE49173B1 (en) 1985-08-21
KE3252A (en) 1983-01-28
IT1116198B (it) 1986-02-10
SE8402887D0 (sv) 1984-05-28
DK216779A (da) 1979-11-27
FI67555B (fi) 1984-12-31
NL176855B (nl) 1985-01-16
ES480915A1 (es) 1980-02-01
IL57400A0 (en) 1979-09-30
FR2445835A1 (fr) 1980-08-01
NO791731L (no) 1979-11-27
IE791025L (en) 1979-11-26
PH16961A (en) 1984-04-27
ES480914A1 (es) 1980-02-01
PT69670A (en) 1979-06-01
DK157685C (da) 1990-07-09

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