IL145922A0 - Di-aryl acid derivatives as ppar receptor ligands - Google Patents
Di-aryl acid derivatives as ppar receptor ligandsInfo
- Publication number
- IL145922A0 IL145922A0 IL14592200A IL14592200A IL145922A0 IL 145922 A0 IL145922 A0 IL 145922A0 IL 14592200 A IL14592200 A IL 14592200A IL 14592200 A IL14592200 A IL 14592200A IL 145922 A0 IL145922 A0 IL 145922A0
- Authority
- IL
- Israel
- Prior art keywords
- acid derivatives
- receptor ligands
- aryl acid
- ppar receptor
- ppar
- Prior art date
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- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- C07C233/02—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
- C07C233/11—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to carbon atoms of an unsaturated carbon skeleton containing six-membered aromatic rings
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- C07C235/32—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
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- C07C65/24—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups polycyclic
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- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
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- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US13145599P | 1999-04-28 | 1999-04-28 | |
PCT/US2000/011833 WO2000064888A1 (en) | 1999-04-28 | 2000-04-28 | Di-aryl acid derivatives as ppar receptor ligands |
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IL145922A0 true IL145922A0 (en) | 2002-07-25 |
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Application Number | Title | Priority Date | Filing Date |
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IL14592200A IL145922A0 (en) | 1999-04-28 | 2000-04-28 | Di-aryl acid derivatives as ppar receptor ligands |
IL145922A IL145922A (en) | 1999-04-28 | 2001-10-14 | History of diarylic acid as PPAR receptor ligands, pharmaceutical preparations containing them and their use in the preparation of drugs |
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IL145922A IL145922A (en) | 1999-04-28 | 2001-10-14 | History of diarylic acid as PPAR receptor ligands, pharmaceutical preparations containing them and their use in the preparation of drugs |
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US (2) | US6635655B1 (no) |
EP (1) | EP1177187B1 (no) |
JP (1) | JP4598278B2 (no) |
KR (1) | KR100709498B1 (no) |
CN (2) | CN1331862C (no) |
AT (1) | ATE368037T1 (no) |
AU (1) | AU781266B2 (no) |
BR (1) | BR0010605A (no) |
CA (1) | CA2370250C (no) |
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EE (1) | EE200100556A (no) |
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PL (1) | PL196957B1 (no) |
PT (1) | PT1177187E (no) |
RU (1) | RU2267484C2 (no) |
SK (1) | SK15532001A3 (no) |
WO (1) | WO2000064888A1 (no) |
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- 2000-04-28 YU YU72201A patent/YU72201A/sh unknown
- 2000-04-28 PT PT00928698T patent/PT1177187E/pt unknown
- 2000-04-28 MX MXPA01010880A patent/MXPA01010880A/es active IP Right Grant
- 2000-04-28 NZ NZ515086A patent/NZ515086A/en unknown
- 2000-04-28 AU AU46895/00A patent/AU781266B2/en not_active Ceased
- 2000-04-28 KR KR1020017013757A patent/KR100709498B1/ko not_active IP Right Cessation
- 2000-04-28 WO PCT/US2000/011833 patent/WO2000064888A1/en active IP Right Grant
- 2000-04-28 ES ES00928698T patent/ES2287016T3/es not_active Expired - Lifetime
- 2000-09-14 US US09/662,649 patent/US6635655B1/en not_active Ceased
-
2001
- 2001-10-14 IL IL145922A patent/IL145922A/en not_active IP Right Cessation
- 2001-10-18 NO NO20015075A patent/NO323643B1/no unknown
- 2001-10-24 ZA ZA200108798A patent/ZA200108798B/en unknown
- 2001-10-26 HR HR20010795A patent/HRP20010795A2/hr not_active Application Discontinuation
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2002
- 2002-09-26 HK HK02107034.1A patent/HK1045515B/zh not_active IP Right Cessation
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2005
- 2005-10-20 US US11/254,215 patent/USRE40558E1/en not_active Expired - Lifetime
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