IL126902A - Tetrahydrolipstatin containing compositions - Google Patents

Tetrahydrolipstatin containing compositions

Info

Publication number
IL126902A
IL126902A IL12690298A IL12690298A IL126902A IL 126902 A IL126902 A IL 126902A IL 12690298 A IL12690298 A IL 12690298A IL 12690298 A IL12690298 A IL 12690298A IL 126902 A IL126902 A IL 126902A
Authority
IL
Israel
Prior art keywords
weight
composition
pellets
polyvinylpyrrolidone
tetrahydrolipstatin
Prior art date
Application number
IL12690298A
Other languages
English (en)
Other versions
IL126902A0 (en
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26671373&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL126902(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of IL126902A0 publication Critical patent/IL126902A0/xx
Publication of IL126902A publication Critical patent/IL126902A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Organic Chemistry (AREA)
  • Zoology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Biophysics (AREA)
  • Child & Adolescent Psychology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL12690298A 1997-02-05 1998-01-24 Tetrahydrolipstatin containing compositions IL126902A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US3738497P 1997-02-05 1997-02-05
US09/003,137 US6004996A (en) 1997-02-05 1998-01-06 Tetrahydrolipstatin containing compositions
PCT/EP1998/000395 WO1998034607A1 (en) 1997-02-05 1998-01-24 Tetrahydrolipstatin containing compositions

Publications (2)

Publication Number Publication Date
IL126902A0 IL126902A0 (en) 1999-09-22
IL126902A true IL126902A (en) 2002-12-01

Family

ID=26671373

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12690298A IL126902A (en) 1997-02-05 1998-01-24 Tetrahydrolipstatin containing compositions

Country Status (30)

Country Link
US (1) US6004996A (es)
EP (1) EP0921796B1 (es)
CN (1) CN1193752C (es)
AR (1) AR010704A1 (es)
AT (1) ATE200027T1 (es)
AU (1) AU713192B2 (es)
CA (1) CA2258095C (es)
CO (1) CO4920214A1 (es)
CY (1) CY2264B1 (es)
CZ (1) CZ287154B6 (es)
DE (1) DE69800639T2 (es)
DK (1) DK0921796T3 (es)
ES (1) ES2156028T3 (es)
GR (1) GR3036064T3 (es)
HK (1) HK1021313A1 (es)
HR (1) HRP980057B1 (es)
HU (1) HU225035B1 (es)
ID (1) ID26509A (es)
IL (1) IL126902A (es)
MA (1) MA24466A1 (es)
MY (1) MY118371A (es)
NO (1) NO320445B1 (es)
NZ (1) NZ332659A (es)
PE (1) PE57599A1 (es)
PT (1) PT921796E (es)
RU (1) RU2170579C2 (es)
SI (1) SI0921796T1 (es)
UY (1) UY24875A1 (es)
WO (1) WO1998034607A1 (es)
YU (1) YU49423B (es)

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Also Published As

Publication number Publication date
ID26509A (id) 2001-01-11
HUP0001468A2 (hu) 2000-09-28
ES2156028T3 (es) 2001-06-01
IL126902A0 (en) 1999-09-22
US6004996A (en) 1999-12-21
NO985337D0 (no) 1998-11-16
UY24875A1 (es) 2000-12-29
CY2264B1 (en) 2003-07-04
HRP980057B1 (en) 2001-08-31
DE69800639D1 (de) 2001-05-03
NO320445B1 (no) 2005-12-05
HU225035B1 (en) 2006-05-29
HRP980057A2 (en) 1998-12-31
PL330972A1 (en) 1999-06-21
RU2170579C2 (ru) 2001-07-20
CN1220600A (zh) 1999-06-23
HUP0001468A3 (en) 2000-12-28
EP0921796B1 (en) 2001-03-28
CZ287154B6 (en) 2000-09-13
HU0001468D0 (en) 2000-05-28
AU713192B2 (en) 1999-11-25
CA2258095C (en) 2000-02-22
YU49423B (sh) 2006-01-16
YU49698A (sh) 1999-09-27
CO4920214A1 (es) 2000-05-29
DK0921796T3 (da) 2001-07-16
CA2258095A1 (en) 1998-08-13
PT921796E (pt) 2001-09-28
CN1193752C (zh) 2005-03-23
NZ332659A (en) 2000-03-27
NO985337L (no) 1998-11-16
DE69800639T2 (de) 2001-10-31
GR3036064T3 (en) 2001-09-28
MA24466A1 (fr) 1998-10-01
CZ352898A3 (cs) 1999-02-17
WO1998034607A1 (en) 1998-08-13
EP0921796A1 (en) 1999-06-16
MY118371A (en) 2004-10-30
AR010704A1 (es) 2000-06-28
HK1021313A1 (en) 2000-06-09
AU6097298A (en) 1998-08-26
SI0921796T1 (en) 2001-06-30
PE57599A1 (es) 1999-06-11
ATE200027T1 (de) 2001-04-15

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