HUE028987T2 - BI-aryl-meta-pyrimidine inhibitors of kinases - Google Patents

BI-aryl-meta-pyrimidine inhibitors of kinases Download PDF

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Publication number
HUE028987T2
HUE028987T2 HUE06836583A HUE06836583A HUE028987T2 HU E028987 T2 HUE028987 T2 HU E028987T2 HU E06836583 A HUE06836583 A HU E06836583A HU E06836583 A HUE06836583 A HU E06836583A HU E028987 T2 HUE028987 T2 HU E028987T2
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Hungary
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mmol
mixture
filtered
methyl
concentrated
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HUE06836583A
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English (en)
Hungarian (hu)
Inventor
Jianguo Cao
John Hood
Daniel Lohse
Chi Ching Mak
Pherson Andrew Mc
Glenn Noronha
Ved PATHAK
Joel Renick
Richard M Soll
Binqi Zeng
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Targegen Inc
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Publication of HUE028987T2 publication Critical patent/HUE028987T2/en

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    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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HUE06836583A 2005-11-01 2006-10-26 BI-aryl-meta-pyrimidine inhibitors of kinases HUE028987T2 (en)

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US73262905P 2005-11-01 2005-11-01
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