HK1100004A1 - Synthesis of boronic ester and acid compounds - Google Patents

Synthesis of boronic ester and acid compounds

Info

Publication number
HK1100004A1
HK1100004A1 HK07107789.3A HK07107789A HK1100004A1 HK 1100004 A1 HK1100004 A1 HK 1100004A1 HK 07107789 A HK07107789 A HK 07107789A HK 1100004 A1 HK1100004 A1 HK 1100004A1
Authority
HK
Hong Kong
Prior art keywords
synthesis
acid compounds
boronic ester
boronic
ester
Prior art date
Application number
HK07107789.3A
Other languages
English (en)
Inventor
Pickersgill I Fraser
Bishop John
Koellner Christoph
Gomez Jean-Marc
Geiser Achim
Hett Robert
Ammoscato Vince
Munk Stephen
Lo Young
Chui Fang-Ting
V R Kulkarni
Original Assignee
Millennium Pharmaceuticalsinc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34968044&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1100004(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Millennium Pharmaceuticalsinc filed Critical Millennium Pharmaceuticalsinc
Publication of HK1100004A1 publication Critical patent/HK1100004A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/04—Esters of boric acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Virology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Transplantation (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
HK07107789.3A 2004-03-30 2007-07-19 Synthesis of boronic ester and acid compounds HK1100004A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55753504P 2004-03-30 2004-03-30
PCT/US2005/009774 WO2005097809A2 (fr) 2004-03-30 2005-03-24 Synthese d'ester borique et de composes acides

Publications (1)

Publication Number Publication Date
HK1100004A1 true HK1100004A1 (en) 2007-08-31

Family

ID=34968044

Family Applications (4)

Application Number Title Priority Date Filing Date
HK07107789.3A HK1100004A1 (en) 2004-03-30 2007-07-19 Synthesis of boronic ester and acid compounds
HK12103590.4A HK1164320A1 (en) 2004-03-30 2012-04-12 Synthesis of bortezomib
HK18105728.8A HK1246300A1 (zh) 2004-03-30 2018-05-03 硼的酯和酸化合物的合成
HK18116447.5A HK1257298A1 (zh) 2004-03-30 2018-12-21 硼的酯和酸化合物的合成

Family Applications After (3)

Application Number Title Priority Date Filing Date
HK12103590.4A HK1164320A1 (en) 2004-03-30 2012-04-12 Synthesis of bortezomib
HK18105728.8A HK1246300A1 (zh) 2004-03-30 2018-05-03 硼的酯和酸化合物的合成
HK18116447.5A HK1257298A1 (zh) 2004-03-30 2018-12-21 硼的酯和酸化合物的合成

Country Status (41)

Country Link
US (14) US7714159B2 (fr)
EP (5) EP2377868A1 (fr)
JP (4) JP4558039B2 (fr)
KR (1) KR100939598B1 (fr)
CN (5) CN107474062A (fr)
AR (3) AR049374A1 (fr)
AT (1) ATE521612T1 (fr)
AU (1) AU2005230930B2 (fr)
BR (1) BRPI0509587A (fr)
CA (4) CA2560886C (fr)
CL (2) CL2010000350A1 (fr)
CR (1) CR8653A (fr)
CY (3) CY1112053T1 (fr)
DK (4) DK4008721T3 (fr)
DO (1) DOP2011000293A (fr)
EA (1) EA012927B1 (fr)
EC (1) ECSP066960A (fr)
ES (4) ES2371652T3 (fr)
FI (1) FI4008721T3 (fr)
HK (4) HK1100004A1 (fr)
HR (4) HRP20240307T3 (fr)
HU (1) HUE056859T2 (fr)
IL (3) IL178250A (fr)
LT (2) LT3385267T (fr)
ME (1) ME01975B (fr)
MX (1) MX367324B (fr)
MY (1) MY145427A (fr)
NL (3) NL1028639C2 (fr)
NO (4) NO338905B1 (fr)
NZ (3) NZ586824A (fr)
PE (3) PE20060162A1 (fr)
PL (4) PL1756121T3 (fr)
PT (4) PT1756121E (fr)
RS (4) RS62738B1 (fr)
SG (5) SG182998A1 (fr)
SI (4) SI2377869T1 (fr)
TW (1) TWI386212B (fr)
UA (1) UA90108C2 (fr)
UY (3) UY28830A1 (fr)
WO (1) WO2005097809A2 (fr)
ZA (1) ZA200608689B (fr)

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AU2016253697A1 (en) * 2007-08-06 2016-11-24 Millennium Pharmaceuticals, Inc. Proteasome inhibitors
US7442830B1 (en) 2007-08-06 2008-10-28 Millenium Pharmaceuticals, Inc. Proteasome inhibitors
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EA034601B1 (ru) * 2007-08-06 2020-02-25 Милленниум Фармасьютикалз, Инк. Способ получения бороновых кислот
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Also Published As

Publication number Publication date
EP2377869A1 (fr) 2011-10-19
NO20191065A1 (no) 2006-12-22
US20200157143A1 (en) 2020-05-21
US20220204558A1 (en) 2022-06-30
MY145427A (en) 2012-02-15
EP2377869B1 (fr) 2014-01-29
HRP20240307T3 (hr) 2024-05-10
PT4008721T (pt) 2024-03-21
PT1756121E (pt) 2011-11-30
SI3385267T1 (sl) 2022-04-29
ES2371652T3 (es) 2012-01-05
LT3385267T (lt) 2021-11-10
NZ598172A (en) 2013-08-30
CN107474062A (zh) 2017-12-15
NL1028639C2 (nl) 2007-01-17
RS51983B (en) 2012-02-29
US20130005968A1 (en) 2013-01-03
US20210395301A1 (en) 2021-12-23
IL178250A0 (en) 2006-12-31
US20050240047A1 (en) 2005-10-27
WO2005097809A3 (fr) 2006-02-16
NZ550522A (en) 2010-08-27
ATE521612T1 (de) 2011-09-15
CA2738706C (fr) 2014-10-14
CN108329337B (zh) 2021-06-25
NO338905B1 (no) 2016-10-31
JP4558039B2 (ja) 2010-10-06
KR100939598B1 (ko) 2010-02-01
ES2974758T3 (es) 2024-07-01
US20190112334A1 (en) 2019-04-18
HK1257298A1 (zh) 2019-10-18
EP4008721A1 (fr) 2022-06-08
US10000529B2 (en) 2018-06-19
ZA200608689B (en) 2007-09-26
AU2005230930A1 (en) 2005-10-20
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