GT201100056AA - Metodo para preparar compuestos macrocíclicos inhibidores de serina proteasas de hepatitis c (solicitud fraccionaria de la solicitud de patente de invencion no. a-2011-00056) - Google Patents

Metodo para preparar compuestos macrocíclicos inhibidores de serina proteasas de hepatitis c (solicitud fraccionaria de la solicitud de patente de invencion no. a-2011-00056)

Info

Publication number
GT201100056AA
GT201100056AA GT201100056AK GT201100056K GT201100056AA GT 201100056A A GT201100056A A GT 201100056AA GT 201100056A K GT201100056A K GT 201100056AK GT 201100056 K GT201100056 K GT 201100056K GT 201100056A A GT201100056A A GT 201100056AA
Authority
GT
Guatemala
Prior art keywords
application
hepatitis
fractionary
invention patent
serine proteases
Prior art date
Application number
GT201100056AK
Other languages
English (en)
Spanish (es)
Inventor
Yiyin Ku
Keith F Mcdaniel
Hui-Ju Chen
Jason P Shanley
Dale J Kempf
David J Grampovnik
Ying Sun
Dong Liu
Yonghua Gai
Sun Yay Or
Sable H Wagaw
Ken Engstrom
Tim Grieme
Ahmad Sheik
Jianzhang Mei
Original Assignee
Enanta Pharm Inc
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42005677&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT201100056A(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Enanta Pharm Inc, Abbott Lab filed Critical Enanta Pharm Inc
Publication of GT201100056AA publication Critical patent/GT201100056AA/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C07K1/113—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides without change of the primary structure
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Analytical Chemistry (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
GT201100056AK 2008-09-11 2011-03-28 Metodo para preparar compuestos macrocíclicos inhibidores de serina proteasas de hepatitis c (solicitud fraccionaria de la solicitud de patente de invencion no. a-2011-00056) GT201100056AA (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US19172508P 2008-09-11 2008-09-11
US20968909P 2009-03-10 2009-03-10

Publications (1)

Publication Number Publication Date
GT201100056AA true GT201100056AA (es) 2014-09-26

Family

ID=42005677

Family Applications (2)

Application Number Title Priority Date Filing Date
GT201100056AK GT201100056AA (es) 2008-09-11 2011-03-28 Metodo para preparar compuestos macrocíclicos inhibidores de serina proteasas de hepatitis c (solicitud fraccionaria de la solicitud de patente de invencion no. a-2011-00056)
GT201100056BA GT201100056BA (es) 2008-09-11 2013-12-10 Inhibidores macrocíclicos de serina proteasas de hepatitis c (segunda solicitud fraccionaria de la solicitud de patentes de invención no. a-2011-00056).

Family Applications After (1)

Application Number Title Priority Date Filing Date
GT201100056BA GT201100056BA (es) 2008-09-11 2013-12-10 Inhibidores macrocíclicos de serina proteasas de hepatitis c (segunda solicitud fraccionaria de la solicitud de patentes de invención no. a-2011-00056).

Country Status (41)

Country Link
US (3) US8420596B2 (xx)
EP (5) EP2805726B1 (xx)
JP (4) JP5259537B2 (xx)
KR (3) KR101379365B1 (xx)
CN (3) CN103896950A (xx)
AR (3) AR073568A1 (xx)
AU (1) AU2009292182B2 (xx)
BR (2) BR122012005261A8 (xx)
CA (1) CA2736895C (xx)
CL (2) CL2011000512A1 (xx)
CO (1) CO6341565A2 (xx)
CR (1) CR20140180A (xx)
CY (6) CY1115137T1 (xx)
DK (5) DK2468286T3 (xx)
DO (1) DOP2011000077A (xx)
EA (2) EA020580B1 (xx)
EC (2) ECSP11010879A (xx)
ES (5) ES2459390T3 (xx)
GT (2) GT201100056AA (xx)
HK (4) HK1159515A1 (xx)
HR (5) HRP20140494T1 (xx)
HU (2) HUE039478T2 (xx)
IL (2) IL218441A (xx)
LT (2) LT2805726T (xx)
LU (1) LU92667I2 (xx)
MX (1) MX2011002486A (xx)
MY (1) MY159820A (xx)
NL (1) NL300730I1 (xx)
NO (1) NO2015014I1 (xx)
NZ (2) NZ592170A (xx)
PA (1) PA8842201A1 (xx)
PE (3) PE20110704A1 (xx)
PL (5) PL2805726T3 (xx)
PT (5) PT2805726T (xx)
SG (1) SG179414A1 (xx)
SI (5) SI2805726T1 (xx)
TR (1) TR201809771T4 (xx)
TW (3) TWI450723B (xx)
UY (3) UY32099A (xx)
WO (1) WO2010030359A2 (xx)
ZA (2) ZA201101558B (xx)

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