FR05C0045I1 - - Google Patents

Info

Publication number
FR05C0045I1
FR05C0045I1 FR05C0045C FR05C0045I1 FR 05C0045 I1 FR05C0045 I1 FR 05C0045I1 FR 05C0045 C FR05C0045 C FR 05C0045C FR 05C0045 I1 FR05C0045 I1 FR 05C0045I1
Authority
FR
France
Prior art keywords
pct
date sep
sec
pub
antiobiotic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
Other languages
English (en)
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of FR05C0045I1 publication Critical patent/FR05C0045I1/fr
Application granted granted Critical
Publication of FR05C0045I2 publication Critical patent/FR05C0045I2/fr
Active legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
FR05C0045C 1993-03-12 2005-11-17 Active FR05C0045I2 (enExample)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3329193A 1993-03-12 1993-03-12
PCT/US1994/001862 WO1994020505A1 (en) 1993-03-12 1994-03-07 Crystalline ceftiofur free acid

Publications (2)

Publication Number Publication Date
FR05C0045I1 true FR05C0045I1 (enExample) 2006-01-06
FR05C0045I2 FR05C0045I2 (enExample) 2007-08-03

Family

ID=21869579

Family Applications (1)

Application Number Title Priority Date Filing Date
FR05C0045C Active FR05C0045I2 (enExample) 1993-03-12 2005-11-17

Country Status (31)

Country Link
US (1) US5721359A (enExample)
EP (1) EP0690864B1 (enExample)
JP (1) JP3852946B2 (enExample)
KR (1) KR100296810B1 (enExample)
CN (1) CN1055090C (enExample)
AT (1) ATE202109T1 (enExample)
AU (1) AU694419B2 (enExample)
BR (1) BR1101034A (enExample)
CA (1) CA2155322C (enExample)
CZ (1) CZ289332B6 (enExample)
DE (2) DE122005000055I2 (enExample)
DK (1) DK0690864T3 (enExample)
ES (1) ES2157254T3 (enExample)
FI (1) FI120307B (enExample)
FR (1) FR05C0045I2 (enExample)
GR (1) GR3036514T3 (enExample)
HU (1) HU222244B1 (enExample)
IL (1) IL108910A (enExample)
LU (1) LU91206I2 (enExample)
LV (1) LV12889B (enExample)
NL (1) NL300208I2 (enExample)
NO (2) NO313199B1 (enExample)
NZ (1) NZ263002A (enExample)
PL (1) PL184611B1 (enExample)
PT (1) PT690864E (enExample)
RU (1) RU2136685C1 (enExample)
SI (1) SI0690864T1 (enExample)
SK (1) SK283674B6 (enExample)
TW (1) TW267170B (enExample)
WO (1) WO1994020505A1 (enExample)
ZA (1) ZA941586B (enExample)

Families Citing this family (73)

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US6074657A (en) * 1997-03-20 2000-06-13 Pharmacia & Upjohn Company Administration of an injectable antibiotic in the ear of an animal
AU2001288323B2 (en) * 2000-09-12 2006-11-23 Zoetis Services Llc Pharmaceutical composition having modified carrier
US7829100B2 (en) * 2000-09-12 2010-11-09 Teagarden Dirk L Pharmaceutical composition having modified carrier
KR100423895B1 (ko) * 2001-02-19 2004-03-24 주식회사 엘지생명과학 셉티오퍼 하이드로클로라이드의 현탁제 조성물
JP2005502628A (ja) * 2001-07-10 2005-01-27 ファルマシア・アンド・アップジョン・カンパニー 結晶性チアジンオキサゾリジノン
CZ2004196A3 (cs) 2001-08-15 2005-01-12 Pharmacia & Upjohn Company Krystaly obsahující sůl N-[2-(diethylamino)ethyl]-5-[(5-fluor-2-oxo-3H-indol-3-yliden) methyl]-2,4-dimethyl-1H-pyrrol 3-karboxamidu s kyselinou jablečnou, způsob jejich výroby a kompozice na jejich bázi
CN1635856A (zh) 2002-03-21 2005-07-06 法玛西雅厄普约翰有限责任公司 向动物耳施用可注射抗生物的方法
US20040022815A1 (en) * 2002-08-05 2004-02-05 Orchid Health Care Novel pharmaceutical composition of ceftiofur
KR20040015622A (ko) * 2002-08-13 2004-02-19 대한뉴팜(주) 세프티오푸르나트륨을 활성성분으로 함유하는 현탁주사액조성물
US20040115822A1 (en) * 2002-09-12 2004-06-17 Schapaugh Randal Lee Methods of measuring the dissolution rate of an analyte in a non-aqueous liquid composition
US7659061B2 (en) * 2002-11-19 2010-02-09 Pharmacia & Upjohn Company Pharmaceutical compositions having a modified vehicle
US20040115837A1 (en) * 2002-11-27 2004-06-17 Schapaugh Randal Lee Methods of measuring the dissolution rate of an analyte in a non-aqueous liquid composition
US7842791B2 (en) * 2002-12-19 2010-11-30 Nancy Jean Britten Dispersible pharmaceutical compositions
PT1606293E (pt) * 2003-03-27 2009-10-14 Basilea Pharmaceutica Ag Cefalosporina sob forma cristalina
PL2156824T3 (pl) 2004-03-25 2013-03-29 Astellas Pharma Inc Kompozycja solifenacyny lub jej soli do zastosowania w formulacji stałej
US7815939B2 (en) 2005-07-20 2010-10-19 Astellas Pharma Inc. Coated fine particles containing drug for intrabuccally fast disintegrating dosage forms
US8470809B2 (en) * 2005-10-12 2013-06-25 Orchid Chemicals & Pharmaceuticals Limited Crystalline sodium salt of cephalosporin antibiotic
WO2007042917A1 (en) * 2005-10-12 2007-04-19 Orchid Chemicals And Pharmaceuticals Limited Crystalline sodium salt of cephalosporin antibiotic
UA101809C2 (uk) 2007-08-22 2013-05-13 Астразенека Аб Похідні циклопропіламіду
US9943614B2 (en) 2008-06-17 2018-04-17 Brigham Young University Cationic steroid antimicrobial diagnostic, detection, screening and imaging methods
WO2010020871A2 (en) * 2008-08-22 2010-02-25 Orchid Chemicals & Pharmaceuticals Limited Crystalline sodium salt of cephalosporin antibiotic
MX2011005217A (es) * 2008-11-19 2011-06-01 Merial Ltd Formulaciones que comprenden ceftiofur y cetoprofeno o ceftiofur y alcohol bencilico.
MY161598A (en) * 2009-01-30 2017-04-28 Glaxosmithkline Llc Crystalline n-{ (1s)-2-amino-1-[(3-fluorophenyl)methyl]ethyl} -5-chloro-4-(4-chloro-1-methyl-1h-pyrazol-5-yl)-2-thiophenecarboxamide hydrochloride
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
AR080203A1 (es) * 2010-02-18 2012-03-21 Astrazeneca Ab Formas solidas que comprenden una ciclopropilamida
KR20130002316A (ko) * 2010-02-18 2013-01-07 아스트라제네카 아베 시클로프로필 벤즈아미드 유도체의 신규 결정질 형태
JP2014513116A (ja) * 2011-05-02 2014-05-29 ゾエティス・エルエルシー 抗菌剤として有用な新規セファロスポリン
CA2842462C (en) 2011-07-20 2020-01-28 Brigham Young University Hydrogel materials incorporating eluting ceragenin compound
US9603859B2 (en) 2011-09-13 2017-03-28 Brigham Young University Methods and products for increasing the rate of healing of tissue wounds
EP2755661A1 (en) 2011-09-13 2014-07-23 Brigham Young University Compositions for treating bone diseases and broken bones
MX369385B (es) 2011-09-13 2019-11-07 Univ Brigham Young Productos para cicatrizar heridas tisulares.
US9694019B2 (en) 2011-09-13 2017-07-04 Brigham Young University Compositions and methods for treating bone diseases and broken bones
JP6051230B2 (ja) 2011-12-21 2016-12-27 ブリガム ヤング ユニバーシティ 口腔ケア組成物
CN102584855B (zh) * 2012-02-16 2014-06-25 青岛科技大学 一种改进的头孢噻呋的制备方法
US9533063B1 (en) 2012-03-01 2017-01-03 Brigham Young University Aerosols incorporating ceragenin compounds and methods of use thereof
EP3225113B1 (en) 2012-05-02 2020-09-02 Brigham Young University Methods for making ceragenin particulate materials
US9314472B2 (en) 2012-10-17 2016-04-19 Brigham Young University Treatment and prevention of mastitis
JP6310396B2 (ja) * 2012-12-03 2018-04-11 株式会社カネカ 還元型補酵素q10誘導体およびその製造方法
AU2014203882B2 (en) 2013-01-07 2016-06-23 Brigham Young University Methods for reducing cellular proliferation and treating certain diseases
US11524015B2 (en) 2013-03-15 2022-12-13 Brigham Young University Methods for treating inflammation, autoimmune disorders and pain
US10568893B2 (en) 2013-03-15 2020-02-25 Brigham Young University Methods for treating inflammation, autoimmune disorders and pain
RU2669800C2 (ru) 2013-03-15 2018-10-16 Брихэм Янг Юниверсити Способы лечения воспаления, аутоиммунных расстройств и боли
RU2546675C2 (ru) * 2013-04-11 2015-04-10 Федеральное казённое предприятие "Государственный научно-исследовательский институт химических продуктов" (ФКП "ГосНИИХП") Способ определения степени кристалличности составов на основе дифениламина
US9387215B2 (en) 2013-04-22 2016-07-12 Brigham Young University Animal feed including cationic cholesterol additive and related methods
KR102177643B1 (ko) * 2013-09-05 2020-11-11 미쓰비시 타나베 파마 코퍼레이션 신규한 결정성 아릴알킬아민 화합물 및 그의 제조 방법
US11690855B2 (en) 2013-10-17 2023-07-04 Brigham Young University Methods for treating lung infections and inflammation
US20150203527A1 (en) 2014-01-23 2015-07-23 Brigham Young University Cationic steroidal antimicrobials
CA2844321C (en) 2014-02-27 2021-03-16 Brigham Young University Cationic steroidal antimicrobial compounds
US9867836B2 (en) 2014-03-13 2018-01-16 Brigham Young University Lavage and/or infusion using CSA compounds for increasing fertility in a mammal
US10220045B2 (en) 2014-03-13 2019-03-05 Brigham Young University Compositions and methods for forming stabilized compositions with reduced CSA agglomeration
US9931350B2 (en) 2014-03-14 2018-04-03 Brigham Young University Anti-infective and osteogenic compositions and methods of use
US9686966B2 (en) 2014-04-30 2017-06-27 Brigham Young University Methods and apparatus for cleaning or disinfecting a water delivery system
US10441595B2 (en) 2014-06-26 2019-10-15 Brigham Young University Methods for treating fungal infections
US10238665B2 (en) 2014-06-26 2019-03-26 Brigham Young University Methods for treating fungal infections
US10227376B2 (en) 2014-08-22 2019-03-12 Brigham Young University Radiolabeled cationic steroid antimicrobials and diagnostic methods
US10155788B2 (en) 2014-10-07 2018-12-18 Brigham Young University Cationic steroidal antimicrobial prodrug compositions and uses thereof
LT3209647T (lt) * 2014-10-21 2020-09-25 Ariad Pharmaceuticals, Inc. Kristalinės 5-chlor-n4-[-2-(dimetilfosforil)fenil]-n2-{2-metoksi-4-[4-(4-metilpiperazin-1-il) piperidin-1-il]pirimidin-2,4-diamino formos
US9527883B2 (en) 2015-04-22 2016-12-27 Brigham Young University Methods for the synthesis of ceragenins
WO2016172543A1 (en) 2015-04-22 2016-10-27 Savage Paul B Methods for the synthesis of ceragenins
KR101753842B1 (ko) * 2015-05-12 2017-07-04 한국화학연구원 불화퀴놀론계 항생제를 담지한 서방형 제제 및 이의 제조방법
US9434759B1 (en) 2015-05-18 2016-09-06 Brigham Young University Cationic steroidal antimicrobial compounds and methods of manufacturing such compounds
CN106543203B (zh) * 2015-09-18 2019-07-02 瑞普(天津)生物药业有限公司 一种长效头孢噻呋自由酸晶体的制备方法
ES2834049T3 (es) * 2016-01-22 2021-06-16 Sandoz Ag Bisclorhidrato de eravaciclina cristalino
US10226550B2 (en) 2016-03-11 2019-03-12 Brigham Young University Cationic steroidal antimicrobial compositions for the treatment of dermal tissue
KR101898282B1 (ko) * 2016-05-24 2018-09-13 주식회사 고려비엔피 항생제의 서방형 수의학적 조성물 및 이의 제조방법
JP2019524710A (ja) * 2016-07-07 2019-09-05 アイアンウッド ファーマシューティカルズ インコーポレイテッド Sgc刺激剤の固体形態
US10959433B2 (en) 2017-03-21 2021-03-30 Brigham Young University Use of cationic steroidal antimicrobials for sporicidal activity
US11186556B1 (en) * 2018-10-16 2021-11-30 Celgene Corporation Salts of a thiazolidinone compound, solid forms, compositions and methods of use thereof
UA119735C2 (uk) 2018-12-20 2019-07-25 Анатолій Семенович Редер Фармацевтична сполука, спосіб її отримання та застосування як лікарського засобу
US12186328B2 (en) 2019-05-23 2025-01-07 Brigham Young University Use of CSA compounds to stimulate stem cells and hair growth
TW202233625A (zh) * 2020-11-18 2022-09-01 美商傳達治療有限公司 Fgfr抑制劑及其製造及使用方法
CN117229296A (zh) * 2023-09-14 2023-12-15 广东温氏大华农生物科技有限公司 一种头孢噻呋酸晶体及其制备方法与应用

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Also Published As

Publication number Publication date
FR05C0045I2 (enExample) 2007-08-03
CA2155322C (en) 2000-02-29
HU222244B1 (hu) 2003-05-28
WO1994020505A1 (en) 1994-09-15
NO2005025I2 (no) 2010-11-22
ATE202109T1 (de) 2001-06-15
SK111495A3 (en) 1995-12-06
CN1055090C (zh) 2000-08-02
NO953564L (no) 1995-11-07
FI120307B (fi) 2009-09-15
LU91206I2 (fr) 2006-05-30
JPH08507519A (ja) 1996-08-13
DE122005000055I1 (de) 2006-02-23
IL108910A (en) 1999-10-28
ZA941586B (en) 1995-09-07
CZ9502290A3 (cs) 2001-08-15
FI954250A0 (fi) 1995-09-11
SI0690864T1 (en) 2001-10-31
BR1101034A (pt) 2002-04-30
JP3852946B2 (ja) 2006-12-06
PL184611B1 (pl) 2002-11-29
DK0690864T3 (da) 2001-09-17
NO2005025I1 (no) 2005-12-05
KR100296810B1 (ko) 2001-10-24
US5721359A (en) 1998-02-24
NL300208I2 (nl) 2006-05-01
CA2155322A1 (en) 1994-09-15
DE122005000055I2 (de) 2008-06-05
AU694419B2 (en) 1998-07-23
SK283674B6 (sk) 2003-11-04
IL108910A0 (en) 1994-06-24
HUT73781A (en) 1996-09-30
CZ289332B6 (cs) 2002-01-16
NZ263002A (en) 1996-12-20
CN1119016A (zh) 1996-03-20
ES2157254T3 (es) 2001-08-16
FI954250L (fi) 1995-09-11
NO953564D0 (no) 1995-09-11
DE69427469T2 (de) 2001-10-31
TW267170B (enExample) 1996-01-01
AU6351094A (en) 1994-09-26
LV12889B (lv) 2002-12-20
NO313199B1 (no) 2002-08-26
NL300208I1 (nl) 2006-02-01
DE69427469D1 (en) 2001-07-19
HU9501960D0 (en) 1995-09-28
PT690864E (pt) 2001-11-30
RU2136685C1 (ru) 1999-09-10
PL310556A1 (en) 1995-12-27
GR3036514T3 (en) 2001-12-31
EP0690864A1 (en) 1996-01-10
EP0690864B1 (en) 2001-06-13

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