ES2906078T3 - Moduladores del canal de potasio - Google Patents

Moduladores del canal de potasio Download PDF

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Publication number
ES2906078T3
ES2906078T3 ES18704122T ES18704122T ES2906078T3 ES 2906078 T3 ES2906078 T3 ES 2906078T3 ES 18704122 T ES18704122 T ES 18704122T ES 18704122 T ES18704122 T ES 18704122T ES 2906078 T3 ES2906078 T3 ES 2906078T3
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ES
Spain
Prior art keywords
compound
disease
mmol
composition
pharmaceutically acceptable
Prior art date
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Active
Application number
ES18704122T
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English (en)
Spanish (es)
Inventor
Dipak Amrutkar
Kelly Foster
Thomas Jacobsen
Martin JEFSON
Gregg Keaney
Janus Larsen
Karin Nielsen
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Cadent Therapeutics Inc
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Cadent Therapeutics Inc
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5355Non-condensed oxazines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Addiction (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Surface Acoustic Wave Elements And Circuit Networks Thereof (AREA)
ES18704122T 2017-01-23 2018-01-23 Moduladores del canal de potasio Active ES2906078T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201762449270P 2017-01-23 2017-01-23
PCT/US2018/014792 WO2018136917A1 (en) 2017-01-23 2018-01-23 Potassium channel modulators

Publications (1)

Publication Number Publication Date
ES2906078T3 true ES2906078T3 (es) 2022-04-13

Family

ID=61188924

Family Applications (1)

Application Number Title Priority Date Filing Date
ES18704122T Active ES2906078T3 (es) 2017-01-23 2018-01-23 Moduladores del canal de potasio

Country Status (30)

Country Link
US (4) US9975886B1 (enExample)
EP (1) EP3571193B1 (enExample)
JP (1) JP6997197B2 (enExample)
KR (1) KR102664772B1 (enExample)
CN (1) CN110198935B (enExample)
AR (1) AR110770A1 (enExample)
BR (1) BR112019014814B1 (enExample)
CL (1) CL2019002031A1 (enExample)
CO (1) CO2019009060A2 (enExample)
CU (1) CU24560B1 (enExample)
CY (1) CY1125463T1 (enExample)
DK (1) DK3571193T3 (enExample)
EA (1) EA036668B1 (enExample)
ES (1) ES2906078T3 (enExample)
HR (1) HRP20220079T1 (enExample)
HU (1) HUE057710T2 (enExample)
IL (1) IL267954B (enExample)
LT (1) LT3571193T (enExample)
MX (1) MX376080B (enExample)
MY (1) MY195123A (enExample)
PH (1) PH12019501678A1 (enExample)
PL (1) PL3571193T3 (enExample)
PT (1) PT3571193T (enExample)
RS (1) RS62899B1 (enExample)
SG (1) SG11201905893WA (enExample)
SI (1) SI3571193T1 (enExample)
TW (1) TWI751271B (enExample)
UA (1) UA123810C2 (enExample)
WO (1) WO2018136917A1 (enExample)
ZA (1) ZA201904458B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2017275657B2 (en) * 2016-06-02 2021-08-19 Novartis Ag Potassium channel modulators
EP3571193B1 (en) * 2017-01-23 2021-12-01 Cadent Therapeutics, Inc. Potassium channel modulators
EP3870291A1 (en) 2018-10-22 2021-09-01 Cadent Therapeutics, Inc. Crystalline forms of potassium channel modulators
CN118985622B (zh) * 2024-07-05 2025-12-02 云南大学 一种吡唑类化合物在防治植物根结线虫中的应用

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