CZ187995A3 - 2,6-diaminopurine derivatives, process of their preparation, their use for preparing pharmaceutical preparations and and pharmaceutical composition containing thereof - Google Patents

2,6-diaminopurine derivatives, process of their preparation, their use for preparing pharmaceutical preparations and and pharmaceutical composition containing thereof Download PDF

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Publication number
CZ187995A3
CZ187995A3 CZ951879A CZ187995A CZ187995A3 CZ 187995 A3 CZ187995 A3 CZ 187995A3 CZ 951879 A CZ951879 A CZ 951879A CZ 187995 A CZ187995 A CZ 187995A CZ 187995 A3 CZ187995 A3 CZ 187995A3
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CZ
Czechia
Prior art keywords
amino
ethyl
diphenylethyl
deoxy
purin
Prior art date
Application number
CZ951879A
Other languages
Czech (cs)
English (en)
Inventor
Michael Gregson
Diana Sally Ayres
George Blanch Ewan
Frank Ellis
John Knight
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of CZ187995A3 publication Critical patent/CZ187995A3/cs

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • C07H19/167—Purine radicals with ribosyl as the saccharide radical

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Immunology (AREA)
  • Biotechnology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Transplantation (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
CZ951879A 1993-01-20 1994-01-18 2,6-diaminopurine derivatives, process of their preparation, their use for preparing pharmaceutical preparations and and pharmaceutical composition containing thereof CZ187995A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB939301000A GB9301000D0 (en) 1993-01-20 1993-01-20 Chemical compounds

Publications (1)

Publication Number Publication Date
CZ187995A3 true CZ187995A3 (en) 1996-01-17

Family

ID=10728948

Family Applications (1)

Application Number Title Priority Date Filing Date
CZ951879A CZ187995A3 (en) 1993-01-20 1994-01-18 2,6-diaminopurine derivatives, process of their preparation, their use for preparing pharmaceutical preparations and and pharmaceutical composition containing thereof

Country Status (29)

Country Link
US (2) US5925624A (ref)
EP (1) EP0680488B1 (ref)
JP (1) JP3768232B2 (ref)
KR (1) KR960700261A (ref)
CN (1) CN1043997C (ref)
AP (1) AP457A (ref)
AT (1) ATE164849T1 (ref)
AU (1) AU679714B2 (ref)
CA (1) CA2153688A1 (ref)
CZ (1) CZ187995A3 (ref)
DE (1) DE69409503T2 (ref)
DK (1) DK0680488T3 (ref)
EC (1) ECSP941104A (ref)
ES (1) ES2117249T3 (ref)
FI (1) FI953489L (ref)
GB (1) GB9301000D0 (ref)
HU (1) HU211914A9 (ref)
IL (1) IL108372A (ref)
IS (1) IS4121A (ref)
NO (1) NO305603B1 (ref)
NZ (1) NZ259880A (ref)
PE (1) PE54194A1 (ref)
PL (1) PL309975A1 (ref)
RU (1) RU2129561C1 (ref)
SI (1) SI9400021A (ref)
SK (1) SK281229B6 (ref)
TW (1) TW267168B (ref)
WO (1) WO1994017090A1 (ref)
ZA (1) ZA94335B (ref)

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JPH08505864A (ja) 1996-06-25
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CA2153688A1 (en) 1994-08-04
SK91895A3 (en) 1996-04-03
NO305603B1 (no) 1999-06-28
AP457A (en) 1996-02-01
FI953489A0 (fi) 1995-07-19
SI9400021A (en) 1994-09-30
ZA94335B (en) 1994-10-24
DE69409503D1 (de) 1998-05-14
FI953489A7 (fi) 1995-09-13
AP9400613A0 (en) 1994-01-31
PL309975A1 (en) 1995-11-13
NO952872L (no) 1995-09-13
SK281229B6 (sk) 2001-01-18
IL108372A0 (en) 1994-04-12
US5889178A (en) 1999-03-30
ATE164849T1 (de) 1998-04-15
AU679714B2 (en) 1997-07-10
RU2129561C1 (ru) 1999-04-27
TW267168B (ref) 1996-01-01
DE69409503T2 (de) 1998-08-06
DK0680488T3 (da) 1999-01-25
NO952872D0 (no) 1995-07-19
ES2117249T3 (es) 1998-08-01
HU211914A9 (en) 1996-01-29
WO1994017090A1 (en) 1994-08-04
CN1043997C (zh) 1999-07-07
EP0680488A1 (en) 1995-11-08
FI953489L (fi) 1995-09-13
US5925624A (en) 1999-07-20
AU5885194A (en) 1994-08-15
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KR960700261A (ko) 1996-01-19
EP0680488B1 (en) 1998-04-08
CN1119440A (zh) 1996-03-27
PE54194A1 (es) 1995-01-06

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