CN1767819B - 包含s1p受体激动剂和糖醇的固体药物组合物 - Google Patents

包含s1p受体激动剂和糖醇的固体药物组合物 Download PDF

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Publication number
CN1767819B
CN1767819B CN2004800092370A CN200480009237A CN1767819B CN 1767819 B CN1767819 B CN 1767819B CN 2004800092370 A CN2004800092370 A CN 2004800092370A CN 200480009237 A CN200480009237 A CN 200480009237A CN 1767819 B CN1767819 B CN 1767819B
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China
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composition
mannitol
alkyl
receptor agonist
weight
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Expired - Lifetime
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Chinese (zh)
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CN1767819A (zh
Inventor
大村朋幸
M·普迪派迪
A·E·罗伊斯
C·吕埃格尔
佐佐木正喜
田村德裕
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Novartis AG
Mitsubishi Tanabe Pharma Corp
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Novartis AG
Mitsubishi Pharma Corp
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    • A61K31/13—Amines
    • A61K31/145—Amines having sulfur, e.g. thiurams (>N—C(S)—S—C(S)—N< and >N—C(S)—S—S—C(S)—N<), Sulfinylamines (—N=SO), Sulfonylamines (—N=SO2)
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Oil, Petroleum & Natural Gas (AREA)
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  • Physiology (AREA)
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  • Hospice & Palliative Care (AREA)
  • Transplantation (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Virology (AREA)
  • Surgery (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
CN2004800092370A 2003-04-08 2004-04-06 包含s1p受体激动剂和糖醇的固体药物组合物 Expired - Lifetime CN1767819B (zh)

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US46121503P 2003-04-08 2003-04-08
US60/461,215 2003-04-08
PCT/EP2004/003656 WO2004089341A1 (en) 2003-04-08 2004-04-06 Organic compounds

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CN1767819A CN1767819A (zh) 2006-05-03
CN1767819B true CN1767819B (zh) 2010-07-28

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CN2010101213007A Expired - Lifetime CN101797241B (zh) 2003-04-08 2004-04-06 包含s1p受体激动剂和糖醇的固体药物组合物

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