CN1094757C - 用于治疗疼痛的异丁基γ－氨基丁酸及其衍生物 - Google Patents

用于治疗疼痛的异丁基γ－氨基丁酸及其衍生物 Download PDF

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Publication number
CN1094757C
CN1094757C CN97196041A CN97196041A CN1094757C CN 1094757 C CN1094757 C CN 1094757C CN 97196041 A CN97196041 A CN 97196041A CN 97196041 A CN97196041 A CN 97196041A CN 1094757 C CN1094757 C CN 1094757C
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pain
use according
treated
gabapentin
isobutyl
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Expired - Lifetime
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CN97196041A
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Chinese (zh)
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CN1223574A (zh
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L·辛格
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Warner Lambert Co LLC
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Warner Lambert Co LLC
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Anesthesiology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
CN97196041A 1996-07-24 1997-07-16 用于治疗疼痛的异丁基γ－氨基丁酸及其衍生物 Expired - Lifetime CN1094757C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2233796P 1996-07-24 1996-07-24
US60/022,337 1996-07-24

Publications (2)

Publication Number Publication Date
CN1223574A CN1223574A (zh) 1999-07-21
CN1094757C true CN1094757C (zh) 2002-11-27

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CN97196041A Expired - Lifetime CN1094757C (zh) 1996-07-24 1997-07-16 用于治疗疼痛的异丁基γ－氨基丁酸及其衍生物

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US (2) US6001876A (cg-RX-API-DMAC7.html)
EP (1) EP0934061B3 (cg-RX-API-DMAC7.html)
JP (1) JP3693258B2 (cg-RX-API-DMAC7.html)
KR (1) KR100491282B1 (cg-RX-API-DMAC7.html)
CN (1) CN1094757C (cg-RX-API-DMAC7.html)
AT (1) ATE241351T1 (cg-RX-API-DMAC7.html)
AU (1) AU714980B2 (cg-RX-API-DMAC7.html)
BR (1) BR9710536A (cg-RX-API-DMAC7.html)
CU (1) CU22850A3 (cg-RX-API-DMAC7.html)
DE (1) DE69722426T3 (cg-RX-API-DMAC7.html)
DK (1) DK0934061T6 (cg-RX-API-DMAC7.html)
ES (1) ES2200184T7 (cg-RX-API-DMAC7.html)
HR (1) HRP970387A2 (cg-RX-API-DMAC7.html)
HU (2) HU228426B1 (cg-RX-API-DMAC7.html)
IL (1) IL126999A (cg-RX-API-DMAC7.html)
NO (2) NO325822B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ332762A (cg-RX-API-DMAC7.html)
PL (1) PL189872B1 (cg-RX-API-DMAC7.html)
PT (1) PT934061E (cg-RX-API-DMAC7.html)
SI (1) SI0934061T1 (cg-RX-API-DMAC7.html)
WO (1) WO1998003167A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA976562B (cg-RX-API-DMAC7.html)

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