CN101657436A - 大环生长素释放肽受体调节剂及其使用方法 - Google Patents

大环生长素释放肽受体调节剂及其使用方法 Download PDF

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CN101657436A
CN101657436A CN200880010587A CN200880010587A CN101657436A CN 101657436 A CN101657436 A CN 101657436A CN 200880010587 A CN200880010587 A CN 200880010587A CN 200880010587 A CN200880010587 A CN 200880010587A CN 101657436 A CN101657436 A CN 101657436A
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forming
low alkyl
alkyl group
independently selected
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H·霍维达
G·弗拉泽
S·博歇明
M·布拉萨
D·德鲁茨
E·马索尔特
L·厄勒特
M·L·彼得森
Z·王
K·贝纳克利
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Tranzyme Pharma Inc
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CN200880010587A 2007-02-09 2008-02-08 大环生长素释放肽受体调节剂及其使用方法 Pending CN101657436A (zh)

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US88916307P 2007-02-09 2007-02-09
US60/889,163 2007-02-09
PCT/US2008/001754 WO2008130464A1 (en) 2007-02-09 2008-02-08 Macrocyclic ghrelin receptor modulators and methods of using the same

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Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102557989A (zh) * 2011-12-19 2012-07-11 深圳翰宇药业股份有限公司 优利莫瑞林中间体以及优利莫瑞林制备方法
CN109879935A (zh) * 2019-03-04 2019-06-14 南京工业大学 一种多肽的液相合成方法
CN115960080A (zh) * 2021-10-13 2023-04-14 南京知和医药科技有限公司 一种多环化合物及其作为胃饥饿素受体激动剂的用途

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7476653B2 (en) * 2003-06-18 2009-01-13 Tranzyme Pharma, Inc. Macrocyclic modulators of the ghrelin receptor
EP2210612B1 (en) * 2003-06-18 2016-10-05 Ocera Therapeutics, Inc. Macrocyclic antagonists of the motilin receptor
US20090198050A1 (en) * 2003-06-18 2009-08-06 Tranzyme Pharma Inc. Macrocyclic Modulators of the Ghrelin Receptor
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CN115960080B (zh) * 2021-10-13 2024-03-15 南京知和医药科技有限公司 一种多环化合物及其作为胃饥饿素受体激动剂的用途

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US10258602B2 (en) 2019-04-16
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EP2644618B1 (en) 2016-08-17
MX2009008574A (es) 2009-12-09
US20180228768A1 (en) 2018-08-16
CA2677399A1 (en) 2008-10-30
US9371297B2 (en) 2016-06-21
BRPI0807046A2 (pt) 2015-05-26
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JP2010518090A (ja) 2010-05-27
AU2008241532A1 (en) 2008-10-30
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ES2604943T3 (es) 2017-03-10
CA2677399C (en) 2016-09-13
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