BRPI0314344B8 - composto 2,3-diidro-6-nitroimidazo[2,1-b]oxazol, composição farmacêutica compreendendo o mesmo e método para produzir um composto - Google Patents

composto 2,3-diidro-6-nitroimidazo[2,1-b]oxazol, composição farmacêutica compreendendo o mesmo e método para produzir um composto

Info

Publication number
BRPI0314344B8
BRPI0314344B8 BRPI0314344A BR0314344A BRPI0314344B8 BR PI0314344 B8 BRPI0314344 B8 BR PI0314344B8 BR PI0314344 A BRPI0314344 A BR PI0314344A BR 0314344 A BR0314344 A BR 0314344A BR PI0314344 B8 BRPI0314344 B8 BR PI0314344B8
Authority
BR
Brazil
Prior art keywords
compound
nitroimidazo
dihydro
producing
pharmaceutical composition
Prior art date
Application number
BRPI0314344A
Other languages
English (en)
Portuguese (pt)
Other versions
BR0314344A (pt
BRPI0314344B1 (pt
Inventor
Kuroda Hideaki
Tsubouchi Hidetsugu
Sasaki Hirofumi
Hashizume Hiroyuki
Tai Kuninori
Komatsu Makoto
Matsumoto Makoto
Kawasaki Masanori
Itotani Motohiro
Miyamura Shin
Matsuzaki Takayuki
Hasegawa Takeshi
Kuroda Takeshi
Sumida Takumi
Tomishige Tatsuo
Haraguchi Yoshikazu
Seike Yuji
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of BR0314344A publication Critical patent/BR0314344A/pt
Publication of BRPI0314344B1 publication Critical patent/BRPI0314344B1/pt
Publication of BRPI0314344B8 publication Critical patent/BRPI0314344B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/20—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
BRPI0314344A 2002-10-11 2003-10-10 composto 2,3-diidro-6-nitroimidazo[2,1-b]oxazol, composição farmacêutica compreendendo o mesmo e método para produzir um composto BRPI0314344B8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002298259 2002-10-11
PCT/JP2003/013070 WO2004033463A1 (ja) 2002-10-11 2003-10-10 ２，３−ジヒドロ−６−ニトロイミダゾ[２，１−ｂ]オキサゾール化合物

Publications (3)

Publication Number Publication Date
BR0314344A BR0314344A (pt) 2005-07-12
BRPI0314344B1 BRPI0314344B1 (pt) 2019-11-26
BRPI0314344B8 true BRPI0314344B8 (pt) 2021-05-25

Family

ID=32089299

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0314344A BRPI0314344B8 (pt) 2002-10-11 2003-10-10 composto 2,3-diidro-6-nitroimidazo[2,1-b]oxazol, composição farmacêutica compreendendo o mesmo e método para produzir um composto

Country Status (26)

Country Link
US (1) US7262212B2 (enExample)
EP (2) EP2570418A3 (enExample)
JP (1) JP4186065B2 (enExample)
KR (1) KR100723847B1 (enExample)
CN (4) CN102532162B (enExample)
AR (4) AR041198A1 (enExample)
AU (1) AU2003272979B2 (enExample)
BE (1) BE2014C053I2 (enExample)
BR (1) BRPI0314344B8 (enExample)
CA (1) CA2497569C (enExample)
CY (2) CY1113578T1 (enExample)
DK (1) DK1555267T3 (enExample)
ES (1) ES2400179T3 (enExample)
FR (1) FR14C0066I2 (enExample)
HU (1) HUS1400046I1 (enExample)
LU (1) LU92517I2 (enExample)
MX (1) MXPA05003674A (enExample)
MY (1) MY139244A (enExample)
PL (3) PL217919B1 (enExample)
PT (1) PT1555267E (enExample)
RU (1) RU2326121C3 (enExample)
SI (1) SI1555267T1 (enExample)
TW (1) TWI347946B (enExample)
UA (1) UA83200C2 (enExample)
WO (1) WO2004033463A1 (enExample)
ZA (1) ZA200501033B (enExample)

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CN110483549B (zh) * 2019-08-30 2021-03-05 沈阳药科大学 一种硝基咪唑吡喃类抗结核药物的制备方法
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CN116640106B (zh) * 2023-05-11 2024-03-08 郑州大学 一种苯基哌嗪类化合物及其制备方法、应用
CN119059990B (zh) * 2024-11-01 2025-02-07 安徽昊帆生物有限公司 1-氨基甲酸叔丁酯哌嗪的制备方法

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BE2014C053I2 (enExample) 2022-08-30
RU2005114017A (ru) 2006-01-20
PT1555267E (pt) 2013-01-29
WO2004033463A1 (ja) 2004-04-22
KR100723847B1 (ko) 2007-05-31
JP4186065B2 (ja) 2008-11-26
AU2003272979B2 (en) 2009-07-23
HK1171018A1 (en) 2013-03-15
RU2326121C2 (ru) 2008-06-10
EP2570418A3 (en) 2013-07-03
US20060094767A1 (en) 2006-05-04
AR089950A2 (es) 2014-10-01
ES2400179T3 (es) 2013-04-08
BR0314344A (pt) 2005-07-12
AR086485A2 (es) 2013-12-18
CN101255170A (zh) 2008-09-03
PL217919B1 (pl) 2014-09-30
AR041198A1 (es) 2005-05-04
EP1555267B1 (en) 2013-01-16
CY2014041I1 (el) 2016-07-27
HK1085463A1 (zh) 2006-08-25
DK1555267T3 (da) 2013-02-11
PL409525A1 (pl) 2014-11-10
CN100366624C (zh) 2008-02-06
US7262212B2 (en) 2007-08-28
TW200420568A (en) 2004-10-16
EP2570418A2 (en) 2013-03-20
ZA200501033B (en) 2006-06-28
CN102532162A (zh) 2012-07-04
PL404913A1 (pl) 2013-09-30
HUS1400046I1 (hu) 2017-04-28
CA2497569A1 (en) 2004-04-22
AR091771A2 (es) 2015-02-25
BRPI0314344B1 (pt) 2019-11-26
CN1705670A (zh) 2005-12-07
SI1555267T1 (sl) 2013-05-31
CN101172981A (zh) 2008-05-07
EP1555267A4 (en) 2010-08-18
CY1113578T1 (el) 2016-06-22
FR14C0066I1 (enExample) 2014-10-17
CY2014041I2 (el) 2016-07-27
JP2004149527A (ja) 2004-05-27
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CA2497569C (en) 2011-05-24
AU2003272979A1 (en) 2004-05-04
CN102532162B (zh) 2015-05-27
MY139244A (en) 2009-09-30
FR14C0066I2 (fr) 2015-05-22
UA83200C2 (en) 2008-06-25
MXPA05003674A (es) 2005-06-08
RU2326121C3 (ru) 2021-09-17
TWI347946B (en) 2011-09-01
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LU92517I2 (fr) 2014-10-13

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