BE2014C053I2 - - Google Patents

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Publication number
BE2014C053I2
BE2014C053I2 BE2014C053C BE2014C053C BE2014C053I2 BE 2014C053 I2 BE2014C053 I2 BE 2014C053I2 BE 2014C053 C BE2014C053 C BE 2014C053C BE 2014C053 C BE2014C053 C BE 2014C053C BE 2014C053 I2 BE2014C053 I2 BE 2014C053I2
Authority
BE
Belgium
Application number
BE2014C053C
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of BE2014C053I2 publication Critical patent/BE2014C053I2/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/20—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
BE2014C053C 2002-10-11 2014-09-09 BE2014C053I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002298259 2002-10-11
PCT/JP2003/013070 WO2004033463A1 (fr) 2002-10-11 2003-10-10 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles

Publications (1)

Publication Number Publication Date
BE2014C053I2 true BE2014C053I2 (fr) 2022-08-30

Family

ID=32089299

Family Applications (1)

Application Number Title Priority Date Filing Date
BE2014C053C BE2014C053I2 (fr) 2002-10-11 2014-09-09

Country Status (27)

Country Link
US (1) US7262212B2 (fr)
EP (2) EP2570418A3 (fr)
JP (1) JP4186065B2 (fr)
KR (1) KR100723847B1 (fr)
CN (4) CN101255170A (fr)
AR (4) AR041198A1 (fr)
AU (1) AU2003272979B2 (fr)
BE (1) BE2014C053I2 (fr)
BR (1) BRPI0314344B8 (fr)
CA (1) CA2497569C (fr)
CY (2) CY1113578T1 (fr)
DK (1) DK1555267T3 (fr)
ES (1) ES2400179T3 (fr)
FR (1) FR14C0066I2 (fr)
HK (2) HK1085463A1 (fr)
HU (1) HUS1400046I1 (fr)
LU (1) LU92517I2 (fr)
MX (1) MXPA05003674A (fr)
MY (1) MY139244A (fr)
PL (3) PL404913A1 (fr)
PT (1) PT1555267E (fr)
RU (1) RU2326121C3 (fr)
SI (1) SI1555267T1 (fr)
TW (1) TWI347946B (fr)
UA (1) UA83200C2 (fr)
WO (1) WO2004033463A1 (fr)
ZA (1) ZA200501033B (fr)

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PL1678185T3 (pl) 2003-10-31 2009-04-30 Otsuka Pharma Co Ltd Związki 2,3-dihydro-6-nitroimidazo[2,1-B]oksazolu do leczenia gruźlicy
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US7408066B2 (en) * 2005-06-20 2008-08-05 Schering Corproation Carbon-linked substituted piperidines and derivatives thereof useful as histamine H3 antagonists
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JP5105818B2 (ja) * 2005-10-05 2012-12-26 大塚製薬株式会社 医薬組成物
TW201233389A (en) * 2005-10-05 2012-08-16 Otsuka Pharma Co Ltd Antituberculous therapeutic drugs and kit containing the same
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EP1968961A2 (fr) 2005-12-21 2008-09-17 Decode Genetics EHF Inhibiteurs de biaryl-azote-heterocycle de lta4h pour traiter l'inflammation
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AR070301A1 (es) 2007-05-08 2010-03-31 Otsuka Pharma Co Ltd Compuesto epoxi y metodo para producir el mismo
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EP2205585A1 (fr) * 2007-10-16 2010-07-14 Glaxo Group Limited Dérivés de quinoléine utilisés pour traiter des maladies inflammatoires et allergiques
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CA2708303A1 (fr) 2007-12-11 2009-06-18 Vitae Pharmaceuticals, Inc. Inhibiteurs cycliques d'uree de la 11.beta.-hydroxysteroide dehydrogenase 1
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US9540322B2 (en) 2008-08-18 2017-01-10 Yale University MIF modulators
WO2010143007A1 (fr) * 2009-06-10 2010-12-16 Dynamit Nobel Gmbh Explosivstoff-Und Systemtechnik Procédé de production de 2-halogéno-4-nitroimidazole
US8558005B2 (en) 2008-08-21 2013-10-15 Dynamit Nobel Gmbh Explosivstoff-Und Systemtechnik Methods for the production of 2-halo-4-nitroimidazole and intermediates thereof
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CN103524492A (zh) * 2013-10-23 2014-01-22 中国药科大学 侧链含硝基咪唑基团取代的喹诺酮类化合物、其制备及用途
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CN105732659B (zh) * 2014-12-12 2019-07-16 上海阳帆医药科技有限公司 硝基咪唑类化合物及其制备方法和在制药中的用途
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CN106317072B (zh) * 2015-06-17 2020-03-17 盟科医药技术(上海)有限公司 用于分枝杆菌感染治疗的杂环化合物及其应用
WO2017146246A1 (fr) 2016-02-26 2017-08-31 大塚製薬株式会社 Dérivé de pipéridine
CN105859628B (zh) * 2016-04-19 2018-08-07 清远职业技术学院 一种抗菌化合物对n咪唑苯甲醛缩邻甲苯胺希夫碱及其制备方法和应用
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MX2020001808A (es) * 2017-08-16 2022-07-19 Glaxosmithkline Ip Dev Ltd Nuevos compuestos.
CN112236141A (zh) 2018-06-11 2021-01-15 大塚制药株式会社 包含德拉马尼的组合物
CN109705022A (zh) * 2018-12-28 2019-05-03 上海彩迩文生化科技有限公司 一种芳香胺中间体的制备方法
CN112300192B (zh) * 2019-08-02 2023-08-11 南京长澳医药科技有限公司 硝基咪唑类化合物及其制备方法和用途
CN110483549B (zh) * 2019-08-30 2021-03-05 沈阳药科大学 一种硝基咪唑吡喃类抗结核药物的制备方法
CN110615800A (zh) * 2019-10-16 2019-12-27 李丽丽 硝基咪唑类化合物及其制备方法和用途
CN112156088B (zh) * 2020-10-30 2021-08-31 健民药业集团股份有限公司 一种化合物在制备结核分枝杆菌抑制剂中的用途
CN113603706A (zh) * 2021-08-04 2021-11-05 深圳市泰力生物医药有限公司 德拉马尼的晶型、含有该晶型的活性药物和药物组合物
CN115368252B (zh) * 2022-09-19 2024-01-12 西北农林科技大学 一种4-胺基酚类衍生物及应用
CN116640106B (zh) * 2023-05-11 2024-03-08 郑州大学 一种苯基哌嗪类化合物及其制备方法、应用

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Also Published As

Publication number Publication date
AU2003272979B2 (en) 2009-07-23
EP1555267A4 (fr) 2010-08-18
CY2014041I1 (el) 2016-07-27
CY1113578T1 (el) 2016-06-22
DK1555267T3 (da) 2013-02-11
EP1555267B1 (fr) 2013-01-16
AR089950A2 (es) 2014-10-01
FR14C0066I1 (fr) 2014-10-17
HK1085463A1 (en) 2006-08-25
TWI347946B (en) 2011-09-01
KR100723847B1 (ko) 2007-05-31
PL376157A1 (en) 2005-12-27
PL409525A1 (pl) 2014-11-10
CY2014041I2 (el) 2016-07-27
US20060094767A1 (en) 2006-05-04
US7262212B2 (en) 2007-08-28
CA2497569A1 (fr) 2004-04-22
AR041198A1 (es) 2005-05-04
BRPI0314344B1 (pt) 2019-11-26
MY139244A (en) 2009-09-30
FR14C0066I2 (fr) 2015-05-22
AU2003272979A1 (en) 2004-05-04
UA83200C2 (en) 2008-06-25
TW200420568A (en) 2004-10-16
SI1555267T1 (sl) 2013-05-31
LU92517I2 (fr) 2014-10-13
CN1705670A (zh) 2005-12-07
PL404913A1 (pl) 2013-09-30
BR0314344A (pt) 2005-07-12
CN101172981A (zh) 2008-05-07
AR091771A2 (es) 2015-02-25
RU2326121C3 (ru) 2021-09-17
AR086485A2 (es) 2013-12-18
CN102532162B (zh) 2015-05-27
JP2004149527A (ja) 2004-05-27
HK1171018A1 (en) 2013-03-15
CN102532162A (zh) 2012-07-04
CN101255170A (zh) 2008-09-03
EP2570418A2 (fr) 2013-03-20
WO2004033463A1 (fr) 2004-04-22
KR20050061473A (ko) 2005-06-22
ES2400179T3 (es) 2013-04-08
BRPI0314344B8 (pt) 2021-05-25
JP4186065B2 (ja) 2008-11-26
PT1555267E (pt) 2013-01-29
RU2005114017A (ru) 2006-01-20
EP1555267A1 (fr) 2005-07-20
EP2570418A3 (fr) 2013-07-03
HUS1400046I1 (hu) 2017-04-28
PL217919B1 (pl) 2014-09-30
CN100366624C (zh) 2008-02-06
RU2326121C2 (ru) 2008-06-10
ZA200501033B (en) 2006-06-28
CA2497569C (fr) 2011-05-24
MXPA05003674A (es) 2005-06-08

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