BR9714059A - S-omeprazol em uma forma neutra, processo para preparar o mesmo, uso deste, composição farmacêutica, e, processo para tratar uma condição relacionada com ácido gástrico. - Google Patents
S-omeprazol em uma forma neutra, processo para preparar o mesmo, uso deste, composição farmacêutica, e, processo para tratar uma condição relacionada com ácido gástrico.Info
- Publication number
- BR9714059A BR9714059A BR9714059-7A BR9714059A BR9714059A BR 9714059 A BR9714059 A BR 9714059A BR 9714059 A BR9714059 A BR 9714059A BR 9714059 A BR9714059 A BR 9714059A
- Authority
- BR
- Brazil
- Prior art keywords
- omeprazole
- treat
- prepare
- pharmaceutical composition
- neutral form
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
"S-OMEPRAZOL EM UMA FORMA NEUTRA, PROCESSO PARA PREPARAR O MESMO, USO DESTE, COMPOSIçãO FARMACêUTICA, E, PROCESSO PARA TRATAR UMA CONDIçãO RELACIONADA COM áCIDO GáSTRICO". A invenção fornece S-omeprazol em uma forma neutra, caracterizado em que está em um estado sólido, preferivelmente em um estado parcialmente cristalino ou substancialmente cristalino, tal como a forma A ou a forma B. Além disso, a invenção fornece processos para a preparação do S-omeptrazol e seu uso na medicina.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE9604793A SE510666C2 (sv) | 1996-12-20 | 1996-12-20 | Nya Kristallmodifikationer |
PCT/SE1997/002125 WO1998028294A1 (en) | 1996-12-20 | 1997-12-16 | A novel compound form |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9714059A true BR9714059A (pt) | 2000-05-09 |
Family
ID=20405146
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9714059-7A BR9714059A (pt) | 1996-12-20 | 1997-12-16 | S-omeprazol em uma forma neutra, processo para preparar o mesmo, uso deste, composição farmacêutica, e, processo para tratar uma condição relacionada com ácido gástrico. |
Country Status (37)
Country | Link |
---|---|
US (1) | US6162816A (pt) |
EP (1) | EP0946547B1 (pt) |
JP (1) | JP4402174B2 (pt) |
KR (1) | KR20000069595A (pt) |
CN (1) | CN1109684C (pt) |
AR (1) | AR010361A1 (pt) |
AT (1) | ATE236898T1 (pt) |
AU (1) | AU730129B2 (pt) |
BR (1) | BR9714059A (pt) |
CA (1) | CA2274076C (pt) |
CZ (1) | CZ294784B6 (pt) |
DE (1) | DE69720774T2 (pt) |
DK (1) | DK0946547T3 (pt) |
EE (1) | EE03923B1 (pt) |
EG (1) | EG24414A (pt) |
ES (1) | ES2194231T3 (pt) |
HK (1) | HK1022909A1 (pt) |
HU (1) | HU227589B1 (pt) |
ID (1) | ID21850A (pt) |
IL (1) | IL130450A0 (pt) |
IS (1) | IS1981B (pt) |
MY (1) | MY117032A (pt) |
NO (1) | NO317191B1 (pt) |
NZ (1) | NZ336024A (pt) |
PL (1) | PL190377B1 (pt) |
PT (1) | PT946547E (pt) |
RS (1) | RS49685B (pt) |
RU (1) | RU2184734C2 (pt) |
SA (1) | SA97180739B1 (pt) |
SE (1) | SE510666C2 (pt) |
SI (1) | SI0946547T1 (pt) |
SK (1) | SK285151B6 (pt) |
TR (1) | TR199901410T2 (pt) |
TW (1) | TW538039B (pt) |
UA (1) | UA55436C2 (pt) |
WO (1) | WO1998028294A1 (pt) |
ZA (1) | ZA9711046B (pt) |
Families Citing this family (60)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6645988B2 (en) | 1996-01-04 | 2003-11-11 | Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and method of using same |
US5840737A (en) | 1996-01-04 | 1998-11-24 | The Curators Of The University Of Missouri | Omeprazole solution and method for using same |
US6699885B2 (en) | 1996-01-04 | 2004-03-02 | The Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and methods of using same |
US6489346B1 (en) | 1996-01-04 | 2002-12-03 | The Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and method of using same |
SI20019A (sl) | 1998-07-13 | 2000-02-29 | LEK, tovarna farmacevtskih in kemi�nih izdelkov, d.d. | Izboljšan postopek sinteze 5-metoksi -2-/(4-metoksi-3,5-dimetil-2-piridil)metil/ sulfinil-1H-benzimidazola |
UA72748C2 (en) * | 1998-11-10 | 2005-04-15 | Astrazeneca Ab | A novel crystalline form of omeprazole |
IL142703A (en) | 1998-11-10 | 2006-04-10 | Astrazeneca Ab | Crystalline form of omeprazole |
JP3926936B2 (ja) * | 1998-11-16 | 2007-06-06 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | スルホキシド誘導体・アセトン錯体およびその製造法 |
SE9804003D0 (sv) * | 1998-11-23 | 1998-11-23 | Astra Ab | A method of producing drug particles |
SE9900274D0 (sv) * | 1999-01-28 | 1999-01-28 | Astra Ab | New compound |
JP2000344739A (ja) * | 1999-06-01 | 2000-12-12 | Sumitomo Chem Co Ltd | N−保護−アゼチジン−2−カルボン酸の製造方法 |
TWI289557B (en) | 1999-06-17 | 2007-11-11 | Takeda Chemical Industries Ltd | A crystal of a hydrate of (R)-2-[[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridyl]methyl]sulfinyl]-1H-benzimidazole |
SE0000774D0 (sv) * | 2000-03-08 | 2000-03-08 | Astrazeneca Ab | New formulation |
SE0000773D0 (sv) * | 2000-03-08 | 2000-03-08 | Astrazeneca Ab | New formulation |
KR101035534B1 (ko) | 2000-05-15 | 2011-05-23 | 다케다 야쿠힌 고교 가부시키가이샤 | 결정의 제조방법 |
GB0016040D0 (en) * | 2000-06-29 | 2000-08-23 | Glaxo Group Ltd | Novel process for preparing crystalline particles |
CA2417311C (en) | 2000-08-04 | 2012-07-10 | Takeda Chemical Industries, Ltd. | Crystalline alkali metal salts of lansoprazole and their production and use |
SI20875A (sl) * | 2001-04-25 | 2002-10-31 | LEK, tovarna farmacevtskih in kemi�nih izdelkov, d.d. | Kristalna oblika omeprazola |
DE60237087D1 (de) | 2001-06-01 | 2010-09-02 | Pozen Inc | Pharmazeutische zusammensetzungen für die koordinierte abgabe von nsaid |
US8206741B2 (en) | 2001-06-01 | 2012-06-26 | Pozen Inc. | Pharmaceutical compositions for the coordinated delivery of NSAIDs |
GB2376231A (en) | 2001-06-06 | 2002-12-11 | Cipla Ltd | Benzimidazole-cyclodextrin inclusion complex |
SE0102993D0 (sv) | 2001-09-07 | 2001-09-07 | Astrazeneca Ab | New self emulsifying drug delivery system |
US7169793B2 (en) | 2002-06-27 | 2007-01-30 | Dr. Reddy's Laboratories Limited | Process for preparation of optically pure or optically enriched sulfoxide compounds, including amorphous esomeprazole and salts thereof |
ATE353887T1 (de) * | 2002-06-27 | 2007-03-15 | Reddys Lab Ltd Dr | Verfahren zur herstellung optisch reiner oder optisch angereicherter sulfoxidverbindungen einschliesslich amorphen esomeprazols und dessen salze |
CA2501424A1 (en) * | 2002-08-30 | 2004-03-11 | Dr. Reddy's Laboratories Limited | Amorphous hydrates of esomeprazole magnesium and process for the preparation thereof |
US8697094B2 (en) | 2002-10-16 | 2014-04-15 | Takeda Pharmaceutical Company Limited | Stable solid preparations |
EP1556043A1 (en) * | 2002-10-22 | 2005-07-27 | Ranbaxy Laboratories, Ltd. | Amorphous form of esomeprazole salts |
US20040242642A1 (en) * | 2002-11-18 | 2004-12-02 | Dr. Reddy's Laboratories Limited | Crystalline esomeprazole compounds and process for the preparation thereof |
EP1606279A1 (en) * | 2003-02-28 | 2005-12-21 | Ranbaxy Laboratories, Ltd. | Polymorphs of s-omeprazole |
EP1607395B1 (en) * | 2003-03-24 | 2011-05-04 | Eisai R&D Management Co., Ltd. | Process for the preparation of amorphous rabeprazole sodium salt |
CN1842525A (zh) * | 2003-05-05 | 2006-10-04 | 兰贝克赛实验室有限公司 | 苯并咪唑衍生物的钡盐 |
US8993599B2 (en) | 2003-07-18 | 2015-03-31 | Santarus, Inc. | Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them |
SE0400410D0 (sv) * | 2004-02-20 | 2004-02-20 | Astrazeneca Ab | New compounds |
US8815916B2 (en) | 2004-05-25 | 2014-08-26 | Santarus, Inc. | Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them |
US8906940B2 (en) | 2004-05-25 | 2014-12-09 | Santarus, Inc. | Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them |
JP5563735B2 (ja) | 2004-06-16 | 2014-07-30 | タケダ ファーマシューティカルズ ユー.エス.エー. インコーポレイティド | Ppi多回剤形 |
CN1972928A (zh) * | 2004-06-24 | 2007-05-30 | 阿斯利康(瑞典)有限公司 | 制备用于制备依美拉唑钠盐的结晶修饰物的新方法 |
ES2246149B1 (es) * | 2004-07-02 | 2007-06-01 | Esteve Quimica, S.A. | Formas solidas de la sal magnesica de s-omeprazol y procedimientos para su preparacion. |
RU2007145207A (ru) * | 2005-05-06 | 2009-06-20 | Гленмарк Фармасьютикалз Лимитед (In) | Стронциваемая соль эзомепразола, способ ее получения и содержащее ее фармацевтические композиции |
JP2008545768A (ja) * | 2005-06-08 | 2008-12-18 | レツク・フアーマシユーテイカルズ・デー・デー | オメプラゾールナトリウムの結晶性溶媒和物 |
US7563812B2 (en) | 2005-06-15 | 2009-07-21 | Hetero Drugs Limited | Amorphous esomeprazole hydrate |
NL2000126C2 (nl) * | 2005-07-15 | 2008-01-29 | Solvay | Werkwijze voor de vervaardiging van eptifibatide. |
US20070043085A1 (en) * | 2005-08-19 | 2007-02-22 | Glenmark Pharmaceuticals Limited | Process for the preparation of amorphous form of neutral esomeprazole |
US7576219B2 (en) | 2005-10-26 | 2009-08-18 | Hanmi Pharm. Co., Ltd | Crystalline S-omeprazole strontium hydrate, method for preparing same, and pharmaceutical composition containing same |
US20090082572A1 (en) * | 2005-11-14 | 2009-03-26 | Hetero Drugs Limited | Process for amorphous esomeprazole |
AU2006323245B2 (en) | 2005-12-05 | 2011-03-03 | Astrazeneca Ab | New process for the preparation of esomeprazole non-salt form |
EP1801110A1 (en) | 2005-12-22 | 2007-06-27 | KRKA, tovarna zdravil, d.d., Novo mesto | Esomeprazole arginine salt |
CA2631459A1 (en) | 2005-12-28 | 2007-07-05 | Union Quimico Farmaceutica, S.A. | A process for the preparation of the (s)-enantiomer of omeprazole |
EP2000468A1 (en) * | 2007-05-09 | 2008-12-10 | Dr. Reddy's Laboratories Ltd. | Esomeprazole salts and processes for preparation thereof |
EP2195309A4 (en) * | 2007-10-08 | 2013-04-24 | Hetero Drugs Ltd | SALT POLYMORPHS OF THE ESOMEPRAZOLE |
EP2262790B1 (en) | 2008-03-10 | 2017-06-07 | Takeda Pharmaceutical Company Limited | Crystal of benzimidazole compound |
EP2143722A1 (en) | 2008-07-09 | 2010-01-13 | Lek Pharmaceuticals D.D. | Process for preparation of esomeprazole sodium of high chemical purity and new forms of esomeprazole sodium |
AU2009290712A1 (en) | 2008-09-09 | 2010-03-18 | Astrazeneca Ab | Method for delivering a pharmaceutical composition to patient in need thereof |
WO2010151216A1 (en) | 2009-06-25 | 2010-12-29 | Astrazeneca Ab | Method for treating a patient at risk for developing an nsaid-associated ulcer |
WO2011071982A2 (en) | 2009-12-08 | 2011-06-16 | Codexis, Inc. | Synthesis of prazole compounds |
DK2649187T3 (da) | 2010-12-08 | 2018-01-29 | Codexis Inc | Biokatalysatorer og fremgangsmåder til syntesen af armodafinil |
CA2860231A1 (en) | 2011-12-28 | 2013-07-04 | Pozen Inc. | Improved compositions and methods for delivery of omeprazole plus acetylsalicylic acid |
RU2501549C1 (ru) | 2012-08-30 | 2013-12-20 | Авва Девелопмент Лтд | Фармацевтическая композиция для лечения гастроэзофагеальной рефлюксной болезни |
CN107043367A (zh) * | 2017-05-26 | 2017-08-15 | 重庆莱美隆宇药业有限公司 | 一种中性s‑奥美拉唑的干燥工艺 |
WO2024075017A1 (en) | 2022-10-04 | 2024-04-11 | Zabirnyk Arsenii | Inhibition of aortic valve calcification |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE7804231L (sv) * | 1978-04-14 | 1979-10-15 | Haessle Ab | Magsyrasekretionsmedel |
SE8301182D0 (sv) * | 1983-03-04 | 1983-03-04 | Haessle Ab | Novel compounds |
GB2189698A (en) * | 1986-04-30 | 1987-11-04 | Haessle Ab | Coated omeprazole tablets |
DE4035455A1 (de) * | 1990-11-08 | 1992-05-14 | Byk Gulden Lomberg Chem Fab | Enantiomerentrennung |
SE9301830D0 (sv) * | 1993-05-28 | 1993-05-28 | Ab Astra | New compounds |
US5877192A (en) * | 1993-05-28 | 1999-03-02 | Astra Aktiebolag | Method for the treatment of gastric acid-related diseases and production of medication using (-) enantiomer of omeprazole |
SE9302396D0 (sv) * | 1993-07-09 | 1993-07-09 | Ab Astra | A novel compound form |
PT1078628E (pt) * | 1994-07-08 | 2009-01-27 | Astrazeneca Ab | Forma de dosagem em comprimidos com unidades múltiplas |
-
1996
- 1996-12-20 SE SE9604793A patent/SE510666C2/sv unknown
-
1997
- 1997-12-08 TW TW086118449A patent/TW538039B/zh not_active IP Right Cessation
- 1997-12-09 ZA ZA9711046A patent/ZA9711046B/xx unknown
- 1997-12-16 CZ CZ19992202A patent/CZ294784B6/cs not_active IP Right Cessation
- 1997-12-16 IL IL13045097A patent/IL130450A0/xx not_active IP Right Cessation
- 1997-12-16 JP JP52868598A patent/JP4402174B2/ja not_active Expired - Fee Related
- 1997-12-16 SI SI9730528T patent/SI0946547T1/xx unknown
- 1997-12-16 AU AU55026/98A patent/AU730129B2/en not_active Ceased
- 1997-12-16 NZ NZ336024A patent/NZ336024A/en not_active IP Right Cessation
- 1997-12-16 EP EP97951367A patent/EP0946547B1/en not_active Expired - Lifetime
- 1997-12-16 US US09/000,154 patent/US6162816A/en not_active Expired - Lifetime
- 1997-12-16 RU RU99116303/04A patent/RU2184734C2/ru not_active IP Right Cessation
- 1997-12-16 WO PCT/SE1997/002125 patent/WO1998028294A1/en not_active Application Discontinuation
- 1997-12-16 AT AT97951367T patent/ATE236898T1/de active
- 1997-12-16 CN CN97180849A patent/CN1109684C/zh not_active Expired - Fee Related
- 1997-12-16 RS YUP-281/99A patent/RS49685B/sr unknown
- 1997-12-16 AR ARP970105920A patent/AR010361A1/es active IP Right Grant
- 1997-12-16 TR TR1999/01410T patent/TR199901410T2/xx unknown
- 1997-12-16 CA CA002274076A patent/CA2274076C/en not_active Expired - Fee Related
- 1997-12-16 PL PL97334297A patent/PL190377B1/pl not_active IP Right Cessation
- 1997-12-16 ID IDW990483A patent/ID21850A/id unknown
- 1997-12-16 PT PT97951367T patent/PT946547E/pt unknown
- 1997-12-16 DE DE69720774T patent/DE69720774T2/de not_active Expired - Lifetime
- 1997-12-16 KR KR1019997005574A patent/KR20000069595A/ko active Search and Examination
- 1997-12-16 DK DK97951367T patent/DK0946547T3/da active
- 1997-12-16 ES ES97951367T patent/ES2194231T3/es not_active Expired - Lifetime
- 1997-12-16 BR BR9714059-7A patent/BR9714059A/pt not_active Application Discontinuation
- 1997-12-16 SK SK765-99A patent/SK285151B6/sk not_active IP Right Cessation
- 1997-12-16 EE EEP199900259A patent/EE03923B1/xx not_active IP Right Cessation
- 1997-12-16 UA UA99073869A patent/UA55436C2/uk unknown
- 1997-12-16 HU HU0001547A patent/HU227589B1/hu not_active IP Right Cessation
- 1997-12-19 MY MYPI97006176A patent/MY117032A/en unknown
- 1997-12-20 EG EG136097A patent/EG24414A/xx active
- 1997-12-27 SA SA97180739A patent/SA97180739B1/ar unknown
-
1999
- 1999-06-07 IS IS5070A patent/IS1981B/is unknown
- 1999-06-21 NO NO19993068A patent/NO317191B1/no not_active IP Right Cessation
-
2000
- 2000-03-31 HK HK00101986A patent/HK1022909A1/xx not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BR9714059A (pt) | S-omeprazol em uma forma neutra, processo para preparar o mesmo, uso deste, composição farmacêutica, e, processo para tratar uma condição relacionada com ácido gástrico. | |
BR9907270A (pt) | Composto, composição farmacêutica, uso de um composto, e, processos para tratamento ou profilaxia de doenças inflamatórias, por exemplo, asma ou copd, e para a preparação de um composto | |
BR9907886A (pt) | Composto, uso do mesmo, composição farmacêutica, e, processo de tratamento ou profilaxia de doenças inflamatórias, por exemplo asma ou copd. | |
BR9910066A (pt) | Composição farmacêutica fluida que permite a liberação controlada de pelo menos uma substância ativa, processo de fabricação de uma composição farmacêutica, e, utilização de uma composição | |
BR9911482A (pt) | Composto, composição farmacêutica, uso do composto, e, processos para o tratamento ou profilaxia de doenças inflamatórias, e para a preparação de um composto | |
BR9712314A (pt) | Método de uso de inibidores de ciclooxigenase-2 no tratamento e prevenção de neoplasia | |
BR0114321A (pt) | Composto, composição farmacêutica, uso de um composto, método de tratamento ou profilaxia de doenças inflamatórias, e, processo para preparar um composto | |
BRPI0113042B8 (pt) | composto da fórmula ou um seu solvato fisiologicamente aceitável, uso do mesmo, composição farmacêutica, formulação farmacêutica, método para o tratamento de um indivíduo humano ou animal com uma condição inflamatória e/ou alérgica, e, processo para preparar um composto ou um seu solvato | |
BR9911488A (pt) | Composto, uso do mesmo, composição farmacêutica, e, processos para tratamento ou de profilaxia de doenças inflamatórias, e para a preparação de um composto | |
BR0111328A (pt) | Composto, mistura, processos para a preparação e produção de um composto, composição farmacêutica, uso de um composto, e, método para o tratamento ou prevenção de complicações de trombose arterial em pacientes com doença de artéria coronária, cerebrovascular ou vascular periférica | |
BR9810592A (pt) | Composto, processos para preparar um composto, para tratar ou prevenir doenças do sistema endócrino e para a fabricação de um medicamento, composição farmacêutica, e, uso de um composto | |
BR9913945A (pt) | Composição farmacêutica para o tratamento de distúrbios agudos por meio de administração sublingual, e, processo para o tratamento de distúrbios agudos | |
ATE257386T1 (de) | Pharmazeutische zusammensetzungen enthaltend eine mischung von selbstvernetzter und nichtselbstvernetzter hyaluronsäure zur behandlung von arthropathien | |
BR0109729A (pt) | Uso de uma combinação de um agente anti-angiogênico e um agente anti-hipertensivo, kit para uso na produção de um efeito anti-angiogênico e/ou efeito redutor da permeabilidade vascular em um animal de sangue quente, e, método de tratamento de um estado doentio associado com a angiogênese | |
BG101118A (en) | Therapeutical compounds | |
BR9808812A (pt) | Composição compreendendo partìculas cristalinas, finamente divididas de budesonida | |
AR012671A1 (es) | Composiciones farmaceuticas para el tratamiento o profilaxis de la constipacion, los usos de dichas composiciones y los procesos para prepararlos | |
DE60120691D1 (de) | Zusammensetzungen zur verwendung bei der behandlung der osteoporose und/oder der entzündlichen gelenkerkrankungen | |
ATE201597T1 (de) | Verabreichung von riluzol zur behandlung von neuro-aids | |
BR9910329A (pt) | Composto, composição farmacêutica, processo para estimular a liberação do hormÈnio de crescimento da pituitária de um mamìfero, e, uso de um composto | |
KR870700599A (ko) | 카르복실산유도체, 그의 제조방법, 이화합물을 함유한 약제조성물 및 그의 용도 | |
ITMI931649A1 (it) | Derivati dell'acido 2-ammino-4-fenil-4-osso butirrico | |
BR9913464A (pt) | Composto, processos para a produção de um composto e para a conversão de uma forma cristalina de um composto, formulação farmacêutica, uso de um composto, e, processo para tratamento de uma condição onde a inibição da trombina é requerida ou desejada | |
BR0010808A (pt) | Composições farmacêuticas e usos | |
BR9909958A (pt) | Formulação farmacêutica, respectivos processo de preparação e uso e método de tratamento ou prevenção de distúrbios ósseos |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PRESENTE PEDIDO, UMA VEZ QUE A MATERIA REIVINDICADA CONTRARIA O DISPOSTO NOS ARTS. 8O, 13 E 25 E O RELATORIO DESCRITIVO NAO ATENDE AO DISPOSTO NO ART. 24 DA MESMA LEI |
|
B12B | Appeal against refusal [chapter 12.2 patent gazette] |