BG107624A - Бициклени пиролил амиди като гликоген фосфорилазни инхибитори - Google Patents

Бициклени пиролил амиди като гликоген фосфорилазни инхибитори Download PDF

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Publication number
BG107624A
BG107624A BG107624A BG10762403A BG107624A BG 107624 A BG107624 A BG 107624A BG 107624 A BG107624 A BG 107624A BG 10762403 A BG10762403 A BG 10762403A BG 107624 A BG107624 A BG 107624A
Authority
BG
Bulgaria
Prior art keywords
carbamoyl
pyrrole
thieno
dichloro
alkyl
Prior art date
Application number
BG107624A
Other languages
Bulgarian (bg)
English (en)
Inventor
Julie B. Bartlet
Sue Freeman
Peter Kenny
Andrew Morley
Raul Whittamore
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BG107624A publication Critical patent/BG107624A/bg

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BG107624A 2000-09-06 2003-03-10 Бициклени пиролил амиди като гликоген фосфорилазни инхибитори BG107624A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0021831.3A GB0021831D0 (en) 2000-09-06 2000-09-06 Chemical compounds
PCT/SE2001/001880 WO2002020530A1 (en) 2000-09-06 2001-08-31 Bicyclic pyrrolyl amides as glucogen phosphorylase inhibitors

Publications (1)

Publication Number Publication Date
BG107624A true BG107624A (bg) 2004-01-30

Family

ID=9898927

Family Applications (1)

Application Number Title Priority Date Filing Date
BG107624A BG107624A (bg) 2000-09-06 2003-03-10 Бициклени пиролил амиди като гликоген фосфорилазни инхибитори

Country Status (31)

Country Link
US (1) US20030232875A1 (xx)
EP (1) EP1317459B1 (xx)
JP (1) JP2004508376A (xx)
KR (1) KR100802369B1 (xx)
CN (2) CN1264846C (xx)
AT (1) ATE263772T1 (xx)
AU (2) AU8283301A (xx)
BG (1) BG107624A (xx)
BR (1) BR0113606A (xx)
CA (1) CA2417594A1 (xx)
CZ (1) CZ2003616A3 (xx)
DE (1) DE60102710T2 (xx)
DK (1) DK1317459T3 (xx)
EE (1) EE200300083A (xx)
ES (1) ES2217183T3 (xx)
GB (1) GB0021831D0 (xx)
HK (1) HK1055299A1 (xx)
HU (1) HUP0400784A3 (xx)
IL (1) IL154291A0 (xx)
IS (1) IS2110B (xx)
MX (1) MXPA03001512A (xx)
NO (1) NO20031024D0 (xx)
NZ (1) NZ524011A (xx)
PL (1) PL361024A1 (xx)
PT (1) PT1317459E (xx)
RU (1) RU2003104013A (xx)
SK (1) SK2592003A3 (xx)
TR (1) TR200401659T4 (xx)
UA (1) UA73781C2 (xx)
WO (1) WO2002020530A1 (xx)
ZA (1) ZA200301013B (xx)

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Also Published As

Publication number Publication date
IS6727A (is) 2003-02-24
DK1317459T3 (da) 2004-07-12
AU8283301A (en) 2002-03-22
PT1317459E (pt) 2004-08-31
CN1264846C (zh) 2006-07-19
CA2417594A1 (en) 2002-03-14
ATE263772T1 (de) 2004-04-15
HK1055299A1 (en) 2004-01-02
WO2002020530A1 (en) 2002-03-14
HUP0400784A2 (hu) 2004-07-28
DE60102710T2 (de) 2005-04-14
EP1317459A1 (en) 2003-06-11
CN1473163A (zh) 2004-02-04
TR200401659T4 (tr) 2004-09-21
JP2004508376A (ja) 2004-03-18
BR0113606A (pt) 2003-06-24
CN1896078A (zh) 2007-01-17
NO20031024L (no) 2003-03-05
EP1317459B1 (en) 2004-04-07
MXPA03001512A (es) 2003-06-09
IS2110B (is) 2006-05-15
HUP0400784A3 (en) 2007-09-28
KR20030025305A (ko) 2003-03-28
IL154291A0 (en) 2003-09-17
ZA200301013B (en) 2004-05-05
EE200300083A (et) 2004-12-15
DE60102710D1 (de) 2004-05-13
PL361024A1 (en) 2004-09-20
UA73781C2 (en) 2005-09-15
RU2003104013A (ru) 2004-08-20
GB0021831D0 (en) 2000-10-18
SK2592003A3 (en) 2003-08-05
NZ524011A (en) 2004-08-27
CZ2003616A3 (cs) 2003-05-14
KR100802369B1 (ko) 2008-02-14
AU2001282833B2 (en) 2006-07-06
US20030232875A1 (en) 2003-12-18
ES2217183T3 (es) 2004-11-01
NO20031024D0 (no) 2003-03-05

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